E-LIB Suche - Ergebnisse für: Pietruś, Wojciech

1

From NMR to AI: Designing a Novel Chemical Representation t..:

Leniak, Arkadiusz ; Pietruś, Wojciech ; Kurczab, Rafał
Journal of Chemical Information and Modeling. 64 (2024) 8 - p. 3302-3321 , 2024

Link: https://doi.org/10.1021/..

2

5-HT6 receptor neutral antagonists protect astrocytes: A le..:

Drop, Marcin ; Koczurkiewicz-Adamczyk, Paulina ; Bento, Ophélie...
European Journal of Medicinal Chemistry. 275 (2024) - p. 116615 , 2024

Link: https://doi.org/10.1016/..

3

Unlocking the potential of higher-molecular-weight 5-HT7R l..:

Pyka, Patryk ; Garbo, Sabrina ; Murzyn, Aleksandra...
Bioorganic Chemistry. 151 (2024) - p. 107668 , 2024

Link: https://doi.org/10.1016/..

4

Preclinical characterization of CPL304110 as a potent and s..:

Popiel, Delfina ; Stańczak, Aleksandra ; Skupińska, Monika...
Frontiers in Oncology. 13 (2024) - p. , 2024

Link: https://doi.org/10.3389/..

5

Tuning the Biological Activity of PI3Kδ Inhibitor by the In..:

Pietruś, Wojciech ; Stypik, Mariola ; Zagozda, Marcin...
Molecules. 28 (2023) 8 - p. 3531 , 2023

Link: https://doi.org/10.3390/..

6

Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Lig..:

Szczepańska, Katarzyna ; Karcz, Tadeusz ; Dichiara, Maria...
Journal of Medicinal Chemistry. 66 (2023) 14 - p. 9658-9683 , 2023

Link: https://doi.org/10.1021/..

7

Impact of the Substitution Pattern at the Basic Center and ..:

Grychowska, Katarzyna ; Pietruś, Wojciech ; Kulawik, Ludmiła...
Molecules. 28 (2023) 3 - p. 1096 , 2023

Link: https://doi.org/10.3390/..

8

Superiority of the Triple-Acting 5-HT6R/5-HT3R Antagonist a..:

Grychowska, Katarzyna ; López-Sánchez, Uriel ; Vitalis, Mathieu...
Journal of Medicinal Chemistry. 66 (2023) 21 - p. 14928-14947 , 2023

Link: https://doi.org/10.1021/..

9

Isomeric Activity Cliffs—A Case Study for Fluorine Substitu..:

Pietruś, Wojciech ; Kurczab, Rafał ; Warszycki, Dawid..
Molecules. 28 (2023) 2 - p. 490 , 2023

Link: https://doi.org/10.3390/..

10

Overcoming undesirable hERG affinity by incorporating fluor..:

Grychowska, Katarzyna ; Olejarz-Maciej, Agnieszka ; Blicharz, Klaudia...
European Journal of Medicinal Chemistry. 236 (2022) - p. 114329 , 2022

Link: https://doi.org/10.1016/..

11

Hydrogen Bonds with Fluorine in Ligand–Protein Complexes-th..:

Pietruś, Wojciech ; Kafel, Rafał ; Bojarski, Andrzej J..
Molecules. 27 (2022) 3 - p. 1005 , 2022

Link: https://doi.org/10.3390/..

12

Design, Synthesis, and Development of Pyrazolo[1,5-a]pyrimi..:

Stypik, Mariola ; Michałek, Stanisław ; Orłowska, Nina...
Pharmaceuticals. 15 (2022) 8 - p. 927 , 2022

Link: https://doi.org/10.3390/..

13

Data-Driven Analysis of Fluorination of Ligands of Aminergi..:

Pietruś, Wojciech ; Kurczab, Rafał ; Stumpfe, Dagmar..
Biomolecules. 11 (2021) 11 - p. 1647 , 2021

Link: https://doi.org/10.3390/..

14

Tuning the activity of known drugs via the introduction of ..:

Staroń, Jakub ; Pietruś, Wojciech ; Bugno, Ryszard...
European Journal of Medicinal Chemistry. 220 (2021) - p. 113533 , 2021

Link: https://doi.org/10.1016/..

15

Imidazopyridine-Based 5-HT6 Receptor Neutral Antagonists: I..:

Vanda, David ; Canale, Vittorio ; Chaumont-Dubel, Severine...
Journal of Medicinal Chemistry. 64 (2021) 2 - p. 1180-1196 , 2021

Link: https://doi.org/10.1021/..