E-LIB Suche - Ergebnisse für: Demont, Emmanuel H.

1

Structure-guided design of a domain-selective bromodomain a..:

Bradley, Erin ; Fusani, Lucia ; Chung, Chun-wa...
https://strathprints.strath.ac.uk/87361/7/Bradley-etal-JMC-2023-Structure-guided-design-of-a-domain-selective-bromodomain-and-extra-terminal-N-terminal.pdf. , 2023

Link: https://strathprints.str..

2

Structure-Guided Design of a Domain-Selective Bromodomain a..:

Bradley, Erin ; Fusani, Lucia ; Chung, Chun-wa...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC10726358/. , 2023

Link: http://www.ncbi.nlm.nih...

3

Optimization of Naphthyridones into Selective TATA-Binding ..:

Clegg, Michael A ; Theodoulou, Natalie H ; Bamborough, Paul...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC8366007/. , 2021

Link: http://www.ncbi.nlm.nih...

4

Selective targeting of BD1 and BD2 of the BET proteins in c..:

Gilan, Omer ; Rioja, Inmaculada ; Knezevic, Kathy...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7610820/. , 2020

Link: http://www.ncbi.nlm.nih...

5

GSK973 Is an Inhibitor of the Second Bromodomains (BD2s) of..:

Preston, Alex ; Atkinson, Stephen J ; Bamborough, Paul...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7429977/. , 2020

Link: http://www.ncbi.nlm.nih...

6

A Chemical Probe for the ATAD2 Bromodomain:

Bamborough, Paul ; Chung, Chun-wa ; Demont, Emmanuel H...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC7314595/. , 2016

Link: http://www.ncbi.nlm.nih...

7

GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromo..:

Bamborough, Paul ; Barnett, Heather A ; Becher, Isabelle...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4904261/. , 2016

Link: http://www.ncbi.nlm.nih...

8

1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibit..:

Demont, Emmanuel H ; Bamborough, Paul ; Chung, Chun-wa...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC4233354/. , 2014

Link: http://www.ncbi.nlm.nih...

9

Discovery of a Selective S1P1 Receptor Agonist Efficacious ..:

Demont, Emmanuel H ; Andrews, Benjamin I ; Bit, Rino A...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC. , 2011

Link: http://www.ncbi.nlm.nih...

10

Structure-Guided Design of a Domain-Selective Bromodomain a..:

Erin Bradley ; Lucia Fusani ; Chun-wa Chung...
doi:10.1021/acs.jmedchem.3c00906.s002. , 2023

Link: https://doi.org/10.1021/..

11

Structure-Guided Design of a Domain-Selective Bromodomain a..:

Erin Bradley ; Lucia Fusani ; Chun-wa Chung...
doi:10.1021/acs.jmedchem.3c00906.s003. , 2023

Link: https://doi.org/10.1021/..

12

Structure-Guided Design of a Domain-Selective Bromodomain a..:

Erin Bradley ; Lucia Fusani ; Chun-wa Chung...
doi:10.1021/acs.jmedchem.3c00906.s001. , 2023

Link: https://doi.org/10.1021/..

13

Multigram Synthesis of Tetrasubsituted Dihydrobenzofuran GS..:

Catherine M. Alder (11991938) ; Matthew Gray (2402251) ; Chelsea A. Huff (1682536)...
https://figshare.com/articles/journal_contribution/Multigram_Synthesis_of_Tetrasubsituted_Dihydrobenzofuran_GSK973_Enabled_by_High-Throughput_Experimentation_and_a_Claisen_Rearrangement_in_Flow/18973037. , 2022

Link: https://doi.org/10.1021/..

14

Optimization of Naphthyridones into Selective TATA-Binding ..:

Michael A. Clegg (8907155) ; Natalie H. Theodoulou (1508650) ; Paul Bamborough (1343466)...
https://figshare.com/articles/journal_contribution/Optimization_of_Naphthyridones_into_Selective_TATA-Binding_Protein_Associated_Factor_1_TAF1_Bromodomain_Inhibitors/15097571. , 2021

Link: https://doi.org/10.1021/..

15

Identification of a Series of N ‑Methylpyridine-2-carboxami..:

Lee A. Harrison (2160145) ; Stephen J. Atkinson (1297362) ; Anna Bassil (10233082)...
https://figshare.com/articles/journal_contribution/Identification_of_a_Series_of_i_N_i_Methylpyridine-2-carboxamides_as_Potent_and_Selective_Inhibitors_of_the_Second_Bromodomain_BD2_of_the_Bromo_and_Extra_Terminal_Domain_BET_Proteins/14924558. , 2021

Link: https://doi.org/10.1021/..