E-LIB Suche - Ergebnisse für: Achab, Abdelghani

1

Oxetane Promise Delivered: Discovery of Long-Acting IDO1 In..:

Li, Derun ; Sloman, David L. ; Achab, Abdelghani...
Journal of Medicinal Chemistry. 65 (2022) 8 - p. 6001-6016 , 2022

Link: https://doi.org/10.1021/..

2

Comprehensive Strategies to Bicyclic Prolines: Applications..:

Li, Derun ; Zhang, Hongjun ; Lyons, Thomas W....
ACS Medicinal Chemistry Letters. 12 (2021) 11 - p. 1678-1688 , 2021

Link: https://doi.org/10.1021/..

3

Discovery of Diaminopyrimidine Carboxamide HPK1 Inhibitors ..:

Vara, Brandon A. ; Levi, Samuel M. ; Achab, Abdelghani...
ACS Medicinal Chemistry Letters. 12 (2021) 4 - p. 653-661 , 2021

Link: https://doi.org/10.1021/..

4

Carbamate andN-Pyrimidine Mitigate Amide Hydrolysis: Struct..:

Li, Derun ; Deng, Yongqi ; Achab, Abdelghani...
ACS Medicinal Chemistry Letters. 12 (2021) 3 - p. 389-396 , 2021

Link: https://doi.org/10.1021/..

5

Projected Dose Optimization of Amino- and Hydroxypyrrolidin..:

Methot, Joey L. ; Zhou, Hua ; McGowan, Meredeth A....
Journal of Medicinal Chemistry. 64 (2021) 8 - p. 5137-5156 , 2021

Link: https://doi.org/10.1021/..

6

Discovery and optimization of heteroaryl piperazines as pot..:

Zhou, Hua ; McGowan, Meredeth A. ; Lipford, Kathryn...
Bioorganic & Medicinal Chemistry Letters. 30 (2020) 1 - p. 126715 , 2020

Link: https://doi.org/10.1016/..

7

Discovery and Optimization of Rationally Designed Bicyclic ..:

Mitcheltree, Matthew J. ; Li, Derun ; Achab, Abdelghani...
ACS Medicinal Chemistry Letters. 11 (2020) 4 - p. 582-588 , 2020

Link: https://doi.org/10.1021/..

8

Optimization of Versatile Oxindoles as Selective PI3Kδ Inhi..:

Methot, Joey L. ; Achab, Abdelghani ; Christopher, Matthew...
ACS Medicinal Chemistry Letters. 11 (2020) 12 - p. 2461-2469 , 2020

Link: https://doi.org/10.1021/..

9

Corrigendum to "Design of selective PI3Kδ inhibitors using ..:

Fradera, Xavier ; Methot, Joey L. ; Achab, Abdelghani...
Bioorganic & Medicinal Chemistry Letters. 30 (2020) 16 - p. 127363 , 2020

Link: https://doi.org/10.1016/..

10

Discovery of Amino-cyclobutarene-derived Indoleamine-2,3-di..:

Zhang, Hongjun ; Liu, Kun ; Pu, Qinglin...
ACS Medicinal Chemistry Letters. 10 (2019) 11 - p. 1530-1536 , 2019

Link: https://doi.org/10.1021/..

11

Design of selective PI3Kδ inhibitors using an iterative sca..:

Fradera, Xavier ; Methot, Joey L. ; Achab, Abdelghani...
Bioorganic & Medicinal Chemistry Letters. 29 (2019) 18 - p. 2575-2580 , 2019

Link: https://doi.org/10.1016/..

12

Structural characterization of nonactive site, TrkA-selecti..:

Su, Hua-Poo ; Rickert, Keith ; Burlein, Christine...
Proceedings of the National Academy of Sciences of the United States of America. 114 (2017) 3 - p. E297-E306 , 2017

Link: https://www.jstor.org/st..

13

Structural characterization of nonactive site, TrkA-selecti..:

Su, Hua-Poo ; Rickert, Keith ; Burlein, Christine...
Proceedings of the National Academy of Sciences. 114 (2016) 3 - p. , 2016

Link: https://doi.org/10.1073/..

14

Discovery and Hit-to-Lead Optimization of Non-ATP Competiti..:

Huang, Xiaohua ; Shipps Jr., Gerald W. ; Cheng, Cliff C....
ACS Medicinal Chemistry Letters. 2 (2011) 8 - p. 632-637 , 2011

Link: https://doi.org/10.1021/..

15

Discovery of Diaminopyrimidine Carboxamide HPK1 Inhibitors ..:

Vara, Brandon A ; Levi, Samuel M ; Achab, Abdelghani...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC8040257/. , 2021

Link: http://www.ncbi.nlm.nih...