E-LIB Suche - Ergebnisse für: Bit, Rino A.

1

Design, Synthesis, and Characterization of I-BET567, a Pan-..:

Humphreys, Philip G. ; Atkinson, Stephen J. ; Bamborough, Paul...
Journal of Medicinal Chemistry. 65 (2022) 3 - p. 2262-2287 , 2022

Link: https://doi.org/10.1021/..

2

Discovery of a Novel Bromodomain and Extra Terminal Domain ..:

Jones, Katherine L. ; Beaumont, Dominic M. ; Bernard, Sharon G....
Journal of Medicinal Chemistry. 64 (2021) 16 - p. 12200-12227 , 2021

Link: https://doi.org/10.1021/..

3

Discovery of a Bromodomain and Extraterminal Inhibitor with..:

Wellaway, Christopher R. ; Amans, Dominique ; Bamborough, Paul...
Journal of Medicinal Chemistry. 63 (2020) 2 - p. 714-746 , 2020

Link: https://doi.org/10.1021/..

4

Discovery of Tetrahydropyrazolopyridine as Sphingosine 1-Ph..:

Demont, Emmanuel H. ; Bailey, James M. ; Bit, Rino A....
Journal of Medicinal Chemistry. 59 (2016) 3 - p. 1003-1020 , 2016

Link: https://doi.org/10.1021/..

5

Discovery of I-BRD9, a Selective Cell Active Chemical Probe..:

Theodoulou, Natalie H. ; Bamborough, Paul ; Bannister, Andrew J....
Journal of Medicinal Chemistry. 59 (2015) 4 - p. 1425-1439 , 2015

Link: https://doi.org/10.1021/..

6

Navigating CYP1A Induction and Arylhydrocarbon Receptor Ago..:

Taylor, Simon J. ; Demont, Emmanuel H. ; Gray, James...
Journal of Medicinal Chemistry. 58 (2015) 20 - p. 8236-8256 , 2015

Link: https://doi.org/10.1021/..

7

Optimization of Sphingosine-1-phosphate-1 Receptor Agonists..:

Skidmore, John ; Heer, Jag ; Johnson, Christopher N....
Journal of Medicinal Chemistry. 57 (2014) 24 - p. 10424-10442 , 2014

Link: https://doi.org/10.1021/..

8

Discovery of a Brain-Penetrant S1P3-Sparing Direct Agonist ..:

Demont, Emmanuel H. ; Arpino, Sandra ; Bit, Rino A....
Journal of Medicinal Chemistry. 54 (2011) 19 - p. 6724-6733 , 2011

Link: https://doi.org/10.1021/..

9

Discovery of a Selective S1P1 Receptor Agonist Efficacious ..:

Demont, Emmanuel H. ; Andrews, Benjamin I. ; Bit, Rino A....
ACS Medicinal Chemistry Letters. 2 (2011) 6 - p. 444-449 , 2011

Link: https://doi.org/10.1021/..

10

Pyrazolopyridazine alpha-2-delta-1 ligands for the treatmen..:

Myatt, James W. ; Healy, Mark P. ; Bravi, Gianpaolo S....
Bioorganic & Medicinal Chemistry Letters. 20 (2010) 15 - p. 4683-4688 , 2010

Link: https://doi.org/10.1016/..

11

Novel methylene-linked heterocyclic EP1 receptor antagonist:

Hall, Adrian ; Bit, Rino A. ; Brown, Susan H....
Bioorganic & Medicinal Chemistry Letters. 18 (2008) 5 - p. 1592-1597 , 2008

Link: https://doi.org/10.1016/..

12

The discovery of 6-[2-(5-chloro-2-{[(2,4-difluorophenyl)met..:

Giblin, Gerard M.P. ; Bit, Rino A. ; Brown, Susan H....
Bioorganic & Medicinal Chemistry Letters. 17 (2007) 2 - p. 385-389 , 2007

Link: https://doi.org/10.1016/..

13

Discovery of novel biaryl heterocyclic EP1 receptor antagon..:

Hall, Adrian ; Bit, Rino A. ; Brown, Susan H....
Bioorganic & Medicinal Chemistry Letters. 16 (2006) 10 - p. 2666-2671 , 2006

Link: https://doi.org/10.1016/..

14

Structure-based design of peptidomimetic antagonists of p56..:

Hobbs, Christopher J. ; Bit, Rino A. ; Cansfield, Andrew D....
Bioorganic & Medicinal Chemistry Letters. 12 (2002) 10 - p. 1365-1369 , 2002

Link: https://doi.org/10.1016/..

15

A convenient synthesis of bisindolylmaleimides:

Bit, Rino A. ; Crackett, Peter H. ; Harris, William.
Tetrahedron Letters. 34 (1993) 35 - p. 5623-5626 , 1993

Link: https://doi.org/10.1016/..