E-LIB Suche - Ergebnisse für: CHAPMAN, KEVIN T.

1

Hit-to-Lead Optimization and Discovery of 5-((5-([1,1′-Biph..:

Lan, Ping ; Romero, F. Anthony ; Wodka, Dariusz...
Journal of Medicinal Chemistry. 60 (2017) 21 - p. 9040-9052 , 2017

2

Discovery of novel, potent, selective, and orally active hu..:

Shen, Dong-Ming ; Brady, Edward J. ; Candelore, Mari R....
Bioorganic & Medicinal Chemistry Letters. 21 (2011) 1 - p. 76-81 , 2011

Link: https://doi.org/10.1016/..

3

Design and Synthesis of Prolylcarboxypeptidase (PrCP) Inhib..:

Zhou, Changyou ; Garcia-Calvo, Margareta ; Pinto, Shirly...
Journal of Medicinal Chemistry. 53 (2010) 19 - p. 7251-7263 , 2010

Link: https://doi.org/10.1021/..

4

Design and synthesis of a new class of malonyl-CoA decarbox..:

Tang, Haifeng ; Yan, Yan ; Feng, Zhe...
Bioorganic & Medicinal Chemistry Letters. 20 (2010) 20 - p. 6088-6092 , 2010

Link: https://doi.org/10.1016/..

5

Application of Affinity Selection/Mass Spectrometry to Dete..:

Adam, Gregory C. ; Parish, Craig A. ; Wisniewski, Douglas...
Journal of the American Chemical Society. 130 (2008) 49 - p. 16704-16710 , 2008

Link: https://doi.org/10.1021/..

6

Synthesis of novel HIV protease inhibitors (PI) with activi..:

Raghavan, Subharekha ; Lu, Zhijian ; Beeson, Teresa...
Bioorganic & Medicinal Chemistry Letters. 17 (2007) 19 - p. 5432-5436 , 2007

Link: https://doi.org/10.1016/..

7

Affinity-based ranking of ligands for DPP-4 from mixtures:

Adam, Gregory C. ; Meng, Juncai ; Athanasopoulos, John..
Bioorganic & Medicinal Chemistry Letters. 17 (2007) 9 - p. 2404-2407 , 2007

Link: https://doi.org/10.1016/..

8

The discovery of a potent and selective lethal factor inhib..:

Xiong, Yusheng ; Wiltsie, Judyann ; Woods, Andrea...
Bioorganic & Medicinal Chemistry Letters. 16 (2006) 4 - p. 964-968 , 2006

Link: https://doi.org/10.1016/..

9

Discovery of novel, potent, and orally active spiro-urea hu..:

Shen, Dong-Ming ; Zhang, Fengqi ; Brady, Edward J....
Bioorganic & Medicinal Chemistry Letters. 15 (2005) 20 - p. 4564-4569 , 2005

Link: https://doi.org/10.1016/..

10

Discovery and investigation of a novel class of thiophene-d..:

Duffy, Joseph L. ; Kirk, Brian A. ; Konteatis, Zenon...
Bioorganic & Medicinal Chemistry Letters. 15 (2005) 5 - p. 1401-1405 , 2005

Link: https://doi.org/10.1016/..

11

The target of ezetimibe is Niemann-Pick C1-Like 1 (NPC1L1):

Garcia-Calvo, Margarita ; Lisnock, JeanMarie ; Bull, Herbert G....
Proceedings of the National Academy of Sciences. 102 (2005) 23 - p. 8132-8137 , 2005

Link: https://doi.org/10.1073/..

12

The Target of Ezetimibe Is Niemann-Pick C1-Like 1 (NPC1L1):

Garcia-Calvo, Margarita ; Lisnock, JeanMarie ; Bull, Herbert G....
Proceedings of the National Academy of Sciences of the United States of America. 102 (2005) 23 - p. 8132-8137 , 2005

Link: https://www.jstor.org/st..

13

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)..:

Shen, Dong-Ming ; Shu, Min ; Mills, Sander G....
Bioorganic & Medicinal Chemistry Letters. 14 (2004) 4 - p. 935-939 , 2004

Link: https://doi.org/10.1016/..

14

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)..:

Shu, Min ; Loebach, Jennifer L ; Parker, Kerry A...
Bioorganic & Medicinal Chemistry Letters. 14 (2004) 4 - p. 947-952 , 2004

Link: https://doi.org/10.1016/..

15

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)..:

Shen, Dong-Ming ; Shu, Min ; Willoughby, Christopher A....
Bioorganic & Medicinal Chemistry Letters. 14 (2004) 4 - p. 941-945 , 2004

Link: https://doi.org/10.1016/..