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Chessari, Gianni
43  Ergebnisse:
Personensuche X
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1

Fragment-Based Discovery of Allosteric Inhibitors of SH2 Do..:

Day, James E. H. ; Berdini, Valerio ; Castro, Joan...
Journal of Medicinal Chemistry.  67 (2024)  6 - p. 4655-4675 , 2024
Link: https://doi.org/10.1021/..
 
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2

Fragment-Based Discovery of a Series of Allosteric-Binding ..:

Palmer, Nick ; Agnew, Christopher ; Benn, Caroline...
Journal of Medicinal Chemistry.  67 (2024)  13 - p. 11168-11181 , 2024
Link: https://doi.org/10.1021/..
 
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3

Enabling synthesis in fragment-based drug discovery (FBDD):..:

Townley, Chloe ; Branduardi, Davide ; Chessari, Gianni...
RSC Medicinal Chemistry.  14 (2023)  12 - p. 2699-2713 , 2023
Link: https://doi.org/10.1039/..
 
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4

Accelerated Chemical Reaction Optimization Using Multi-Task..:

Taylor, Connor J. ; Felton, Kobi C. ; Wigh, Daniel...
ACS Central Science.  9 (2023)  5 - p. 957-968 , 2023
Link: https://doi.org/10.1021/..
 
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5

X-ray Screening of an Electrophilic Fragment Library and Ap..:

St. Denis, Jeffrey D. ; Chessari, Gianni ; Cleasby, Anne...
Journal of Medicinal Chemistry.  65 (2022)  18 - p. 12319-12333 , 2022
Link: https://doi.org/10.1021/..
 
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6

Electrostatic Complementarity in Structure-Based Drug Desig..:

Cons, Benjamin D. ; Twigg, David G. ; Kumar, Rajendra.
Journal of Medicinal Chemistry.  65 (2022)  11 - p. 7476-7488 , 2022
Link: https://doi.org/10.1021/..
 
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7

Structure-Based Design of Potent and Orally Active Isoindol..:

Chessari, Gianni ; Hardcastle, Ian R. ; Ahn, Jong Sook...
Journal of Medicinal Chemistry.  64 (2021)  7 - p. 4071-4088 , 2021
Link: https://doi.org/10.1021/..
 
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8

C–H functionalisation tolerant to polar groups could transf..:

Chessari, Gianni ; Grainger, Rachel ; Holvey, Rhian S....
Chemical Science.  12 (2021)  36 - p. 11976-11985 , 2021
Link: https://doi.org/10.1039/..
 
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9

A Fragment-Derived Clinical Candidate for Antagonism of X-L..:

Johnson, Christopher N. ; Ahn, Jong Sook ; Buck, Ildiko M....
Journal of Medicinal Chemistry.  61 (2018)  16 - p. 7314-7329 , 2018
Link: https://doi.org/10.1021/..
 
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10

Discovery of a Potent Nonpeptidomimetic, Small-Molecule Ant..:

Tamanini, Emiliano ; Buck, Ildiko M. ; Chessari, Gianni...
Journal of Medicinal Chemistry.  60 (2017)  11 - p. 4611-4625 , 2017
Link: https://doi.org/10.1021/..
 
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11

PTEN deficiency promotes macrophage infiltration and hypers..:

Armstrong, Chris W.D. ; Maxwell, Pamela J. ; Ong, Chee Wee...
Oncotarget.  7 (2016)  7 - p. 7885-7898 , 2016
Link: https://doi.org/10.18632..
 
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12

Fragment-Based Drug Discovery Targeting Inhibitor of Apopto..:

Chessari, Gianni ; Buck, Ildiko M. ; Day, James E. H....
Journal of Medicinal Chemistry.  58 (2015)  16 - p. 6574-6588 , 2015
Link: https://doi.org/10.1021/..
 
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13

Identification of novel allosteric inhibitors through fragm..:

Pathuri, Puja ; Saalau-Bethell, Susanne M. ; Woodhead, Andrew J....
Acta Crystallographica Section A Foundations and Advances.  71 (2015)  a1 - p. s38-s38 , 2015
Link: https://doi.org/10.1107/..
 
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14

Discovery of (2,4-Dihydroxy-5-isopropylphenyl)-[5-(4-methyl..:

Woodhead, Andrew J. ; Angove, Hayley ; Carr, Maria G....
Journal of Medicinal Chemistry.  53 (2010)  16 - p. 5956-5969 , 2010
Link: https://doi.org/10.1021/..
 
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15

Fragment-Based Drug Discovery Applied to Hsp90. Discovery o..:

Murray, Christopher W. ; Carr, Maria G. ; Callaghan, Owen...
Journal of Medicinal Chemistry.  53 (2010)  16 - p. 5942-5955 , 2010
Link: https://doi.org/10.1021/..
 
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