E-LIB Suche - Ergebnisse für: Cotesta, Simona

1

Design and Synthesis of Inhibitors of the E3 Ligase SMAD Sp..:

Shaw, Duncan E. ; Smith, Nichola ; Beerli, Rene...
Journal of Medicinal Chemistry. 66 (2023) 12 - p. 8130-8139 , 2023

Link: https://doi.org/10.1021/..

2

BET bromodomain inhibitors regulate keratinocyte plasticity:

Schutzius, Gabi ; Kolter, Christian ; Bergling, Sebastian...
Nature Chemical Biology. 17 (2021) 3 - p. 280-290 , 2021

Link: https://doi.org/10.1038/..

3

Evolution of Novartis' Small Molecule Screening Deck Design:

Schuffenhauer, Ansgar ; Schneider, Nadine ; Hintermann, Samuel...
Journal of Medicinal Chemistry. 63 (2020) 23 - p. 14425-14447 , 2020

Link: https://doi.org/10.1021/..

4

Discovery and Optimization of Novel SUCNR1 Inhibitors: Desi..:

Velcicky, Juraj ; Wilcken, Rainer ; Cotesta, Simona...
Journal of Medicinal Chemistry. 63 (2020) 17 - p. 9856-9875 , 2020

Link: https://doi.org/10.1021/..

5

Structural basis of species-selective antagonist binding to..:

Haffke, Matthias ; Fehlmann, Dominique ; Rummel, Gabriele...
Nature. 574 (2019) 7779 - p. 581-585 , 2019

Link: https://doi.org/10.1038/..

6

Discovery of Asciminib (ABL001), an Allosteric Inhibitor of..:

Schoepfer, Joseph ; Jahnke, Wolfgang ; Berellini, Giuliano...
Journal of Medicinal Chemistry. 61 (2018) 18 - p. 8120-8135 , 2018

Link: https://doi.org/10.1021/..

7

High-Resolution Genetics Identifies the Lipid Transfer Prot..:

Filipuzzi, Ireos ; Cotesta, Simona ; Perruccio, Francesca...
PLOS Genetics. 12 (2016) 11 - p. e1006374 , 2016

Link: https://doi.org/10.1371/..

8

Advantages and Challenges of Phenotypic Screens: The Identi..:

Pries, Verena ; Cotesta, Simona ; Riedl, Ralph...
SLAS Discovery. 21 (2016) 3 - p. 306-315 , 2016

Link: https://doi.org/10.1177/..

9

Gezielte Anreicherung von Wirkstoffen am Knochen am Beispie..:

Jahnke, Wolfgang ; Bold, Guido ; Marzinzik, Andreas L....
Angewandte Chemie. 127 (2015) 48 - p. 14783-14787 , 2015

Link: https://doi.org/10.1002/..

10

Discovery of Novel Allosteric Non‐Bisphosphonate Inhibitors..:

Marzinzik, Andreas L. ; Amstutz, René ; Bold, Guido...
ChemMedChem. 10 (2015) 11 - p. 1884-1891 , 2015

Link: https://doi.org/10.1002/..

11

A General Strategy for Targeting Drugs to Bone:

Jahnke, Wolfgang ; Bold, Guido ; Marzinzik, Andreas L....
Angewandte Chemie International Edition. 54 (2015) 48 - p. 14575-14579 , 2015

Link: https://doi.org/10.1002/..

12

Discovery of 1 H -pyrazolo[3,4- b ]pyridines as potent dual..:

Behnke, Dirk ; Cotesta, Simona ; Hintermann, Samuel...
Bioorganic & Medicinal Chemistry Letters. 25 (2015) 23 - p. 5555-5560 , 2015

Link: https://doi.org/10.1016/..

13

Distinct effects of IPSU and suvorexant on mouse sleep arch..:

Hoyer, Daniel ; Dürst, Thomas ; Fendt, Markus...
Frontiers in Neuroscience. 7 (2013) - p. , 2013

Link: https://doi.org/10.3389/..

14

Kinetic properties of "dual" orexin receptor antagonists at..:

Callander, Gabrielle E. ; Olorunda, Morenike ; Monna, Dominique...
Frontiers in Neuroscience. 7 (2013) - p. , 2013

Link: https://doi.org/10.3389/..

15

Identification of a Novel Series of Orexin Receptor Antagon..:

Betschart, Claudia ; Hintermann, Samuel ; Behnke, Dirk...
Journal of Medicinal Chemistry. 56 (2013) 19 - p. 7590-7607 , 2013

Link: https://doi.org/10.1021/..