E-LIB Suche - Ergebnisse für: Degorce, Sébastien L.

1

Discovery and characterisation of quinazolines and 8-Azaqui..:

O' Donovan, Daniel H. ; Baker, David ; Ciotta, Giovanni...
Bioorganic & Medicinal Chemistry Letters. 96 (2023) - p. 129518 , 2023

Link: https://doi.org/10.1016/..

2

Design of rigid protein–protein interaction inhibitors enab..:

Hargreaves, David ; Carbajo, Rodrigo J. ; Bodnarchuk, Michael S....
Proceedings of the National Academy of Sciences. 120 (2023) 21 - p. , 2023

Link: https://doi.org/10.1073/..

3

Discovery, preclinical validation and early human imaging w..:

Cortes Gonzalez, Miguel Angel ; Jucaite, Aurelija ; Cselenyi, Zsolt...
Nuclear Medicine and Biology. 126-127 (2023) - p. 108465 , 2023

Link: https://doi.org/10.1016/..

4

Identification and optimisation of a pyrimidopyridone serie..:

Cumming, Iain A. ; Degorce, Sébastien L. ; Aagaard, Anna...
Bioorganic & Medicinal Chemistry. 63 (2022) - p. 116729 , 2022

Link: https://doi.org/10.1016/..

5

Discovery of 5-{4-[(7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyri..:

Johannes, Jeffrey W. ; Balazs, Amber ; Barratt, Derek...
Journal of Medicinal Chemistry. 64 (2021) 19 - p. 14498-14512 , 2021

Link: https://doi.org/10.1021/..

6

Improving metabolic stability and removing aldehyde oxidase..:

Degorce, Sébastien L. ; Aagaard, Anna ; Anjum, Rana...
Bioorganic & Medicinal Chemistry. 28 (2020) 23 - p. 115815 , 2020

Link: https://doi.org/10.1016/..

7

Discovery of Proteolysis-Targeting Chimera Molecules that S..:

Degorce, Sébastien L. ; Tavana, Omid ; Banks, Erica...
Journal of Medicinal Chemistry. 63 (2020) 18 - p. 10460-10473 , 2020

Link: https://doi.org/10.1021/..

8

Tricyclic Indazoles—A Novel Class of Selective Estrogen Rec..:

Scott, James S. ; Bailey, Andrew ; Buttar, David...
Journal of Medicinal Chemistry. 62 (2019) 3 - p. 1593-1608 , 2019

Link: https://doi.org/10.1021/..

9

Discovery of a Series of 5-Azaquinazolines as Orally Effica..:

Degorce, Sébastien L. ; Anjum, Rana ; Bloecher, Andrew...
Journal of Medicinal Chemistry. 62 (2019) 21 - p. 9918-9930 , 2019

Link: https://doi.org/10.1021/..

10

Lowering Lipophilicity by Adding Carbon: AzaSpiroHeptanes, ..:

Degorce, Sébastien L. ; Bodnarchuk, Michael S. ; Scott, James S.
ACS Medicinal Chemistry Letters. 10 (2019) 8 - p. 1198-1204 , 2019

Link: https://doi.org/10.1021/..

11

Optimization of permeability in a series of pyrrolotriazine..:

Degorce, Sébastien L. ; Anjum, Rana ; Dillman, Keith S....
Bioorganic & Medicinal Chemistry. 26 (2018) 4 - p. 913-924 , 2018

Link: https://doi.org/10.1016/..

12

Correction to Discovery of Novel 3-Quinoline Carboxamides a..:

Degorce, Sébastien L. ; Barlaam, Bernard ; Cadogan, Elaine...
Journal of Medicinal Chemistry. 61 (2018) 14 - p. 6398-6398 , 2018

Link: https://doi.org/10.1021/..

13

The Identification of Potent, Selective, and Orally Availab..:

Pike, Kurt G. ; Barlaam, Bernard ; Cadogan, Elaine...
Journal of Medicinal Chemistry. 61 (2018) 9 - p. 3823-3841 , 2018

Link: https://doi.org/10.1021/..

14

Lowering Lipophilicity by Adding Carbon: One-Carbon Bridges..:

Degorce, Sébastien L. ; Bodnarchuk, Michael S. ; Cumming, Iain A..
Journal of Medicinal Chemistry. 61 (2018) 19 - p. 8934-8943 , 2018

Link: https://doi.org/10.1021/..

15

EXTH-71. HYPERPOLARIZED [1-13C] PYRUVATE AS A BIOMARKER FOR..:

Tiret, Brice ; Autry, Adam ; Park, Ilwoo...
Neuro-Oncology. 19 (2017) suppl_6 - p. vi88-vi88 , 2017

Link: https://doi.org/10.1093/..