E-LIB Suche - Ergebnisse für: Demont, Emmanuel H.

1

Structure- and Property-Based Optimization of Efficient Pan..:

Hirst, David J. ; Bamborough, Paul ; Al-Mahdi, Niam...
Journal of Medicinal Chemistry. , 2024

Link: https://doi.org/10.1021/..

2

Structure-Guided Design of a Domain-Selective Bromodomain a..:

Bradley, Erin ; Fusani, Lucia ; Chung, Chun-wa...
Journal of Medicinal Chemistry. 66 (2023) 23 - p. 15728-15749 , 2023

Link: https://doi.org/10.1021/..

3

Design and Characterization of 1,3-Dihydro-2H-benzo[d]azepi..:

Bamborough, Paul ; Chung, Chun-wa ; Goodwin, Nicole C....
ACS Medicinal Chemistry Letters. 14 (2023) 9 - p. 1231-1236 , 2023

Link: https://doi.org/10.1021/..

4

Multigram Synthesis of Tetrasubstituted Dihydrobenzofuran G..:

Alder, Catherine M. ; Gray, Matthew ; Huff, Chelsea A....
Organic Process Research & Development. 26 (2022) 2 - p. 365-379 , 2022

Link: https://doi.org/10.1021/..

5

Correction to "Multigram Synthesis of Tetrasubstituted Dihy..:

Alder, Catherine M. ; Gray, Matthew ; Huff, Chelsea A....
Organic Process Research & Development. 26 (2022) 4 - p. 1341-1341 , 2022

Link: https://doi.org/10.1021/..

6

Identification of a Series of N-Methylpyridine-2-carboxamid..:

Harrison, Lee A. ; Atkinson, Stephen J. ; Bassil, Anna...
Journal of Medicinal Chemistry. 64 (2021) 15 - p. 10742-10771 , 2021

Link: https://doi.org/10.1021/..

7

Template-Hopping Approach Leads to Potent, Selective, and H..:

Aylott, Helen E. ; Atkinson, Stephen J. ; Bamborough, Paul...
Journal of Medicinal Chemistry. 64 (2021) 6 - p. 3249-3281 , 2021

Link: https://doi.org/10.1021/..

8

Discovery of a Highly Selective BET BD2 Inhibitor from a DN..:

Rianjongdee, Francesco ; Atkinson, Stephen J. ; Chung, Chun-wa...
Journal of Medicinal Chemistry. 64 (2021) 15 - p. 10806-10833 , 2021

Link: https://doi.org/10.1021/..

9

Fragment-based Scaffold Hopping: Identification of Potent, ..:

Seal, Jonathan T. ; Atkinson, Stephen J. ; Bamborough, Paul...
Journal of Medicinal Chemistry. 64 (2021) 15 - p. 10772-10805 , 2021

Link: https://doi.org/10.1021/..

10

Optimization of a Series of 2,3-Dihydrobenzofurans as Highl..:

Lucas, Simon C. C. ; Atkinson, Stephen J. ; Chung, Chun-wa...
Journal of Medicinal Chemistry. 64 (2021) 15 - p. 10711-10741 , 2021

Link: https://doi.org/10.1021/..

11

Discovery of a Novel Bromodomain and Extra Terminal Domain ..:

Jones, Katherine L. ; Beaumont, Dominic M. ; Bernard, Sharon G....
Journal of Medicinal Chemistry. 64 (2021) 16 - p. 12200-12227 , 2021

Link: https://doi.org/10.1021/..

12

Optimization of Naphthyridones into Selective TATA-Binding ..:

Clegg, Michael A. ; Theodoulou, Natalie H. ; Bamborough, Paul...
ACS Medicinal Chemistry Letters. 12 (2021) 8 - p. 1308-1317 , 2021

Link: https://doi.org/10.1021/..

13

Domain-selective targeting of BET proteins in cancer and im..:

Petretich, Massimo ; Demont, Emmanuel H. ; Grandi, Paola
Current Opinion in Chemical Biology. 57 (2020) - p. 184-193 , 2020

Link: https://doi.org/10.1016/..

14

Design and Synthesis of a Highly Selective and In Vivo-Capa..:

Preston, Alex ; Atkinson, Stephen ; Bamborough, Paul...
Journal of Medicinal Chemistry. 63 (2020) 17 - p. 9070-9092 , 2020

Link: https://doi.org/10.1021/..

15

Structure-Based Design of a Bromodomain and Extraterminal D..:

Wellaway, Christopher R. ; Bamborough, Paul ; Bernard, Sharon G....
Journal of Medicinal Chemistry. 63 (2020) 17 - p. 9020-9044 , 2020

Link: https://doi.org/10.1021/..