E-LIB Suche - Ergebnisse für: Dineen, Thomas A.

1

Discovery of BLU-945, a Reversible, Potent, and Wild-Type-S..:

Eno, Meredith S. ; Brubaker, Jason D. ; Campbell, John E....
Journal of Medicinal Chemistry. 65 (2022) 14 - p. 9662-9677 , 2022

Link: https://doi.org/10.1021/..

2

Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Pot..:

Weiss, Matthew M. ; Dineen, Thomas A. ; Marx, Isaac E....
Journal of Medicinal Chemistry. 60 (2017) 14 - p. 5969-5989 , 2017

Link: https://doi.org/10.1021/..

3

Correction to "Sulfonamides as Selective NaV1.7 Inhibitors:..:

Marx, Isaac E. ; Dineen, Thomas A. ; Able, Jessica...
ACS Medicinal Chemistry Letters. 8 (2017) 3 - p. 378-378 , 2017

Link: https://doi.org/10.1021/..

4

Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Pot..:

Graceffa, Russell F. ; Boezio, Alessandro A. ; Able, Jessica...
Journal of Medicinal Chemistry. 60 (2017) 14 - p. 5990-6017 , 2017

Link: https://doi.org/10.1021/..

5

The discovery of benzoxazine sulfonamide inhibitors of Na V..:

La, Daniel S. ; Peterson, Emily A. ; Bode, Christiane...
Bioorganic & Medicinal Chemistry Letters. 27 (2017) 15 - p. 3477-3485 , 2017

Link: https://doi.org/10.1016/..

6

Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Pot..:

Marx, Isaac E. ; Dineen, Thomas A. ; Able, Jessica...
ACS Medicinal Chemistry Letters. 7 (2016) 12 - p. 1062-1067 , 2016

Link: https://doi.org/10.1021/..

7

Development of 2-aminooxazoline 3-azaxanthenes as orally ef..:

Chen, Jian Jeffrey ; Liu, Qingyian ; Yuan, Chester...
Bioorganic & Medicinal Chemistry Letters. 25 (2015) 4 - p. 767-774 , 2015

Link: https://doi.org/10.1016/..

8

Lead Optimization and Modulation of hERG Activity in a Seri..:

Epstein, Oleg ; Bryan, Marian C. ; Cheng, Alan C....
Journal of Medicinal Chemistry. 57 (2014) 23 - p. 9796-9810 , 2014

Link: https://doi.org/10.1021/..

9

Inhibitors of β-Site Amyloid Precursor Protein Cleaving Enz..:

Dineen, Thomas A. ; Chen, Kui ; Cheng, Alan C....
Journal of Medicinal Chemistry. 57 (2014) 23 - p. 9811-9831 , 2014

Link: https://doi.org/10.1021/..

10

Design and Synthesis of Potent, Orally Efficacious Hydroxye..:

Dineen, Thomas A. ; Weiss, Matthew M. ; Williamson, Toni...
Journal of Medicinal Chemistry. 55 (2012) 21 - p. 9025-9044 , 2012

Link: https://doi.org/10.1021/..

11

Structure- and Property-Based Design of Aminooxazoline Xant..:

Huang, Hongbing ; La, Daniel S. ; Cheng, Alan C....
Journal of Medicinal Chemistry. 55 (2012) 21 - p. 9156-9169 , 2012

Link: https://doi.org/10.1021/..

12

Design and Preparation of a Potent Series of Hydroxyethylam..:

Weiss, Matthew M. ; Williamson, Toni ; Babu-Khan, Safura...
Journal of Medicinal Chemistry. 55 (2012) 21 - p. 9009-9024 , 2012

Link: https://doi.org/10.1021/..

13

Ring opening of aziridines with ortho-bromophenyl metal rea..:

Michaelis, David J. ; Dineen, Thomas A.
Tetrahedron Letters. 50 (2009) 17 - p. 1920-1923 , 2009

Link: https://doi.org/10.1016/..

14

Efficient Transamidation of Primary Carboxamides by in Situ..:

Dineen, Thomas A. ; Zajac, Matthew A. ; Myers, Andrew G.
Journal of the American Chemical Society. 128 (2006) 50 - p. 16406-16409 , 2006

Link: https://doi.org/10.1021/..

15

Stereoselective Synthesis of the Octahydronaphthalene Unit ..:

Dineen, Thomas A. ; Roush, William R.
Organic Letters. 7 (2005) 7 - p. 1355-1358 , 2005

Link: https://doi.org/10.1021/..