E-LIB Suche - Ergebnisse für: Fairhurst, Robin A.

1

Identification of NVP-CLR457 as an Orally Bioavailable Non-..:

Fairhurst, Robin A. ; Furet, Pascal ; Imbach-Weese, Patricia...
Journal of Medicinal Chemistry. 65 (2022) 12 - p. 8345-8379 , 2022

Link: https://doi.org/10.1021/..

2

Exploring the kinetic selectivity of drugs targeting the β1..:

Sykes, David A. ; Jiménez‐Rosés, Mireia ; Reilly, John...
Pharmacology Research & Perspectives. 10 (2022) 4 - p. , 2022

Link: https://doi.org/10.1002/..

3

Correction to "2-Formylpyridyl Ureas as Highly Selective Re..:

Knoepfel, Thomas ; Furet, Pascal ; Mah, Robert...
ACS Medicinal Chemistry Letters. 11 (2020) 11 - p. 2341-2341 , 2020

Link: https://doi.org/10.1021/..

4

Discovery of Roblitinib (FGF401) as a Reversible-Covalent I..:

Fairhurst, Robin A. ; Knoepfel, Thomas ; Buschmann, Nicole...
Journal of Medicinal Chemistry. 63 (2020) 21 - p. 12542-12573 , 2020

Link: https://doi.org/10.1021/..

5

Bile Acid Sequestration by Cholestyramine Mitigates FGFR4 I..:

Schadt, Heiko S ; Wolf, Armin ; Mahl, Joerg Andreas...
Toxicological Sciences. 163 (2018) 1 - p. 265-278 , 2018

Link: https://doi.org/10.1093/..

6

2-Formylpyridyl Ureas as Highly Selective Reversible-Covale..:

Knoepfel, Thomas ; Furet, Pascal ; Mah, Robert...
ACS Medicinal Chemistry Letters. 9 (2018) 3 - p. 215-220 , 2018

Link: https://doi.org/10.1021/..

7

Approaches to selective fibroblast growth factor receptor 4..:

Fairhurst, Robin A. ; Knoepfel, Thomas ; Leblanc, Catherine...
MedChemComm. 8 (2017) 8 - p. 1604-1613 , 2017

Link: https://doi.org/10.1039/..

8

Uncoupling the Structure–Activity Relationships of β2 Adren..:

Dickson, Callum J. ; Hornak, Viktor ; Velez-Vega, Camilo...
Journal of Medicinal Chemistry. 59 (2016) 12 - p. 5780-5789 , 2016

Link: https://doi.org/10.1021/..

9

Optimisation of a 5-[3-phenyl-(2-cyclic-ether)-methyl-ether..:

Fairhurst, Robin A. ; Marsilje, Thomas H. ; Stutz, Stefan...
Bioorganic & Medicinal Chemistry Letters. 26 (2016) 8 - p. 2057-2064 , 2016

Link: https://doi.org/10.1016/..

10

Increasing metabolic stability via the deuterium kinetic is..:

Fairhurst, Robin A. ; Caravatti, Giorgio ; Guagnano, Vito...
Bioorganic & Medicinal Chemistry Letters. 26 (2016) 19 - p. 4729-4734 , 2016

Link: https://doi.org/10.1016/..

11

Discovery of a novel tricyclic 4H-thiazolo[5′,4′:4,5]pyrano..:

Gerspacher, Marc ; Fairhurst, Robin A. ; Mah, Robert...
Bioorganic & Medicinal Chemistry Letters. 25 (2015) 17 - p. 3582-3584 , 2015

Link: https://doi.org/10.1016/..

12

Identification and optimisation of a 4′,5-bisthiazole serie..:

Fairhurst, Robin A. ; Imbach-Weese, Patricia ; Gerspacher, Marc...
Bioorganic & Medicinal Chemistry Letters. 25 (2015) 17 - p. 3569-3574 , 2015

Link: https://doi.org/10.1016/..

13

Identification and optimisation of 4,5-dihydrobenzo[1,2-d:3..:

Fairhurst, Robin A. ; Gerspacher, Marc ; Imbach-Weese, Patricia...
Bioorganic & Medicinal Chemistry Letters. 25 (2015) 17 - p. 3575-3581 , 2015

Link: https://doi.org/10.1016/..

14

The identification of 7-[(R)-2-((1S,2S)-2-benzyloxycyclopen..:

Arnold, Nicola ; Beattie, David ; Bradley, Michelle...
Bioorganic & Medicinal Chemistry Letters. 24 (2014) 17 - p. 4341-4347 , 2014

Link: https://doi.org/10.1016/..

15

Discovery of NVP-BYL719 a potent and selective phosphatidyl..:

Furet, Pascal ; Guagnano, Vito ; Fairhurst, Robin A....
Bioorganic & Medicinal Chemistry Letters. 23 (2013) 13 - p. 3741-3748 , 2013

Link: https://doi.org/10.1016/..