E-LIB Suche - Ergebnisse für: Farmer, Luc J.

1

Robust Strategy for Hit-to-Lead Discovery: NMR for SAR:

Larda, Sacha T. ; Ayotte, Yann ; Denk, Maria M....
Journal of Medicinal Chemistry. 66 (2023) 19 - p. 13416-13427 , 2023

2

Discovery of Novel, Orally Bioavailable β-Amino Acid Azaind..:

Farmer, Luc J. ; Clark, Michael P. ; Boyd, Michael J....
ACS Medicinal Chemistry Letters. 8 (2017) 2 - p. 256-260 , 2017

Link: https://doi.org/10.1021/..

3

Discovery of VX-509 (Decernotinib): A Potent and Selective ..:

Farmer, Luc J. ; Ledeboer, Mark W. ; Hoock, Thomas...
Journal of Medicinal Chemistry. 58 (2015) 18 - p. 7195-7216 , 2015

Link: https://doi.org/10.1021/..

4

Discovery of a Novel, First-in-Class, Orally Bioavailable A..:

Clark, Michael P. ; Ledeboer, Mark W. ; Davies, Ioana...
Journal of Medicinal Chemistry. 57 (2014) 15 - p. 6668-6678 , 2014

Link: https://doi.org/10.1021/..

5

Discovery and SAR of novel 4-thiazolyl-2-phenylaminopyrimid..:

Farmer, Luc J. ; Bemis, Guy ; Britt, Shawn D....
Bioorganic & Medicinal Chemistry Letters. 18 (2008) 23 - p. 6231-6235 , 2008

Link: https://doi.org/10.1016/..

6

Aza-retinoids as novel retinoid X receptor-specific agonist:

Farmer, Luc J. ; Marron, Kristen S. ; Canan Koch, Stacie S....
Bioorganic & Medicinal Chemistry Letters. 16 (2006) 9 - p. 2352-2356 , 2006

Link: https://doi.org/10.1016/..

7

Inhibitors of hepatitis C virus NS3·4A protease 2. Warhead ..:

Perni, Robert B. ; Pitlik, Janos ; Britt, Shawn D....
Bioorganic & Medicinal Chemistry Letters. 14 (2004) 6 - p. 1441-1446 , 2004

Link: https://doi.org/10.1016/..

8

Inhibitors of hepatitis C virus NS3·4A protease. Part 3: P2..:

Perni, Robert B ; Farmer, Luc J ; Cottrell, Kevin M...
Bioorganic & Medicinal Chemistry Letters. 14 (2004) 8 - p. 1939-1942 , 2004

Link: https://doi.org/10.1016/..

9

Inhibitors of hepatitis C virus NS3·4A protease 1. Non-Char..:

Perni, Robert B. ; Britt, Shawn D. ; Court, John C....
Bioorganic & Medicinal Chemistry Letters. 13 (2003) 22 - p. 4059-4063 , 2003

Link: https://doi.org/10.1016/..

10

Retinoic acid receptor ligands based on the 6-cyclopropyl-2..:

Farmer, Luc J. ; Zhi, Lin ; Jeong, Susan...
Bioorganic & Medicinal Chemistry Letters. 13 (2003) 2 - p. 261-264 , 2003

Link: https://doi.org/10.1016/..

11

4-Alkyl- and 3,4-dialkyl-1,2,3,4,-tetrahydro-8-pyridono[5,6..:

Higuchi, Robert I. ; Edwards, James P. ; Caferro, Thomas R....
Bioorganic & Medicinal Chemistry Letters. 9 (1999) 9 - p. 1335-1340 , 1999

Link: https://doi.org/10.1016/..

12

Nonsteroidal progesterone receptor antagonists based on a c..:

Hamann, Lawrence G. ; Winn, David T. ; Pooley, Charlotte L.F....
Bioorganic & Medicinal Chemistry Letters. 8 (1998) 19 - p. 2731-2736 , 1998

Link: https://doi.org/10.1016/..

13

New nonsteroidal androgen receptor modulators based on 4-(t..:

Edwards, James P. ; West, Sarah J. ; Pooley, Charlotte L.F....
Bioorganic & Medicinal Chemistry Letters. 8 (1998) 7 - p. 745-750 , 1998

Link: https://doi.org/10.1016/..

14

Synthesis and Biological Activity of a Novel Series of Nons..:

Hamann, Lawrence G. ; Higuchi, Robert I. ; Zhi, Lin...
Journal of Medicinal Chemistry. 41 (1998) 4 - p. 623-639 , 1998

Link: https://doi.org/10.1021/..

15

Synthesis and structure-activity relationships of potent re..:

Farmer, Luc J. ; Jeong, Susan ; Kallel, E.Adam...
Bioorganic & Medicinal Chemistry Letters. 7 (1997) 18 - p. 2393-2398 , 1997

Link: https://doi.org/10.1016/..