E-LIB Suche - Ergebnisse für: Heald, Robert A.

1

Small-Molecule Polθ Inhibitors Provide Safe and Effective T..:

Rodriguez-Berriguete, Gonzalo ; Ranzani, Marco ; Prevo, Remko...
Clinical Cancer Research. 29 (2023) 8 - p. 1631-1642 , 2023

Link: https://doi.org/10.1158/..

2

Quantitative, titratable and high-throughput reporter assay..:

Rajendra, Eeson ; Grande, Diego ; Mason, Bethany...
Nucleic Acids Research. 52 (2023) 4 - p. 1736-1752 , 2023

Link: https://doi.org/10.1093/..

3

Discovery of GDC-0077 (Inavolisib), a Highly Selective Inhi..:

Hanan, Emily J. ; Braun, Marie-Gabrielle ; Heald, Robert A....
Journal of Medicinal Chemistry. 65 (2022) 24 - p. 16589-16621 , 2022

Link: https://doi.org/10.1021/..

4

Polθ inhibitors elicit BRCA-gene synthetic lethality and ta..:

Zatreanu, Diana ; Robinson, Helen M. R. ; Alkhatib, Omar...
Nature Communications. 12 (2021) 1 - p. , 2021

Link: https://doi.org/10.1038/..

5

Design of Selective Benzoxazepin PI3Kδ Inhibitors Through C..:

Safina, Brian S. ; Elliott, Richard L. ; Forrest, Andrew K....
ACS Medicinal Chemistry Letters. 8 (2017) 9 - p. 936-940 , 2017

Link: https://doi.org/10.1021/..

6

Correction to Noncovalent Mutant Selective Epidermal Growth..:

Heald, Robert ; Bowman, Krista K. ; Bryan, Marian C....
Journal of Medicinal Chemistry. 59 (2016) 6 - p. 2848-2848 , 2016

Link: https://doi.org/10.1021/..

7

Discovery of a Noncovalent, Mutant-Selective Epidermal Grow..:

Chan, Bryan K. ; Hanan, Emily J. ; Bowman, Krista K....
Journal of Medicinal Chemistry. 59 (2016) 19 - p. 9080-9093 , 2016

Link: https://doi.org/10.1021/..

8

The Rational Design of Selective Benzoxazepin Inhibitors of..:

Heffron, Timothy P. ; Heald, Robert A. ; Ndubaku, Chudi...
Journal of Medicinal Chemistry. 59 (2016) 3 - p. 985-1002 , 2016

Link: https://doi.org/10.1021/..

9

Common Marginal Cold Pools:

Mahrt, L. ; Heald, Robert
Journal of Applied Meteorology and Climatology. 54 (2015) 2 - p. 339-351 , 2015

Link: https://www.jstor.org/st..

10

Noncovalent Mutant Selective Epidermal Growth Factor Recept..:

Heald, Robert ; Bowman, Krista K. ; Bryan, Marian C....
Journal of Medicinal Chemistry. 58 (2015) 22 - p. 8877-8895 , 2015

Link: https://doi.org/10.1021/..

11

Pyridones as Highly Selective, Noncovalent Inhibitors of T7..:

Bryan, Marian C. ; Burdick, Daniel J. ; Chan, Bryan K....
ACS Medicinal Chemistry Letters. 7 (2015) 1 - p. 100-104 , 2015

Link: https://doi.org/10.1021/..

12

Structure based design of novel 6,5 heterobicyclic mitogen-..:

Robarge, Kirk D. ; Lee, Wendy ; Eigenbrot, Charles...
Bioorganic & Medicinal Chemistry Letters. 24 (2014) 19 - p. 4714-4723 , 2014

Link: https://doi.org/10.1016/..

13

Discovery of Selective and Noncovalent Diaminopyrimidine-Ba..:

Hanan, Emily J. ; Eigenbrot, Charles ; Bryan, Marian C....
Journal of Medicinal Chemistry. 57 (2014) 23 - p. 10176-10191 , 2014

Link: https://doi.org/10.1021/..

14

Discovery of thiazolobenzoxepin PI3-kinase inhibitors that ..:

Staben, Steven T. ; Ndubaku, Chudi ; Blaquiere, Nicole...
Bioorganic & Medicinal Chemistry Letters. 23 (2013) 9 - p. 2606-2613 , 2013

Link: https://doi.org/10.1016/..

15

Discovery of 2-{3-[2-(1-Isopropyl-3-methyl-1H-1,2–4-triazol..:

Ndubaku, Chudi O. ; Heffron, Timothy P. ; Staben, Steven T....
Journal of Medicinal Chemistry. 56 (2013) 11 - p. 4597-4610 , 2013

Link: https://doi.org/10.1021/..