E-LIB Suche - Ergebnisse für: Hebeisen, Paul

1

Investigation of morpholine isosters for the development of..:

De Pascale, Martina ; Bissegger, Lukas ; Tarantelli, Chiara...
European Journal of Medicinal Chemistry. 248 (2023) - p. 115038 , 2023

Link: https://doi.org/10.1016/..

2

Second-generation tricyclic pyrimido-pyrrolo-oxazine mTOR i..:

Borsari, Chiara ; Keles, Erhan ; Treyer, Andrea...
RSC Medicinal Chemistry. 12 (2021) 4 - p. 579-583 , 2021

Link: https://doi.org/10.1039/..

3

4-(Difluoromethyl)-5-(4-((3R,5S)-3,5-dimethylmorpholino)-6-..:

Borsari, Chiara ; Keles, Erhan ; Rageot, Denise...
Journal of Medicinal Chemistry. 63 (2020) 22 - p. 13595-13617 , 2020

Link: https://doi.org/10.1021/..

4

A Conformational Restriction Strategy for the Identificatio..:

Borsari, Chiara ; Rageot, Denise ; Dall'Asen, Alix...
Journal of Medicinal Chemistry. 62 (2019) 18 - p. 8609-8630 , 2019

Link: https://doi.org/10.1021/..

5

(S)-4-(Difluoromethyl)-5-(4-(3-methylmorpholino)-6-morpholi..:

Rageot, Denise ; Bohnacker, Thomas ; Keles, Erhan...
Journal of Medicinal Chemistry. 62 (2019) 13 - p. 6241-6261 , 2019

Link: https://doi.org/10.1021/..

6

Scalable, Economical, and Practical Synthesis of 4-(Difluor..:

Rageot, Denise ; Beaufils, Florent ; Borsari, Chiara...
Organic Process Research & Development. 23 (2019) 11 - p. 2416-2424 , 2019

Link: https://doi.org/10.1021/..

7

Preclinical Development of PQR514, a Highly Potent PI3K Inh..:

Borsari, Chiara ; Rageot, Denise ; Beaufils, Florent...
ACS Medicinal Chemistry Letters. 10 (2019) 10 - p. 1473-1479 , 2019

Link: https://doi.org/10.1021/..

8

Molecular Structure and Crystal Packing of Monofluoromethox..:

Hebeisen, Paul ; Weiss, Urs ; Alker, André...
European Journal of Organic Chemistry. 2018 (2018) 27-28 - p. 3724-3734 , 2018

Link: https://doi.org/10.1002/..

9

Discovery and Preclinical Characterization of 5-[4,6-Bis({3..:

Rageot, Denise ; Bohnacker, Thomas ; Melone, Anna...
Journal of Medicinal Chemistry. 61 (2018) 22 - p. 10084-10105 , 2018

Link: https://doi.org/10.1021/..

10

5-(4,6-Dimorpholino-1,3,5-triazin-2-yl)-4-(trifluoromethyl)..:

Beaufils, Florent ; Cmiljanovic, Natasa ; Cmiljanovic, Vladimir...
Journal of Medicinal Chemistry. 60 (2017) 17 - p. 7524-7538 , 2017

Link: https://doi.org/10.1021/..

11

6-Alkoxy-5-aryl-3-pyridinecarboxamides, a New Series of Bio..:

Röver, Stephan ; Andjelkovic, Mirjana ; Bénardeau, Agnès...
Journal of Medicinal Chemistry. 56 (2013) 24 - p. 9874-9896 , 2013

Link: https://doi.org/10.1021/..

12

A New DNA Gyrase Inhibitor Subclass of the Cyclothialidine ..:

Angehrn, Peter ; Goetschi, Erwin ; Gmuender, Hans...
Journal of Medicinal Chemistry. 54 (2011) 7 - p. 2207-2224 , 2011

Link: https://doi.org/10.1021/..

13

Orally active aminopyridines as inhibitors of tetrameric fr..:

Hebeisen, Paul ; Haap, Wolfgang ; Kuhn, Bernd...
Bioorganic & Medicinal Chemistry Letters. 21 (2011) 11 - p. 3237-3242 , 2011

Link: https://doi.org/10.1016/..

14

Ring opening of cyclic sulfamidates with bromophenyl metal ..:

Hebeisen, Paul ; Weiss, Urs ; Alker, André.
Tetrahedron Letters. 52 (2011) 41 - p. 5229-5233 , 2011

Link: https://doi.org/10.1016/..

15

Sulfonylureido thiazoles as fructose-1,6-bisphosphatase inh..:

Kitas, Eric ; Mohr, Peter ; Kuhn, Bernd...
Bioorganic & Medicinal Chemistry Letters. 20 (2010) 2 - p. 594-599 , 2010

Link: https://doi.org/10.1016/..