E-LIB Suche - Ergebnisse für: Kettle, Jason

1

P127 Web-Based Videoconferencing for Rural Palliative Care ..:

Paul, Linda Read ; Spice, Ron ; Sinnarajah, Ayn...
Journal of Pain and Symptom Management. 52 (2016) 6 - p. e98-e99 , 2016

Link: https://doi.org/10.1016/..

2

In vitro pharmacological profiles of kinase inhibitors: Com..:

Luke, Richard W.A. ; Rolf, Mike G. ; Bradbury, Rob H....
Journal of Pharmacological and Toxicological Methods. 60 (2009) 2 - p. 219 , 2009

Link: https://doi.org/10.1016/..

3

Alkene–Arene meta Photocycloadditions with a Four‐Carbon‐At..:

Boyd, Joseph W. ; Greaves, Nicola ; Kettle, Jason..
Angewandte Chemie. 117 (2005) 6 - p. 966-968 , 2005

Link: https://doi.org/10.1002/..

4

Alkene–Arene meta Photocycloadditions with a Four‐Carbon‐At..:

Boyd, Joseph W. ; Greaves, Nicola ; Kettle, Jason..
Angewandte Chemie International Edition. 44 (2005) 6 - p. 944-946 , 2005

Link: https://doi.org/10.1002/..

5

Hit-to-lead studies: the discovery of potent, orally active..:

Baxter, Andrew ; Brough, Steve ; Cooper, Anne...
Bioorganic & Medicinal Chemistry Letters. 14 (2004) 11 - p. 2817-2822 , 2004

Link: https://doi.org/10.1016/..

6

Design of a Lead-Like Cysteine-Targeting Covalent Library a..:

Lucas, Simon C. C. ; Milbradt, Alexander G. ; Blackwell, J. Henry...
Journal of Medicinal Chemistry. , 2024

Link: https://doi.org/10.1021/..

7

Metabolism-driven in vitro/in vivo disconnect of an oral ER..:

Hayhow, Thomas G. ; Williamson, Beth ; Lawson, Mandy...
Communications Biology. 7 (2024) 1 - p. , 2024

Link: https://doi.org/10.1038/..

8

Vinylpyridine as a Tunable Covalent Warhead Targeting C797 ..:

Pemberton, Nils ; Compagne, Nina ; Argyrou, Argyrides...
ACS Medicinal Chemistry Letters. 15 (2024) 5 - p. 583-589 , 2024

Link: https://doi.org/10.1021/..

9

Effect of Tether Length on endo/exo Stereoselectivity in Al..:

Alshammari, Aljazy A. A. ; Boyd, Joseph W. ; Greaves, Nicola...
European Journal of Organic Chemistry. , 2024

Link: https://doi.org/10.1002/..

10

Discovery of AZD4747, a Potent and Selective Inhibitor of M..:

Kettle, Jason G. ; Bagal, Sharan K. ; Barratt, Derek...
Journal of Medicinal Chemistry. 66 (2023) 13 - p. 9147-9160 , 2023

Link: https://doi.org/10.1021/..

11

Discovery of the Potent and Selective Inhaled Janus Kinase ..:

Nilsson, Magnus ; Berggren, Kristina ; Berglund, Susanne...
Journal of Medicinal Chemistry. 66 (2023) 19 - p. 13400-13415 , 2023

Link: https://doi.org/10.1021/..

12

Chemical Biology Approaches Confirm MCT4 as the Therapeutic..:

Kawatkar, Aarti ; Clark, Roger A. ; Hopcroft, Lorna...
ACS Chemical Biology. 18 (2023) 2 - p. 296-303 , 2023

Link: https://doi.org/10.1021/..

13

AZD4625 is a Potent and Selective Inhibitor of KRASG12C:

Chakraborty, Atanu ; Hanson, Lyndsey ; Robinson, David...
Molecular Cancer Therapeutics. 21 (2022) 10 - p. 1535-1546 , 2022

Link: https://doi.org/10.1158/..

14

Discovery of AZD4625, a Covalent Allosteric Inhibitor of th..:

Kettle, Jason G. ; Bagal, Sharan K. ; Bickerton, Sue...
Journal of Medicinal Chemistry. 65 (2022) 9 - p. 6940-6952 , 2022

Link: https://doi.org/10.1021/..

15

Discovery of Clinical Candidate AZD0095, a Selective Inhibi..:

Goldberg, Frederick W. ; Kettle, Jason G. ; Lamont, Gillian M....
Journal of Medicinal Chemistry. 66 (2022) 1 - p. 384-397 , 2022

Link: https://doi.org/10.1021/..