E-LIB Suche - Ergebnisse für: Kudolo, Mark

1

Design and Optimization of Novel Benzimidazole- and Imidazo..:

Dimitrov, Teodor ; Moschopoulou, Athina Anastasia ; Seidel, Lennart...
Journal of Medicinal Chemistry. 66 (2023) 11 - p. 7304-7330 , 2023

Link: https://doi.org/10.1021/..

2

Pharmacokinetic Optimization of Small Molecule Janus Kinase..:

Laux, Julian ; Forster, Michael ; Riexinger, Laura...
ACS Pharmacology & Translational Science. 5 (2022) 8 - p. 573-602 , 2022

Link: https://doi.org/10.1021/..

3

Decisive role of water and protein dynamics in residence ti..:

Pantsar, Tatu ; Kaiser, Philipp D. ; Kudolo, Mark...
Nature Communications. 13 (2022) 1 - p. , 2022

Link: https://doi.org/10.1038/..

4

Gefitinib-Tamoxifen Hybrid Ligands as Potent Agents against..:

Abdelmalek, Carine M. ; Hu, Zexi ; Kronenberger, Thales...
Journal of Medicinal Chemistry. 65 (2022) 6 - p. 4616-4632 , 2022

Link: https://doi.org/10.1021/..

5

Development of the First Covalent Monopolar Spindle Kinase ..:

M. Serafim, Ricardo A. ; da Silva Santiago, André ; Schwalm, Martin P....
Journal of Medicinal Chemistry. 65 (2022) 4 - p. 3173-3192 , 2022

Link: https://doi.org/10.1021/..

6

Development of novel urea-based ATM kinase inhibitors with ..:

Dimitrov, Teodor ; Anli, Cetin ; Moschopoulou, Athina Anastasia...
European Journal of Medicinal Chemistry. 235 (2022) - p. 114234 , 2022

Link: https://doi.org/10.1016/..

7

Discovery and Development of First-in-Class ACKR3/CXCR7 Sup..:

Bayrak, Alp ; Mohr, Florian ; Kolb, Kyra...
Journal of Medicinal Chemistry. 65 (2022) 19 - p. 13365-13384 , 2022

Link: https://doi.org/10.1021/..

8

Development of a Selective Dual Discoidin Domain Receptor (..:

Röhm, Sandra ; Berger, Benedict-Tilman ; Schröder, Martin...
Journal of Medicinal Chemistry. 64 (2021) 18 - p. 13451-13474 , 2021

Link: https://doi.org/10.1021/..

9

Discovery of a Potent and Highly Isoform-Selective Inhibito..:

Gerstenecker, Stefan ; Haarer, Lisa ; Schröder, Martin...
Cancers. 13 (2021) 20 - p. 5133 , 2021

Link: https://doi.org/10.3390/..

10

Selective targeting of the αC and DFG-out pocket in p38 MAP:

Röhm, Sandra ; Schröder, Martin ; Dwyer, Jessica E....
European Journal of Medicinal Chemistry. 208 (2020) - p. 112721 , 2020

Link: https://doi.org/10.1016/..

11

Discovery and Evaluation of Enantiopure 9H-pyrimido[4,5-b]i..:

Andreev, Stanislav ; Pantsar, Tatu ; El-Gokha, Ahmed...
International Journal of Molecular Sciences. 21 (2020) 21 - p. 7823 , 2020

Link: https://doi.org/10.3390/..

12

Bioisosteric Replacement of Arylamide-Linked Spine Residues..:

Pedreira, Júlia G. B. ; Nahidino, Philipp ; Kudolo, Mark...
Journal of Medicinal Chemistry. 63 (2020) 13 - p. 7347-7354 , 2020

Link: https://doi.org/10.1021/..

13

Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38..:

Heider, Fabian ; Ansideri, Francesco ; Tesch, Roberta...
European Journal of Medicinal Chemistry. 175 (2019) - p. 309-329 , 2019

Link: https://doi.org/10.1016/..

14

Pyridinylimidazoles as GSK3β Inhibitors: The Impact of Taut..:

Heider, Fabian ; Pantsar, Tatu ; Kudolo, Mark...
ACS Medicinal Chemistry Letters. 10 (2019) 10 - p. 1407-1414 , 2019

Link: https://doi.org/10.1021/..

15

Design, Synthesis and Biological Evaluation of 7-Chloro-9H-..:

Andreev, Stanislav ; Pantsar, Tatu ; Ansideri, Francesco...
Molecules. 24 (2019) 12 - p. 2331 , 2019

Link: https://doi.org/10.3390/..