E-LIB Suche - Ergebnisse für: Maw, Graham

1

Discovery of a Selective TRPM8 Antagonist with Clinical Eff..:

Andrews, Mark D. ; af Forselles, Kerry ; Beaumont, Kevin...
ACS Medicinal Chemistry Letters. 6 (2015) 4 - p. 419-424 , 2015

Link: https://doi.org/10.1021/..

2

The discovery of UK-369003, a novel PDE5 inhibitor with the..:

Rawson, David J. ; Ballard, Stephen ; Barber, Christopher...
Bioorganic & Medicinal Chemistry. 20 (2012) 1 - p. 498-509 , 2012

Link: https://doi.org/10.1016/..

3

A Novel, Efficient, Diastereo- and Enantioselective Mukaiya..:

Batsanov, Andrei S. ; Knowles, Jonathan P. ; Lightfoot, Andrew P....
Organic Letters. 9 (2007) 26 - p. 5565-5568 , 2007

Link: https://doi.org/10.1021/..

4

Small molecule inhibitors of IgE synthesis:

Brown, Alan ; Henderson, Alan ; Lane, Charlotte...
Bioorganic & Medicinal Chemistry Letters. 16 (2006) 17 - p. 4697-4699 , 2006

Link: https://doi.org/10.1016/..

5

4,4,6-Trimethyl-2-vinyl-1,3,2-dioxaborinane: a superior 2-c..:

Lightfoot, Andrew P. ; Maw, Graham ; Thirsk, Carl..
Tetrahedron Letters. 44 (2003) 41 - p. 7645-7648 , 2003

Link: https://doi.org/10.1016/..

6

An unusual Michael addition–dealkylation or elimination via..:

Maw, Graham ; Thirsk, Carl ; Whiting, Andrew
Tetrahedron Letters. 42 (2001) 47 - p. 8387-8390 , 2001

Link: https://doi.org/10.1016/..

7

Discovery and Optimization of Selective Nav1.8 Modulator Se..:

Bagal, Sharan K. ; Bungay, Peter J. ; Denton, Stephen M....
ACS Medicinal Chemistry Letters. 6 (2015) 6 - p. 650-654 , 2015

Link: https://doi.org/10.1021/..

8

Part 3: Design and synthesis of proline-derived α2δ ligands:

Rawson, David J. ; Brugier, Delphine ; Harrison, Anthony...
Bioorganic & Medicinal Chemistry Letters. 21 (2011) 12 - p. 3771-3773 , 2011

Link: https://doi.org/10.1016/..

9

Part 1: N-Alkylated glycines as potent α2δ ligands:

Thompson, Lisa R. ; Blakemore, David C. ; Brugier, Delphine...
Bioorganic & Medicinal Chemistry Letters. 21 (2011) 12 - p. 3764-3766 , 2011

Link: https://doi.org/10.1016/..

10

Part 2: Design, synthesis and evaluation of hydroxyproline-..:

Rawson, David J. ; Brugier, Delphine ; Harrison, Anthony...
Bioorganic & Medicinal Chemistry Letters. 21 (2011) 12 - p. 3767-3770 , 2011

Link: https://doi.org/10.1016/..

11

In vitro and in vivo SAR of pyrido[3,4-d]pyramid-4-ylamine ..:

Mantell, Simon J. ; Gibson, Karl R. ; Osborne, Simon A....
Bioorganic & Medicinal Chemistry Letters. 19 (2009) 8 - p. 2190-2194 , 2009

Link: https://doi.org/10.1016/..

12

SAR of a series of inhaled A2A agonists and comparison of i..:

Mantell, Simon J. ; Stephenson, Peter T. ; Monaghan, Sandra M....
Bioorganic & Medicinal Chemistry Letters. 19 (2009) 15 - p. 4471-4475 , 2009

Link: https://doi.org/10.1016/..

13

2,4-Diaminopyridine δ-opioid receptor agonists and their as..:

Owen, Dafydd R. ; Rodriguez-Lens, Margarita ; Corless, Martin D....
Bioorganic & Medicinal Chemistry Letters. 19 (2009) 6 - p. 1702-1706 , 2009

Link: https://doi.org/10.1016/..

14

Inhaled adenosine A2A receptor agonists for the treatment o..:

Mantell, Simon J. ; Stephenson, Peter T. ; Monaghan, Sandra M....
Bioorganic & Medicinal Chemistry Letters. 18 (2008) 4 - p. 1284-1287 , 2008

Link: https://doi.org/10.1016/..

15

Microwave-assisted synthesis of mGluR1 ligands: carbon, nit..:

Harbottle, Gareth W. ; Feeder, Neil ; Gibson, Karl R....
Tetrahedron Letters. 48 (2007) 24 - p. 4293-4296 , 2007

Link: https://doi.org/10.1016/..