E-LIB Suche - Ergebnisse für: Niculescu-Duvaz, Dan

1

Toward the Scale-Up of a Bicyclic Homopiperazine via Schmid..:

Brown, Michael ; Aljarah, Mohammed ; Asiki, Hannah...
Organic Process Research & Development. 25 (2020) 1 - p. 148-156 , 2020

Link: https://doi.org/10.1021/..

2

Author Correction: Lysyl oxidase drives tumour progression ..:

Tang, HaoRan ; Leung, Leo ; Saturno, Grazia...
Nature Communications. 10 (2019) 1 - p. , 2019

Link: https://doi.org/10.1038/..

3

2-Aminomethylene-5-sulfonylthiazole Inhibitors of Lysyl Oxi..:

Smithen, Deborah A. ; Leung, Leo M. H. ; Challinor, Mairi...
Journal of Medicinal Chemistry. 63 (2019) 5 - p. 2308-2324 , 2019

Link: https://doi.org/10.1021/..

4

Anti-metastatic Inhibitors of Lysyl Oxidase (LOX): Design a..:

Leung, Leo ; Niculescu-Duvaz, Dan ; Smithen, Deborah...
Journal of Medicinal Chemistry. 62 (2019) 12 - p. 5863-5884 , 2019

Link: https://doi.org/10.1021/..

5

Lysyl oxidase drives tumour progression by trapping EGF rec..:

Tang, HaoRan ; Leung, Leo ; Saturno, Grazia...
Nature Communications. 8 (2017) 1 - p. , 2017

Link: https://doi.org/10.1038/..

6

Paradox-Breaking RAF Inhibitors that Also Target SRC Are Ef..:

Girotti, Maria Romina ; Lopes, Filipa ; Preece, Natasha...
Cancer Cell. 31 (2017) 3 - p. 466 , 2017

Link: https://doi.org/10.1016/..

7

Design and discovery of 3-aryl-5-substituted-isoquinolin-1-..:

Elliott, Richard J. R. ; Jarvis, Ashley ; Rajasekaran, Mohan B....
MedChemComm. 6 (2015) 9 - p. 1687-1692 , 2015

Link: https://doi.org/10.1039/..

8

Paradox-Breaking RAF Inhibitors that Also Target SRC Are Ef..:

Girotti, Maria Romina ; Lopes, Filipa ; Preece, Natasha...
Cancer Cell. 27 (2015) 1 - p. 85-96 , 2015

Link: https://doi.org/10.1016/..

9

Potent BRAF kinase inhibitors based on 2,4,5-trisubstituted..:

Niculescu-Duvaz, Dan ; Niculescu-Duvaz, Ion ; Suijkerbuijk, Bart M.J.M....
Bioorganic & Medicinal Chemistry. 21 (2013) 5 - p. 1284-1304 , 2013

Link: https://doi.org/10.1016/..

10

Small molecule inhibitors of BRAF in clinical trials:

Zambon, Alfonso ; Niculescu-Duvaz, Ion ; Niculescu-Duvaz, Dan..
Bioorganic & Medicinal Chemistry Letters. 22 (2012) 2 - p. 789-792 , 2012

Link: https://doi.org/10.1016/..

11

Directed Enzyme Prodrug Therapies:

, In: Prodrugs and Targeted Delivery; Methods and Principles in Medicinal Chemistry,

Niculescu-Duvaz, Dan ; Negoita-Giras, Gabriel ; Niculescu-Duvaz, Ion.. - p. 271-344 , 2011

Link: https://doi.org/10.1002/..

12

C-end your drugs using peptide tags: News and Views:

Niculescu-Duvaz, Dan ; Springer, Caroline ; Marais, Richard
Pigment Cell & Melanoma Research. 23 (2010) 2 - p. 157-159 , 2010

Link: https://doi.org/10.1111/..

13

Novel tricyclic pyrazole BRAF inhibitors with imidazole or ..:

Niculescu-Duvaz, Dan ; Niculescu-Duvaz, Ion ; Suijkerbuijk, Bart M.J.M....
Bioorganic & Medicinal Chemistry. 18 (2010) 18 - p. 6934-6952 , 2010

Link: https://doi.org/10.1016/..

14

Novel Hinge Binder Improves Activity and Pharmacokinetic Pr..:

Zambon, Alfonso ; Ménard, Delphine ; Suijkerbuijk, Bart M. J. M....
Journal of Medicinal Chemistry. 53 (2010) 15 - p. 5639-5655 , 2010

Link: https://doi.org/10.1021/..

15

BRAF Inhibitors Based on an Imidazo[4,5]pyridin-2-one Scaff..:

Nourry, Arnaud ; Zambon, Alfonso ; Davies, Lawrence...
Journal of Medicinal Chemistry. 53 (2010) 5 - p. 1964-1978 , 2010

Link: https://doi.org/10.1021/..