E-LIB Suche - Ergebnisse für: Panchal, Sanjay C

1

Inhibition of MALT1 and BCL2 Induces Synergistic Antitumor ..:

Plotnik, Joshua P. ; Richardson, Adam E. ; Yang, Haopeng...
Molecular Cancer Therapeutics. 23 (2024) 7 - p. 949-960 , 2024

Link: https://doi.org/10.1158/..

2

Discovery of Small Molecule Interleukin 17A Inhibitors with..:

Ramos, Ashley L. ; Goedken, Eric R. ; Frank, Kristine E....
Journal of Medicinal Chemistry. 67 (2024) 8 - p. 6456-6494 , 2024

Link: https://doi.org/10.1021/..

3

Discovery of a Potent Chloroacetamide GPX4 Inhibitor with B..:

Randolph, John T. ; O'Connor, Matthew J. ; Han, Fei...
Journal of Medicinal Chemistry. 66 (2023) 6 - p. 3852-3865 , 2023

Link: https://doi.org/10.1021/..

4

New Platform for Label-Free, Proximal Cellular Pharmacodyna..:

Pu, Fan ; Radosevich, Andrew J. ; Bruckner, Brett G....
ACS Chemical Biology. 18 (2023) 4 - p. 942-948 , 2023

Link: https://doi.org/10.1021/..

5

Identification and structure-based drug design of cell-acti..:

Goedken, Eric R. ; Argiriadi, Maria A. ; Dietrich, Justin D....
Scientific Reports. 12 (2022) 1 - p. , 2022

Link: https://doi.org/10.1038/..

6

The HPK1 Inhibitor A-745 Verifies the Potential of Modulati..:

Malchow, Sven ; Korepanova, Alla ; Panchal, Sanjay C....
ACS Chemical Biology. 17 (2022) 3 - p. 556-566 , 2022

Link: https://doi.org/10.1021/..

7

Selective inhibition of the BD2 bromodomain of BET proteins..:

Faivre, Emily J. ; McDaniel, Keith F. ; Albert, Daniel H....
Nature. 578 (2020) 7794 - p. 306-310 , 2020

Link: https://doi.org/10.1038/..

8

Development of Orally Efficacious Allosteric Inhibitors of ..:

Dietrich, Justin D. ; Longenecker, Kenton L. ; Wilson, Noel S....
Journal of Medicinal Chemistry. 64 (2020) 1 - p. 417-429 , 2020

Link: https://doi.org/10.1021/..

9

Fragment-Based Discovery of an Apolipoprotein E4 (apoE4) St..:

Petros, Andrew M. ; Korepanova, Alla ; Jakob, Clarissa G....
Journal of Medicinal Chemistry. 62 (2019) 8 - p. 4120-4130 , 2019

Link: https://doi.org/10.1021/..

10

Fragment-based discovery of a potent NAMPT inhibitor:

Korepanova, Alla ; Longenecker, Kenton L. ; Pratt, Steve D....
Bioorganic & Medicinal Chemistry Letters. 28 (2018) 3 - p. 437-440 , 2018

Link: https://doi.org/10.1016/..

11

Methylpyrrole inhibitors of BET bromodomains:

Hasvold, Lisa A. ; Sheppard, George S. ; Wang, Le...
Bioorganic & Medicinal Chemistry Letters. 27 (2017) 10 - p. 2225-2233 , 2017

Link: https://doi.org/10.1016/..

12

Fragment-Based, Structure-Enabled Discovery of Novel Pyrido..:

Wang, Le ; Pratt, John K. ; Soltwedel, Todd...
Journal of Medicinal Chemistry. 60 (2017) 9 - p. 3828-3850 , 2017

Link: https://doi.org/10.1021/..

13

Are We There Yet? Applying Thermodynamic and Kinetic Profil..:

Wang, Ying ; Edalji, Rohinton P. ; Panchal, Sanjay C....
Journal of Medicinal Chemistry. 60 (2017) 20 - p. 8321-8335 , 2017

Link: https://doi.org/10.1021/..

14

Cracking the molecular weight barrier: Fragment screening o..:

Mendoza, Renaldo ; Petros, Andrew M. ; Liu, Yaya...
Bioorganic & Medicinal Chemistry Letters. 21 (2011) 18 - p. 5248-5250 , 2011

Link: https://doi.org/10.1016/..

15

Structural basis of actin filament nucleation and processiv..:

Otomo, Takanori ; Tomchick, Diana R. ; Otomo, Chinatsu...
Nature. 433 (2005) 7025 - p. 488-494 , 2005

Link: https://doi.org/10.1038/..