E-LIB Suche - Ergebnisse für: Perola, Emanuele

1

BLU-808, a Potent and Selective Small Molecule Inhibitor of..:

Grassian, Alexandra ; Haidle, Andrew ; AuDuong, Sophia...
Journal of Allergy and Clinical Immunology. 153 (2024) 2 - p. AB62 , 2024

Link: https://doi.org/10.1016/..

2

Discovery of BLU-945, a Reversible, Potent, and Wild-Type-S..:

Eno, Meredith S. ; Brubaker, Jason D. ; Campbell, John E....
Journal of Medicinal Chemistry. 65 (2022) 14 - p. 9662-9677 , 2022

Link: https://doi.org/10.1021/..

3

Discovery of Novel, Orally Bioavailable β-Amino Acid Azaind..:

Farmer, Luc J. ; Clark, Michael P. ; Boyd, Michael J....
ACS Medicinal Chemistry Letters. 8 (2017) 2 - p. 256-260 , 2017

Link: https://doi.org/10.1021/..

4

Novel 2-Substituted 7-Azaindole and 7-Azaindazole Analogues..:

Bandarage, Upul K. ; Clark, Michael P. ; Perola, Emanuele...
ACS Medicinal Chemistry Letters. 8 (2017) 2 - p. 261-265 , 2017

Link: https://doi.org/10.1021/..

5

2-N-Arylthiazole inhibitors of Mycobacterium tuberculosis:

Clark, Michael P. ; Wang, Tiansheng ; Perola, Emanuele...
Bioorganic & Medicinal Chemistry Letters. 27 (2017) 17 - p. 3987-3991 , 2017

Link: https://doi.org/10.1016/..

6

Fragment-Based Discovery of Dual JC Virus and BK Virus Heli..:

Bonafoux, Dominique ; Nanthakumar, Suganthini ; Bandarage, Upul K....
Journal of Medicinal Chemistry. 59 (2016) 15 - p. 7138-7151 , 2016

Link: https://doi.org/10.1021/..

7

Corrigendum to "Isosteric replacements of the carboxylic ac..:

Boyd, Michael J. ; Bandarage, Upul K. ; Bennett, Hamilton...
Bioorganic & Medicinal Chemistry Letters. 26 (2016) 1 - p. 240 , 2016

Link: https://doi.org/10.1016/..

8

Novel Inhibitors of Cholesterol Degradation in Mycobacteriu..:

VanderVen, Brian C. ; Fahey, Ruth J. ; Lee, Wonsik...
PLOS Pathogens. 11 (2015) 2 - p. e1004679 , 2015

Link: https://doi.org/10.1371/..

9

Isosteric replacements of the carboxylic acid of drug candi..:

Boyd, Michael J. ; Bandarage, Upul K. ; Bennett, Hamilton...
Bioorganic & Medicinal Chemistry Letters. 25 (2015) 9 - p. 1990-1994 , 2015

Link: https://doi.org/10.1016/..

10

Successful application of serum shift prediction models to ..:

Perola, Emanuele ; Stamos, Dean ; Grillot, Anne-Laure...
Bioorganic & Medicinal Chemistry Letters. 24 (2014) 9 - p. 2177-2181 , 2014

Link: https://doi.org/10.1016/..

11

Second-Generation Antibacterial Benzimidazole Ureas: Discov..:

Grillot, Anne-Laure ; Tiran, Arnaud Le ; Shannon, Dean...
Journal of Medicinal Chemistry. 57 (2014) 21 - p. 8792-8816 , 2014

Link: https://doi.org/10.1021/..

12

Discovery of a Novel, First-in-Class, Orally Bioavailable A..:

Clark, Michael P. ; Ledeboer, Mark W. ; Davies, Ioana...
Journal of Medicinal Chemistry. 57 (2014) 15 - p. 6668-6678 , 2014

Link: https://doi.org/10.1021/..

13

Development of a Rule-Based Method for the Assessment of Pr..:

Perola, Emanuele ; Herman, Lee ; Weiss, Jonathan
Journal of Chemical Information and Modeling. 52 (2012) 4 - p. 1027-1038 , 2012

Link: https://doi.org/10.1021/..

14

Design, synthesis and biological evaluation of potent NAD+-..:

Gu, Wenxin ; Wang, Tiansheng ; Maltais, Francois...
Bioorganic & Medicinal Chemistry Letters. 22 (2012) 11 - p. 3693-3698 , 2012

Link: https://doi.org/10.1016/..

15

Design, synthesis and biological evaluation of potent NAD+-..:

Wang, Tiansheng ; Duncan, Leonard ; Gu, Wenxin...
Bioorganic & Medicinal Chemistry Letters. 22 (2012) 11 - p. 3699-3703 , 2012

Link: https://doi.org/10.1016/..