E-LIB Suche - Ergebnisse für: Petros, Andrew M.

1

Identification and structure-based drug design of cell-acti..:

Goedken, Eric R. ; Argiriadi, Maria A. ; Dietrich, Justin D....
Scientific Reports. 12 (2022) 1 - p. , 2022

Link: https://doi.org/10.1038/..

2

Efficiently driving protein-based fragment screening and le..:

Peng, Chen ; Namanja, Andrew T. ; Munoz, Eva...
Journal of Biomolecular NMR. 77 (2022) 1-2 - p. 39-53 , 2022

Link: https://doi.org/10.1007/..

3

Insights into the Conformation and Self-Association of a Co..:

Xu, Jianwen ; Namanja, Andrew ; Chan, Siew Leong...
Journal of Pharmaceutical Sciences. 110 (2021) 12 - p. 3819-3828 , 2021

Link: https://doi.org/10.1016/..

4

Development of Orally Efficacious Allosteric Inhibitors of ..:

Dietrich, Justin D. ; Longenecker, Kenton L. ; Wilson, Noel S....
Journal of Medicinal Chemistry. 64 (2020) 1 - p. 417-429 , 2020

Link: https://doi.org/10.1021/..

5

NMR-based fragment screening and lead discovery accelerated..:

Namanja, Andrew T. ; Xu, Jia ; Wu, Haihong...
Journal of Biomolecular NMR. 73 (2019) 12 - p. 675-685 , 2019

Link: https://doi.org/10.1007/..

6

Fragment-Based Discovery of an Apolipoprotein E4 (apoE4) St..:

Petros, Andrew M. ; Korepanova, Alla ; Jakob, Clarissa G....
Journal of Medicinal Chemistry. 62 (2019) 8 - p. 4120-4130 , 2019

Link: https://doi.org/10.1021/..

7

Targeting lysine specific demethylase 4A (KDM4A) tandem TUD..:

Upadhyay, Anup K. ; Judge, Russell A. ; Li, Leiming...
Bioorganic & Medicinal Chemistry Letters. 28 (2018) 10 - p. 1708-1713 , 2018

Link: https://doi.org/10.1016/..

8

Fragment-based discovery of a potent NAMPT inhibitor:

Korepanova, Alla ; Longenecker, Kenton L. ; Pratt, Steve D....
Bioorganic & Medicinal Chemistry Letters. 28 (2018) 3 - p. 437-440 , 2018

Link: https://doi.org/10.1016/..

9

Methylpyrrole inhibitors of BET bromodomains:

Hasvold, Lisa A. ; Sheppard, George S. ; Wang, Le...
Bioorganic & Medicinal Chemistry Letters. 27 (2017) 10 - p. 2225-2233 , 2017

Link: https://doi.org/10.1016/..

10

Fragment-Based, Structure-Enabled Discovery of Novel Pyrido..:

Wang, Le ; Pratt, John K. ; Soltwedel, Todd...
Journal of Medicinal Chemistry. 60 (2017) 9 - p. 3828-3850 , 2017

Link: https://doi.org/10.1021/..

11

Turning a Substrate Peptide into a Potent Inhibitor for the..:

Judge, Russell A. ; Zhu, Haizhong ; Upadhyay, Anup K....
ACS Medicinal Chemistry Letters. 7 (2016) 12 - p. 1102-1106 , 2016

Link: https://doi.org/10.1021/..

12

Structure-Guided Design of a Series of MCL-1 Inhibitors wit..:

Bruncko, Milan ; Wang, Le ; Sheppard, George S....
Journal of Medicinal Chemistry. 58 (2015) 5 - p. 2180-2194 , 2015

Link: https://doi.org/10.1021/..

13

Correction to Structure-Guided Design of a Series of MCL-1 ..:

Bruncko, Milan ; Wang, Le ; Sheppard, George S....
Journal of Medicinal Chemistry. 58 (2015) 9 - p. 4089-4089 , 2015

Link: https://doi.org/10.1021/..

14

Fragment-based discovery of potent inhibitors of the anti-a..:

Petros, Andrew M. ; Swann, Steven L. ; Song, Danying...
Bioorganic & Medicinal Chemistry Letters. 24 (2014) 6 - p. 1484-1488 , 2014

Link: https://doi.org/10.1016/..

15

Discovery and Development of Potent and Selective Inhibitor..:

Sweis, Ramzi F. ; Pliushchev, Marina ; Brown, Peter J....
ACS Medicinal Chemistry Letters. 5 (2014) 2 - p. 205-209 , 2014

Link: https://doi.org/10.1021/..