E-LIB Suche - Ergebnisse für: Tian, Gaochao

1

Identification of highly selective SIK1/2 inhibitors that m..:

Babbe, Holger ; Sundberg, Thomas B. ; Tichenor, Mark...
Proceedings of the National Academy of Sciences. 121 (2023) 1 - p. , 2023

Link: https://doi.org/10.1073/..

2

Small molecule-mediated allosteric activation of the base e..:

Tian, Gaochao ; Katchur, Steven R. ; Jiang, Yong...
Scientific Reports. 12 (2022) 1 - p. , 2022

Link: https://doi.org/10.1038/..

3

Gut-Restricted Selective Cyclooxygenase-2 (COX-2) Inhibitor..:

Zhang, Zhuming ; Ghosh, Avijit ; Connolly, Peter J....
Journal of Medicinal Chemistry. 64 (2021) 15 - p. 11570-11596 , 2021

Link: https://doi.org/10.1021/..

4

Potent Phenylpyridine and Oxodihydrofuran Inhibitors of Cyc..:

Tian, Gaochao ; Suarez, Javier ; Zhang, Zhuming..
Biochemistry. 60 (2021) 31 - p. 2407-2418 , 2021

Link: https://doi.org/10.1021/..

5

Bicyclo((aryl)methyl)benzamides as inhibitors of GlyT1:

Varnes, Jeffrey G. ; Xiong, Hui ; Forst, Janet M....
Bioorganic & Medicinal Chemistry Letters. 28 (2018) 6 - p. 1043-1049 , 2018

Link: https://doi.org/10.1016/..

6

Fragment-assisted hit investigation involving integrated HT..:

Varnes, Jeffrey G. ; Geschwindner, Stefan ; Holmquist, Christopher R....
Bioorganic & Medicinal Chemistry Letters. 26 (2016) 1 - p. 197-202 , 2016

Link: https://doi.org/10.1016/..

7

Mechanism of Inhibition of Fatty Acid Amide Hydrolase by Su..:

Tian, Gaochao ; Paschetto, Kathy A. ; Gharahdaghi, Farzin...
Biochemistry. 50 (2011) 32 - p. 6867-6878 , 2011

Link: https://doi.org/10.1021/..

8

Biochemical characterization and in vitro activity of AZ513..:

Scott, Clay W ; Tian, Gaochao ; Yu, Xiao Hong...
European Journal of Pharmacology. 667 (2011) 1-3 - p. 74-79 , 2011

Link: https://doi.org/10.1016/..

9

Identification of N-(2-(azepan-1-yl)-2-phenylethyl)-benzene..:

Varnes, Jeffrey G. ; Forst, Janet M. ; Hoerter, Tiffany N....
Bioorganic & Medicinal Chemistry Letters. 20 (2010) 16 - p. 4878-4881 , 2010

Link: https://doi.org/10.1016/..

10

Application of Fragment-Based Lead Generation to the Discov..:

Edwards, Philip D. ; Albert, Jeffrey S. ; Sylvester, Mark...
Journal of Medicinal Chemistry. 50 (2007) 24 - p. 5912-5925 , 2007

Link: https://doi.org/10.1021/..

11

Non‐Competitive Inhibition of Solubilized Human γ‐Secretase..:

Tian, Gaochao ; Sobotka‐Briner, Cynthia D. ; Zysk, John...
CNS Drug Reviews. 10 (2004) 2 - p. 198-198 , 2004

Link: https://doi.org/10.1111/..

12

Mechanism of γ-Secretase Cleavage Activation: Is γ-Secreta..:

Knappenberger, Katharine S. ; Tian, Gaochao ; Ye, Xiaomei...
Biochemistry. 43 (2004) 20 - p. 6208-6218 , 2004

Link: https://doi.org/10.1021/..

13

The Mechanism of γ-Secretase:

Tian, Gaochao ; Ghanekar, Smita V. ; Aharony, David...
Journal of Biological Chemistry. 278 (2003) 31 - p. 28968-28975 , 2003

Link: https://doi.org/10.1074/..

14

Modulation of cyclin-dependent kinase 4 by binding of magne..:

Tian, Gaochao ; Kane, Laurie S ; Holmes, William D.
Biophysical Chemistry. 95 (2002) 1 - p. 79-90 , 2002

Link: https://doi.org/10.1016/..

15

Linear Non-competitive Inhibition of Solubilized Human γ-Se..:

Tian, Gaochao ; Sobotka-Briner, Cynthia D. ; Zysk, John...
Journal of Biological Chemistry. 277 (2002) 35 - p. 31499-31505 , 2002

Link: https://doi.org/10.1074/..