E-LIB Suche - Ergebnisse für: Van Aller, Glenn S.

1

Structure-Based Design of a Novel SMYD3 Inhibitor that Brid..:

Van Aller, Glenn S. ; Graves, Alan P. ; Elkins, Patricia A....
Structure. 24 (2016) 5 - p. 774-781 , 2016

Link: https://doi.org/10.1016/..

2

SMYD3 links lysine methylation of MAP3K2 to Ras-driven canc..:

Mazur, Pawel K. ; Reynoird, Nicolas ; Khatri, Purvesh...
Nature. 510 (2014) 7504 - p. 283-287 , 2014

Link: https://doi.org/10.1038/..

3

Long Residence Time Inhibition of EZH2 in Activated Polycom..:

Van Aller, Glenn S. ; Pappalardi, Melissa Baker ; Ott, Heidi M....
ACS Chemical Biology. 9 (2013) 3 - p. 622-629 , 2013

Link: https://doi.org/10.1021/..

4

Development and Validation of Reagents and Assays for EZH2 ..:

Diaz, Elsie ; Machutta, Carl A. ; Chen, Stephanie...
SLAS Discovery. 17 (2012) 10 - p. 1279-1292 , 2012

Link: https://doi.org/10.1177/..

5

Acylprolinamides: A new class of peptide deformylase inhibi..:

Axten, Jeffrey M. ; Medina, Jesús R. ; Blackledge, Charles W....
Bioorganic & Medicinal Chemistry Letters. 22 (2012) 12 - p. 4028-4032 , 2012

Link: https://doi.org/10.1016/..

6

Smyd3 regulates cancer cell phenotypes and catalyzes histon..:

Van Aller, Glenn S. ; Reynoird, Nicolas ; Barbash, Olena...
Epigenetics. 7 (2012) 4 - p. 340-343 , 2012

Link: https://doi.org/10.4161/..

7

Identification of Potent, Selective, Cell-Active Inhibitors..:

Verma, Sharad K. ; Tian, Xinrong ; LaFrance, Louis V....
ACS Medicinal Chemistry Letters. 3 (2012) 12 - p. 1091-1096 , 2012

Link: https://doi.org/10.1021/..

8

EZH2 inhibition as a therapeutic strategy for lymphoma with..:

McCabe, Michael T. ; Ott, Heidi M. ; Ganji, Gopinath...
Nature. 492 (2012) 7427 - p. 108-112 , 2012

Link: https://doi.org/10.1038/..

9

Understanding the Origins of Time-Dependent Inhibition by P..:

Totoritis, Rachel ; Duraiswami, Chaya ; Taylor, Amy N....
Biochemistry. 50 (2011) 31 - p. 6642-6654 , 2011

Link: https://doi.org/10.1021/..

10

Epigallocatechin gallate (EGCG), a major component of green..:

Van Aller, Glenn S. ; Carson, Jeff D. ; Tang, Wei...
Biochemical and Biophysical Research Communications. 406 (2011) 2 - p. 194-199 , 2011

Link: https://doi.org/10.1016/..

11

Discovery of GSK2126458, a Highly Potent Inhibitor of PI3K ..:

Knight, Steven D. ; Adams, Nicholas D. ; Burgess, Joelle L....
ACS Medicinal Chemistry Letters. 1 (2010) 1 - p. 39-43 , 2010

Link: https://doi.org/10.1021/..

12

Characterization of PI3K class IA isoforms with regulatory ..:

Aller, Glenn S. Van ; Carson, Jeff D. ; Fernandes, Christine...
Analytical Biochemistry. 383 (2008) 2 - p. 311-315 , 2008

Link: https://doi.org/10.1016/..

13

Mechanism of Time-Dependent Inhibition of Polypeptide Defor..:

Van Aller, Glenn S. ; Nandigama, Ravi ; Petit, Chantal M....
Biochemistry. 44 (2004) 1 - p. 253-260 , 2004

Link: https://doi.org/10.1021/..

14

First X-ray Cocrystal Structure of a Bacterial FabH Condens..:

Daines, Robert A. ; Pendrak, Israil ; Sham, Kelvin...
Journal of Medicinal Chemistry. 46 (2002) 1 - p. 5-8 , 2002

Link: https://doi.org/10.1021/..

15

Identification, Substrate Specificity, and Inhibition of th..:

Khandekar, Sanjay S. ; Gentry, Daniel R. ; Van Aller, Glenn S....
Journal of Biological Chemistry. 276 (2001) 32 - p. 30024-30030 , 2001

Link: https://doi.org/10.1074/..