E-LIB Suche - Ergebnisse für: van Koppen, Chris J.

1

Potent Dual Inhibitors of Steroid Sulfatase and 17β-Hydroxy..:

Salah, Mohamed ; Tahoun, Mariam ; Rudzitis-Auth, Jeannette...
Journal of Medicinal Chemistry. 66 (2023) 13 - p. 8975-8992 , 2023

Link: https://doi.org/10.1021/..

2

17β-Hydroxysteroid Dehydrogenase Type 1 Inhibition: A Poten..:

Gargano, Emanuele M. ; Mohamed, Abdelrahman ; Abdelsamie, Ahmed S....
ACS Medicinal Chemistry Letters. 12 (2021) 12 - p. 1920-1924 , 2021

Link: https://doi.org/10.1021/..

3

Fluorescent small-molecule agonists as follicle-stimulating..:

Hoogendoorn, Sascha ; van Puijvelde, Gijs H. M. ; van der Marel, Gijs A....
RSC Chemical Biology. 1 (2020) 4 - p. 263-272 , 2020

Link: https://doi.org/10.1039/..

4

Molecular mechanisms of posaconazole- and itraconazole-indu..:

Beck, Katharina R. ; Telisman, Lucija ; van Koppen, Chris J...
The Journal of Steroid Biochemistry and Molecular Biology. 199 (2020) - p. 105605 , 2020

Link: https://doi.org/10.1016/..

5

Profiling of anabolic androgenic steroids and selective and..:

Patt, Melanie ; Beck, Katharina R. ; Di Marco, Tobias...
Biochemical Pharmacology. 172 (2020) - p. 113781 , 2020

Link: https://doi.org/10.1016/..

6

Targeted Endocrine Therapy: Design, Synthesis, and Proof-of..:

Abdelsamie, Ahmed S. ; Herath, Steven ; Biskupek, Yannik...
Journal of Medicinal Chemistry. 62 (2019) 3 - p. 1362-1372 , 2019

Link: https://doi.org/10.1021/..

7

Design, Synthesis, and Biological Characterization of Orall..:

Abdelsamie, Ahmed S. ; Salah, Mohamed ; Siebenbürger, Lorenz...
Journal of Medicinal Chemistry. 62 (2019) 15 - p. 7289-7301 , 2019

Link: https://doi.org/10.1021/..

8

Development of potential preclinical candidates with promis..:

Abdelsamie, Ahmed S. ; Salah, Mohamed ; Siebenbürger, Lorenz...
European Journal of Medicinal Chemistry. 178 (2019) - p. 93-107 , 2019

Link: https://doi.org/10.1016/..

9

Effects of 17β-HSD2 inhibition in bones on osteoporosis bas..:

Müller, Sebastian T. ; Pählig, Sophie ; Merabet, Ahmed...
The Journal of Steroid Biochemistry and Molecular Biology. 192 (2019) - p. 105405 , 2019

Link: https://doi.org/10.1016/..

10

Highly Potent 17β-HSD2 Inhibitors with a Promising Pharmaco..:

Siebenbuerger, Lorenz ; Hernandez-Olmos, Victor ; Abdelsamie, Ahmed S....
Journal of Medicinal Chemistry. 61 (2018) 23 - p. 10724-10738 , 2018

Link: https://doi.org/10.1021/..

11

Accelerated skin wound healing by selective 11β-Hydroxylase..:

Emmerich, Juliette ; van Koppen, Chris J. ; Burkhart, Jens L....
European Journal of Medicinal Chemistry. 143 (2018) - p. 591-597 , 2018

Link: https://doi.org/10.1016/..

12

Treatment of estrogen-dependent diseases: Design, synthesis..:

Abdelsamie, Ahmed S. ; van Koppen, Chris J. ; Bey, Emmanuel...
European Journal of Medicinal Chemistry. 127 (2017) - p. 944-957 , 2017

Link: https://doi.org/10.1016/..

13

Lead Optimization Generates CYP11B1 Inhibitors of Pyridylme..:

Emmerich, Juliette ; van Koppen, Chris J. ; Burkhart, Jens L....
Journal of Medicinal Chemistry. 60 (2017) 12 - p. 5086-5098 , 2017

Link: https://doi.org/10.1021/..

14

First Structure–Activity Relationship of 17β-Hydroxysteroid..:

Braun, Florian ; Bertoletti, Nicole ; Möller, Gabriele...
Journal of Medicinal Chemistry. 59 (2016) 23 - p. 10719-10737 , 2016

Link: https://doi.org/10.1021/..

15

Discovery of Triazole CYP11B2 Inhibitors with in Vivo Activ..:

Hoyt, Scott B. ; Petrilli, Whitney ; London, Clare...
ACS Medicinal Chemistry Letters. 6 (2015) 8 - p. 861-865 , 2015

Link: https://doi.org/10.1021/..