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Bara, Thomas
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1

Substituted 4-morpholine N -arylsulfonamides as γ-secretase..:

Zhao, Zhiqiang ; Pissarnitski, Dmitri A. ; Josien, Hubert B....
European Journal of Medicinal Chemistry.  124 (2016)  - p. 36-48 , 2016
Link: https://doi.org/10.1016/..
 
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2

Iminopyrimidinones: A novel pharmacophore for the developme..:

McKittrick, Brian A. ; Caldwell, John P. ; Bara, Thomas...
Bioorganic & Medicinal Chemistry Letters.  25 (2015)  7 - p. 1592-1596 , 2015
Link: https://doi.org/10.1016/..
 
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3

Discovery of MK-8831, A Novel Spiro-Proline Macrocycle as a..:

Neelamkavil, Santhosh F. ; Agrawal, Sony ; Bara, Thomas...
ACS Medicinal Chemistry Letters.  7 (2015)  1 - p. 111-116 , 2015
Link: https://doi.org/10.1021/..
 
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4

Structure activity relationship studies of tricyclic bispyr..:

Wu, Wen-Lian ; Asberom, Theodros ; Bara, Thomas...
Bioorganic & Medicinal Chemistry Letters.  23 (2013)  3 - p. 844-849 , 2013
Link: https://doi.org/10.1016/..
 
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5

The discovery of fused oxadiazepines as gamma secretase mod..:

Li, Hongmei ; Qin, Jun ; Dhondi, Pawan...
Bioorganic & Medicinal Chemistry Letters.  23 (2013)  2 - p. 466-471 , 2013
Link: https://doi.org/10.1016/..
 
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6

Discovery of SCH 900229, a Potent Presenilin 1 Selective γ-..:

Wu, Wen-Lian ; Domalski, Martin ; Burnett, Duane A....
ACS Medicinal Chemistry Letters.  3 (2012)  11 - p. 892-896 , 2012
Link: https://doi.org/10.1021/..
 
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7

Identification of Presenilin 1-Selective γ-Secretase Inhibi..:

Lee, Julie ; Song, Lixin ; Terracina, Giuseppe...
Biochemistry.  50 (2011)  22 - p. 4973-4980 , 2011
Link: https://doi.org/10.1021/..
 
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8

Cyclic Hydroxyamidines as Amide Isosteres: Discovery of Oxa..:

Sun, Zhong-Yue ; Asberom, Theodros ; Bara, Thomas...
Journal of Medicinal Chemistry.  55 (2011)  1 - p. 489-502 , 2011
Link: https://doi.org/10.1021/..
 
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9

Iminoheterocycles as γ-secretase modulators:

Caldwell, John P. ; Bennett, Chad E. ; McCracken, Troy M....
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  18 - p. 5380-5384 , 2010
Link: https://doi.org/10.1016/..
 
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10

Novel orally active morpholine N-arylsulfonamides γ-secreta..:

Josien, Hubert ; Bara, Thomas ; Rajagopalan, Murali...
Bioorganic & Medicinal Chemistry Letters.  19 (2009)  21 - p. 6032-6037 , 2009
Link: https://doi.org/10.1016/..
 
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11

Discovery of γ-secretase inhibitors efficacious in a transg..:

Asberom, Theodros ; Zhao, Zhiqiang ; Bara, Thomas A....
Bioorganic & Medicinal Chemistry Letters.  17 (2007)  2 - p. 511-516 , 2007
Link: https://doi.org/10.1016/..
 
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12

Tetrahydroquinoline sulfonamides as γ-secretase inhibitors:

Asberom, Theodros ; Bara, Thomas A. ; Clader, John W....
Bioorganic & Medicinal Chemistry Letters.  17 (2007)  1 - p. 205-207 , 2007
Link: https://doi.org/10.1016/..
 
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13

2,6-Disubstituted N-arylsulfonyl piperidines as γ-secretase..:

Pissarnitski, Dmitri A. ; Asberom, Theodros ; Bara, Thomas A....
Bioorganic & Medicinal Chemistry Letters.  17 (2007)  1 - p. 57-62 , 2007
Link: https://doi.org/10.1016/..
 
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14

Small conformationally restricted piperidine N-arylsulfonam..:

Josien, Hubert ; Bara, Thomas ; Rajagopalan, Murali...
Bioorganic & Medicinal Chemistry Letters.  17 (2007)  19 - p. 5330-5335 , 2007
Link: https://doi.org/10.1016/..
 
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15

Discovery of 2,4,6-trisubstituted N-arylsulfonyl piperidine..:

Li, Hongmei ; Asberom, Theodros ; Bara, Thomas A....
Bioorganic & Medicinal Chemistry Letters.  17 (2007)  22 - p. 6290-6294 , 2007
Link: https://doi.org/10.1016/..
 
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