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Brooijmans, Natasja
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1

DrugMap: A quantitative pan-cancer analysis of cysteine lig..:

Takahashi, Mariko ; Chong, Harrison B. ; Zhang, Siwen...
Cell.  187 (2024)  10 - p. 2536-2556.e30 , 2024
Link: https://doi.org/10.1016/..
 
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2

STX-478, a Mutant-Selective, Allosteric PI3Kα Inhibitor Spa..:

Buckbinder, Leonard ; St. Jean Jr, David J. ; Tieu, Trang...
Cancer Discovery.  13 (2023)  11 - p. 2432-2447 , 2023
Link: https://doi.org/10.1158/..
 
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3

Precision Oncology Comes of Age: Designing Best-in-Class Sm..:

Stuart, Darrin D. ; Guzman-Perez, Angel ; Brooijmans, Natasja...
Cancer Discovery.  13 (2023)  10 - p. 2131-2149 , 2023
Link: https://doi.org/10.1158/..
 
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4

Discovery of BLU-945, a Reversible, Potent, and Wild-Type-S..:

Eno, Meredith S. ; Brubaker, Jason D. ; Campbell, John E....
Journal of Medicinal Chemistry.  65 (2022)  14 - p. 9662-9677 , 2022
Link: https://doi.org/10.1021/..
 
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5

Targeting kinases with precision:

Gardino, Alexandra K. ; Evans, Erica K. ; Kim, Joseph L....
Molecular & Cellular Oncology.  5 (2018)  3 - p. e1435183 , 2018
Link: https://doi.org/10.1080/..
 
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6

Large Scale Meta-Analysis of Fragment-Based Screening Campa..:

Kutchukian, Peter S. ; Wassermann, Anne Mai ; Lindvall, Mika K....
SLAS Discovery.  20 (2015)  5 - p. 588-596 , 2015
Link: https://doi.org/10.1177/..
 
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7

Inside the Mind of a Medicinal Chemist: The Role of Human B..:

Kutchukian, Peter S. ; Vasilyeva, Nadya Y. ; Xu, Jordan...
PLoS ONE.  7 (2012)  11 - p. e48476 , 2012
Link: https://doi.org/10.1371/..
 
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8

Identification of 2-oxatriazines as highly potent pan-PI3K/..:

Dehnhardt, Christoph M. ; Venkatesan, Aranapakam M. ; Chen, Zecheng...
Bioorganic & Medicinal Chemistry Letters.  21 (2011)  16 - p. 4773-4778 , 2011
Link: https://doi.org/10.1016/..
 
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9

Discovery and optimization of 2-(4-substituted-pyrrolo[2,3-..:

Tsou, Hwei-Ru ; MacEwan, Gloria ; Birnberg, Gary...
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  7 - p. 2321-2325 , 2010
Link: https://doi.org/10.1016/..
 
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10

Novel imidazolopyrimidines as dual PI3-Kinase/mTOR inhibito..:

Venkatesan, Aranapakam M. ; Dehnhardt, Christoph M. ; Chen, Zecheng...
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  2 - p. 653-656 , 2010
Link: https://doi.org/10.1016/..
 
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11

Chemical space sampling by different scoring functions and ..:

Brooijmans, Natasja ; Humblet, Christine
Journal of Computer-Aided Molecular Design.  24 (2010)  5 - p. 433-447 , 2010
Link: https://doi.org/10.1007/..
 
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12

Bis(morpholino-1,3,5-triazine) Derivatives: Potent Adenosin..:

Venkatesan, Aranapakam M. ; Dehnhardt, Christoph M. ; Delos Santos, Efren...
Journal of Medicinal Chemistry.  53 (2010)  6 - p. 2636-2645 , 2010
Link: https://doi.org/10.1021/..
 
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13

Novel benzofuran-3-one indole inhibitors of PI3 kinase-α an..:

Bursavich, Matthew G. ; Brooijmans, Natasja ; Feldberg, Lawrence...
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  8 - p. 2586-2590 , 2010
Link: https://doi.org/10.1016/..
 
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14

Discovery of 3,6-dihydro-2H-pyran as a morpholine replaceme..:

Kaplan, Joshua ; Verheijen, Jeroen C. ; Brooijmans, Natasja...
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  2 - p. 640-643 , 2010
Link: https://doi.org/10.1016/..
 
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15

A lead discovery strategy driven by a comprehensive analysi..:

Sukuru, Sai Chetan K. ; Nigsch, Florian ; Quancard, Jean...
Protein Science.  19 (2010)  11 - p. 2096-2109 , 2010
Link: https://doi.org/10.1002/..
 
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