E-LIB Suche - Ergebnisse für: Combs, Andrew P.

1

INCB050465 (Parsaclisib), a Novel Next-Generation Inhibitor..:

Yue, Eddy W. ; Li, Yun-Long ; Douty, Brent...
ACS Medicinal Chemistry Letters. 10 (2019) 11 - p. 1554-1560 , 2019

Link: https://doi.org/10.1021/..

2

INCB24360 (Epacadostat), a Highly Potent and Selective Indo..:

Yue, Eddy W. ; Sparks, Richard ; Polam, Padmaja...
ACS Medicinal Chemistry Letters. 8 (2017) 5 - p. 486-491 , 2017

Link: https://doi.org/10.1021/..

3

Synthesis and structure–activity relationships of pyrido[3,..:

Dzierba, Carolyn D. ; Sielecki, Thais M. ; Arvanitis, Argyrios G....
Bioorganic & Medicinal Chemistry Letters. 22 (2012) 15 - p. 4986-4989 , 2012

Link: https://doi.org/10.1016/..

4

Synthesis and in vivo evaluation of cyclic diaminopropane B..:

Thompson, Lorin A. ; Shi, Jianliang ; Decicco, Carl P....
Bioorganic & Medicinal Chemistry Letters. 21 (2011) 22 - p. 6909-6915 , 2011

Link: https://doi.org/10.1016/..

5

INCB16562, a JAK1/2 Selective Inhibitor, Is Efficacious aga..:

Li, Jun ; Favata, Margaret ; Kelley, Jennifer A....
Neoplasia. 12 (2010) 1 - p. 28-38 , 2010

Link: https://doi.org/10.1593/..

6

Discovery of Potent Competitive Inhibitors of Indoleamine 2..:

Yue, Eddy W. ; Douty, Brent ; Wayland, Brian...
Journal of Medicinal Chemistry. 52 (2009) 23 - p. 7364-7367 , 2009

Link: https://doi.org/10.1021/..

7

In Vitro Intrinsic Clearance-Based Optimization of N3-Pheny..:

Hartz, Richard A. ; Ahuja, Vijay T. ; Rafalski, Maria...
Journal of Medicinal Chemistry. 52 (2009) 14 - p. 4161-4172 , 2009

Link: https://doi.org/10.1021/..

8

Corrections to In Vitro Intrinsic Clearance-Based Optimizat..:

Hartz, Richard A. ; Ahuja, Vijay T. ; Rafalski, Maria...
Journal of Medicinal Chemistry. 52 (2009) 18 - p. 5770-5770 , 2009

Link: https://doi.org/10.1021/..

9

Recent Advances in the Discovery of Competitive Protein Tyr..:

Combs, Andrew P.
Journal of Medicinal Chemistry. 53 (2009) 6 - p. 2333-2344 , 2009

Link: https://doi.org/10.1021/..

10

Synthesis, Structure−Activity Relationships, and In Vivo Ev..:

Hartz, Richard A. ; Ahuja, Vijay T. ; Arvanitis, Argyrios G....
Journal of Medicinal Chemistry. 52 (2009) 14 - p. 4173-4191 , 2009

Link: https://doi.org/10.1021/..

11

Isothiazolidinone inhibitors of PTP1B containing imidazoles..:

Douty, Brent ; Wayland, Brian ; Ala, Paul J....
Bioorganic & Medicinal Chemistry Letters. 18 (2008) 1 - p. 66-71 , 2008

Link: https://doi.org/10.1016/..

12

Asymmetric Synthesis of the (S)-1,1-Dioxido-isothiazolidin-..:

Combs, Andrew P. ; Glass, Brian ; Galya, Laurine G..
Organic Letters. 9 (2007) 7 - p. 1279-1282 , 2007

Link: https://doi.org/10.1021/..

13

Benzothiazole benzimidazole (S)-isothiazolidinone derivativ..:

Sparks, Richard B. ; Polam, Padmaja ; Zhu, Wenyu...
Bioorganic & Medicinal Chemistry Letters. 17 (2007) 3 - p. 736-740 , 2007

Link: https://doi.org/10.1016/..

14

Dihydropyridopyrazinones and Dihydropteridinones as Cortico..:

Dzierba, Carolyn D. ; Tebben, Andrew J. ; Wilde, Richard G....
Journal of Medicinal Chemistry. 50 (2007) 9 - p. 2269-2272 , 2007

Link: https://doi.org/10.1021/..

15

Structural Insights into the Design of Nonpeptidic Isothiaz..:

Ala, Paul J. ; Gonneville, Lucie ; Hillman, Milton...
Journal of Biological Chemistry. 281 (2006) 49 - p. 38013-38021 , 2006

Link: https://doi.org/10.1074/..