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E. A. Chessum, Nicola
20  results:
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1

HSF1 Pathway Inhibitor Clinical Candidate (CCT361814/NXP800..:

Pasqua, A. Elisa ; Sharp, Swee Y. ; Chessum, Nicola E. A....
Journal of Medicinal Chemistry.  66 (2023)  8 - p. 5907-5936 , 2023
Link: https://doi.org/10.1021/..
 
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2

Determination of Ligand-Binding Affinity (Kd) Using Transve..:

Liu, Manjuan ; Mirza, Amin ; McAndrew, P. Craig...
Journal of Medicinal Chemistry.  66 (2023)  15 - p. 10617-10627 , 2023
Link: https://doi.org/10.1021/..
 
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3

Investigating the phosphinic acid tripeptide mimetic DG013A..:

Wilding, Birgit ; Pasqua, A. Elisa ; E. A. Chessum, Nicola...
Bioorganic & Medicinal Chemistry Letters.  42 (2021)  - p. 128050 , 2021
Link: https://doi.org/10.1016/..
 
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4

Demonstrating In-Cell Target Engagement Using a Pirin Prote..:

Chessum, Nicola E. A. ; Sharp, Swee Y. ; Caldwell, John J....
Journal of Medicinal Chemistry.  61 (2018)  3 - p. 918-933 , 2018
Link: https://doi.org/10.1021/..
 
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5

Privileged Structures and Polypharmacology within and betwe..:

Meyers, Joshua ; Chessum, Nicola E. A. ; Ali, Salyha...
ACS Medicinal Chemistry Letters.  9 (2018)  12 - p. 1199-1204 , 2018
Link: https://doi.org/10.1021/..
 
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6

Discovery of a Chemical Probe Bisamide (CCT251236): An Oral..:

Cheeseman, Matthew D. ; Chessum, Nicola E. A. ; Rye, Carl S....
Journal of Medicinal Chemistry.  60 (2016)  1 - p. 180-201 , 2016
Link: https://doi.org/10.1021/..
 
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7

Discovery of 4,6-disubstituted pyrimidines as potent inhibi..:

Rye, Carl S. ; Chessum, Nicola E. A. ; Lamont, Scott...
MedChemComm.  7 (2016)  8 - p. 1580-1586 , 2016
Link: https://doi.org/10.1039/..
 
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8

Correction: Discovery of 4,6-disubstituted pyrimidines as p..:

Rye, Carl S. ; Chessum, Nicola E. A. ; Lamont, Scott...
MedChemComm.  7 (2016)  9 - p. 1870-1870 , 2016
Link: https://doi.org/10.1039/..
 
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9

A model β-sheet interaction and thermodynamic analysis of β..:

Robinson, Colin W. ; Rye, Carl S. ; Chessum, Nicola E. A..
Organic & Biomolecular Chemistry.  13 (2015)  27 - p. 7402-7407 , 2015
Link: https://doi.org/10.1039/..
 
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10

Synthesis and in vivo evaluation of 3-substituted gababutin:

Blakemore, David C. ; Bryans, Justin S. ; Carnell, Pauline...
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  1 - p. 362-365 , 2010
Link: https://doi.org/10.1016/..
 
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11

Synthesis and in vivo evaluation of bicyclic gababutins:

Blakemore, David C. ; Bryans, Justin S. ; Carnell, Pauline...
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  2 - p. 461-464 , 2010
Link: https://doi.org/10.1016/..
 
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12

Metal-catalysed radical cyclisations leading to N-heterocyc..:

Bryans, Justin S ; Chessum, Nicola E.A ; Huther, Nathalie..
Tetrahedron.  59 (2003)  33 - p. 6221-6231 , 2003
Link: https://doi.org/10.1016/..
 
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13

The synthesis of functionalised β- and γ-lactams by cyclisa..:

Bryans, Justin S ; Chessum, Nicola E.A ; Parsons, Andrew F.
Tetrahedron Letters.  42 (2001)  15 - p. 2901-2905 , 2001
Link: https://doi.org/10.1016/..
 
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14

Confounding Factors in Targeted Degradation of Short-Lived ..:

Vetma, Vesna ; Perez, Laura Casares ; Eliaš, Ján...
ACS Chemical Biology.  19 (2024)  7 - p. 1484-1494 , 2024
Link: https://doi.org/10.1021/..
 
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15

An efficient synthesis of 2,3-diaryl (3H)-quinazolin-4-ones..:

Kalusa, Andrew ; Chessum, Nicola ; Jones, Keith
Tetrahedron Letters.  49 (2008)  41 - p. 5840-5842 , 2008
Link: https://doi.org/10.1016/..
 
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