Fushimi, Makoto
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1

Addition to "Scaffold Hopping and Optimization of Small Mol..:

Sun, Shan ; Fushimi, Makoto ; Rossetti, Thomas...
Journal of Chemical Information and Modeling.  64 (2024)  3 - p. 1106-1106 , 2024
 
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2

Regiodivergent Nucleophilic Fluorination under Hydrogen Bon..:

Horwitz, Matthew A. ; Dürr, Alexander B. ; Afratis, Konstantinos...
Journal of the American Chemical Society.  145 (2023)  17 - p. 9708-9717 , 2023
 
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3

Scaffold Hopping and Optimization of Small Molecule Soluble..:

Sun, Shan ; Fushimi, Makoto ; Rossetti, Thomas...
Journal of Chemical Information and Modeling.  63 (2023)  9 - p. 2828-2841 , 2023
 
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4

Design, Synthesis, and Pharmacological Evaluation of Second..:

Miller, Michael ; Rossetti, Thomas ; Ferreira, Jacob...
Journal of Medicinal Chemistry.  65 (2022)  22 - p. 15208-15226 , 2022
 
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6

Discovery of TDI-10229: A Potent and Orally Bioavailable In..:

Fushimi, Makoto ; Buck, Hannes ; Balbach, Melanie...
ACS Medicinal Chemistry Letters.  12 (2021)  8 - p. 1283-1287 , 2021
 
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7

Discovery of a Novel and Brain-Penetrant O-GlcNAcase Inhibi..:

Tawada, Michiko ; Fushimi, Makoto ; Masuda, Kei...
Journal of Medicinal Chemistry.  64 (2021)  2 - p. 1103-1115 , 2021
 
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8

T‐495, a novel low cooperative M1 receptor positive alloste..:

Mandai, Takao ; Sako, Yuu ; Kurimoto, Emi...
Pharmacology Research & Perspectives.  8 (2020)  1 - p. , 2020
 
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12

Design, Synthesis, and Evaluation of Piperazinyl Pyrrolidin..:

Aida, Jumpei ; Fushimi, Makoto ; Kusumoto, Tomokazu...
Journal of Medicinal Chemistry.  61 (2018)  20 - p. 9205-9217 , 2018
 
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13

Design and synthesis of potent and selective pyridazin-4(1H..:

Yoshikawa, Masato ; Hitaka, Takenori ; Hasui, Tomoaki...
Bioorganic & Medicinal Chemistry.  24 (2016)  16 - p. 3447-3455 , 2016
 
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14

Discovery of 1-[2-Fluoro-4-(1H-pyrazol-1-yl)phenyl]-5-metho..:

Kunitomo, Jun ; Yoshikawa, Masato ; Fushimi, Makoto...
Journal of Medicinal Chemistry.  57 (2014)  22 - p. 9627-9643 , 2014
 
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15

Catalytic Enantioselective 1,3-Dipolar Cycloadditions of Ni..:

Sakakura, Akira ; Hori, Masahiro ; Fushimi, Makoto.
Journal of the American Chemical Society.  132 (2010)  44 - p. 15550-15552 , 2010
 
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