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Gosmini, Romain
24  results:
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1

Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR fo..:

Pizzonero, Mathieu ; Akkari, Rhalid ; Bock, Xavier...
Journal of Medicinal Chemistry.  67 (2024)  7 - p. 5216-5232 , 2024
Link: https://doi.org/10.1021/..
 
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2

Optimization of Selectivity and Pharmacokinetic Properties ..:

Temal-Laib, Taouès ; Peixoto, Christophe ; Desroy, Nicolas...
Journal of Medicinal Chemistry.  67 (2023)  1 - p. 380-401 , 2023
Link: https://doi.org/10.1021/..
 
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3

Discovery of GLPG1972/S201086, a Potent, Selective, and Ora..:

Brebion, Franck ; Gosmini, Romain ; Deprez, Pierre...
Journal of Medicinal Chemistry.  64 (2021)  6 - p. 2937-2952 , 2021
Link: https://doi.org/10.1021/..
 
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4

Three classes of ligands each bind to distinct sites on the..:

Mahmud, Zobaer Al ; Jenkins, Laura ; Ulven, Trond...
Scientific Reports.  7 (2017)  1 - p. , 2017
Link: https://doi.org/10.1038/..
 
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5

The Discovery of I-BET726 (GSK1324726A), a Potent Tetrahydr..:

Gosmini, Romain ; Nguyen, Van Loc ; Toum, Jérôme...
Journal of Medicinal Chemistry.  57 (2014)  19 - p. 8111-8131 , 2014
Link: https://doi.org/10.1021/..
 
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6

BET Inhibition Silences Expression of MYCN and BCL2 and Ind..:

Wyce, Anastasia ; Ganji, Gopinath ; Smitheman, Kimberly N....
PLoS ONE.  8 (2013)  8 - p. e72967 , 2013
Link: https://doi.org/10.1371/..
 
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7

Discovery of Epigenetic Regulator I-BET762: Lead Optimizati..:

Mirguet, Olivier ; Gosmini, Romain ; Toum, Jérôme...
Journal of Medicinal Chemistry.  56 (2013)  19 - p. 7501-7515 , 2013
Link: https://doi.org/10.1021/..
 
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8

From ApoA1 upregulation to BET family bromodomain inhibitio..:

Mirguet, Olivier ; Lamotte, Yann ; Donche, Frédéric...
Bioorganic & Medicinal Chemistry Letters.  22 (2012)  8 - p. 2963-2967 , 2012
Link: https://doi.org/10.1016/..
 
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9

Discovery and Characterization of Small Molecule Inhibitors..:

Chung, Chun-wa ; Coste, Hervé ; White, Julia H....
Journal of Medicinal Chemistry.  54 (2011)  11 - p. 3827-3838 , 2011
Link: https://doi.org/10.1021/..
 
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10

?-t-butyl- and ?-i-propyl-ortho-hydroxybenzylamines: Racemi..:

Bernardinelli, G�rald ; Fernandez, Daniel ; Gosmini, Romain...
Chirality.  12 (2000)  5-6 - p. 529-539 , 2000
Link: https://doi.org/10.1002/..
 
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11

Regio and enantioselective synthesis of 4-carbomethoxymethy..:

Raussou, Sabine ; Gosmini, Romain ; Mangeney, Pierre..
Tetrahedron Letters.  35 (1994)  30 - p. 5433-5436 , 1994
Link: https://doi.org/10.1016/..
 
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12

Diastereoselective addition of organocuprates on 1,4-dihydr..:

Mangeney, Pierre ; Gosmini, Romain ; Raussou, Sabine.
Tetrahedron Letters.  34 (1993)  40 - p. 6399-6402 , 1993
Link: https://doi.org/10.1016/..
 
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13

Enantioselective synthesis of indoloquinolizidines:

Mangeney, Pierre ; Gosmini, Romain ; Alexakis, Alexandre
Tetrahedron Letters.  32 (1991)  32 - p. 3981-3984 , 1991
Link: https://doi.org/10.1016/..
 
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14

Optimization of Selectivity and Pharmacokinetic Properties ..:

Temal-Laib, Taouès ; Peixoto, Christophe ; Desroy, Nicolas...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC10788895/.  , 2023
Link: http://www.ncbi.nlm.nih...
 
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15

Discovery of 9-Cyclopropylethynyl-2-((S)-1-[1,4]dioxan-2-yl..:

Labéguère, Frédéric ; Dupont, Sonia ; Alvey, Luke...
https://eprints.gla.ac.uk/230270/1/230270.pdf.  , 2020
Link: https://eprints.gla.ac.u..
 
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