Hawes, Brian E.
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1

In vitro pharmacological characterization of vorapaxar, a n..:

Hawes, Brian E. ; Zhai, Ying ; Hesk, David...
European Journal of Pharmacology.  762 (2015)  - p. 221-228 , 2015
 
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3

SAR study of bicyclo[4.1.0]heptanes as melanin-concentratin..:

Su, Jing ; McKittrick, Brian A. ; Tang, Haiqun...
Bioorganic & Medicinal Chemistry.  15 (2007)  16 - p. 5369-5385 , 2007
 
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4

Synthesis of novel bicyclo[4.1.0]heptane and bicyclo[3.1.0]..:

Su, Jing ; Tang, Haiqun ; McKittrick, Brian A....
Bioorganic & Medicinal Chemistry Letters.  17 (2007)  17 - p. 4845-4850 , 2007
 
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5

Effects of a selective melanin-concentrating hormone 1 rece..:

Kowalski, Timothy J. ; Spar, Brian D. ; Weig, Blair...
European Journal of Pharmacology.  535 (2006)  1-3 - p. 182-191 , 2006
 
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6

Discovery of Orally Efficacious Melanin-Concentrating Hormo..:

McBriar, Mark D. ; Guzik, Henry ; Shapiro, Sherry...
Journal of Medicinal Chemistry.  49 (2006)  7 - p. 2294-2310 , 2006
 
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7

Synthesis and structure–activity relationships of piperidin..:

Wu, Wen-Lian ; Burnett, Duane A. ; Spring, Richard...
Bioorganic & Medicinal Chemistry Letters.  16 (2006)  14 - p. 3668-3673 , 2006
 
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8

Design and synthesis of orally efficacious benzimidazoles a..:

Wu, Wen-Lian ; Burnett, Duane A. ; Caplen, Mary Ann...
Bioorganic & Medicinal Chemistry Letters.  16 (2006)  14 - p. 3674-3678 , 2006
 
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9

Bicyclic[4.1.0]heptanes as phenyl replacements for melanin ..:

Xu, Ruo ; Li, Shengjian ; Paruchova, Jaroslava...
Bioorganic & Medicinal Chemistry.  14 (2006)  10 - p. 3285-3299 , 2006
 
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10

Novel aminobenzimidazoles as selective MCH-R1 antagonists f..:

Sasikumar, T.K. ; Qiang, Li ; Burnett, Duane A....
Bioorganic & Medicinal Chemistry Letters.  16 (2006)  20 - p. 5427-5431 , 2006
 
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11

Discovery of melanin-concentrating hormone receptor R1 anta..:

Su, Jing ; McKittrick, Brian A. ; Tang, Haiqun...
Bioorganic & Medicinal Chemistry.  13 (2005)  5 - p. 1829-1836 , 2005
 
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12

The target of ezetimibe is Niemann-Pick C1-Like 1 (NPC1L1):

Garcia-Calvo, Margarita ; Lisnock, JeanMarie ; Bull, Herbert G....
Proceedings of the National Academy of Sciences.  102 (2005)  23 - p. 8132-8137 , 2005
 
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13

Discovery of Bicycloalkyl Urea Melanin Concentrating Hormon..:

McBriar, Mark D. ; Guzik, Henry ; Xu, Ruo...
Journal of Medicinal Chemistry.  48 (2005)  7 - p. 2274-2277 , 2005
 
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14

The Target of Ezetimibe Is Niemann-Pick C1-Like 1 (NPC1L1):

Garcia-Calvo, Margarita ; Lisnock, JeanMarie ; Bull, Herbert G....
Proceedings of the National Academy of Sciences of the United States of America.  102 (2005)  23 - p. 8132-8137 , 2005
 
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