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Hayhow, Thomas G.
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1

Metabolism-driven in vitro/in vivo disconnect of an oral ER..:

Hayhow, Thomas G. ; Williamson, Beth ; Lawson, Mandy...
Communications Biology.  7 (2024)  1 - p. , 2024
Link: https://doi.org/10.1038/..
 
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2

Degradation by Design: New Cyclin K Degraders from Old CDK ..:

Thomas, Katie L. ; Bouguenina, Habib ; Miller, Daniel S. J....
ACS Chemical Biology.  19 (2024)  1 - p. 173-184 , 2024
Link: https://doi.org/10.1021/..
 
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3

Design, Synthesis, and Characterization of I-BET567, a Pan-..:

Humphreys, Philip G. ; Atkinson, Stephen J. ; Bamborough, Paul...
Journal of Medicinal Chemistry.  65 (2022)  3 - p. 2262-2287 , 2022
Link: https://doi.org/10.1021/..
 
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4

Modulation of macrophage inflammatory function through sele..:

Ghiboub, Mohammed ; Koster, Jan ; Craggs, Peter D....
BMC Biology.  20 (2022)  1 - p. , 2022
Link: https://doi.org/10.1186/..
 
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5

Template-Hopping Approach Leads to Potent, Selective, and H..:

Aylott, Helen E. ; Atkinson, Stephen J. ; Bamborough, Paul...
Journal of Medicinal Chemistry.  64 (2021)  6 - p. 3249-3281 , 2021
Link: https://doi.org/10.1021/..
 
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6

The Optimization of a Novel, Weak Bromo and Extra Terminal ..:

Seal, Jonathan T. ; Atkinson, Stephen J. ; Aylott, Helen...
Journal of Medicinal Chemistry.  63 (2020)  17 - p. 9093-9126 , 2020
Link: https://doi.org/10.1021/..
 
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7

A Buchwald–Hartwig Protocol to Enable Rapid Linker Explorat..:

Hayhow, Thomas G. ; Borrows, Rachel E. A. ; Diène, Coura R....
Chemistry – A European Journal.  26 (2020)  70 - p. 16818-16823 , 2020
Link: https://doi.org/10.1002/..
 
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8

Discovery of a Potent, Cell Penetrant, and Selective p300/C..:

Humphreys, Philip G. ; Bamborough, Paul ; Chung, Chun-wa...
Journal of Medicinal Chemistry.  60 (2017)  2 - p. 695-709 , 2017
Link: https://doi.org/10.1021/..
 
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9

Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of ..:

Westaway, Susan M. ; Preston, Alex G. S. ; Barker, Michael D....
Journal of Medicinal Chemistry.  59 (2016)  4 - p. 1370-1387 , 2016
Link: https://doi.org/10.1021/..
 
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10

Cell Penetrant Inhibitors of the KDM4 and KDM5 Families of ..:

Westaway, Susan M. ; Preston, Alex G. S. ; Barker, Michael D....
Journal of Medicinal Chemistry.  59 (2016)  4 - p. 1357-1369 , 2016
Link: https://doi.org/10.1021/..
 
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11

Discovery of GSK143, a highly potent, selective and orally ..:

Liddle, John ; Atkinson, Francis L. ; Barker, Michael D....
Bioorganic & Medicinal Chemistry Letters.  21 (2011)  20 - p. 6188-6194 , 2011
Link: https://doi.org/10.1016/..
 
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12

Discovery of GSK345931A: An EP1 receptor antagonist with ef..:

Hall, Adrian ; Brown, Susan H. ; Budd, Christopher...
Bioorganic & Medicinal Chemistry Letters.  19 (2009)  2 - p. 497-501 , 2009
Link: https://doi.org/10.1016/..
 
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13

Discovery of brain penetrant, soluble, pyrazole amide EP1 r..:

Hall, Adrian ; Billinton, Andy ; Bristow, Alan K....
Bioorganic & Medicinal Chemistry Letters.  18 (2008)  14 - p. 4027-4032 , 2008
Link: https://doi.org/10.1016/..
 
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14

Non-acidic pyrazole EP1 receptor antagonists with in vivo a..:

Hall, Adrian ; Billinton, Andy ; Brown, Susan H....
Bioorganic & Medicinal Chemistry Letters.  18 (2008)  11 - p. 3392-3399 , 2008
Link: https://doi.org/10.1016/..
 
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15

Degradation by Design: New Cyclin K Degraders from Old CDK ..:

Thomas, Katie L ; Bouguenina, Habib ; Miller, Daniel S. J...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC10804372/.  , 2024
Link: http://www.ncbi.nlm.nih...
 
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