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Holly Koblish
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1

Discovery of Potent and Selective Inhibitors of Wild-Type a..:

Shvartsbart, Artem ; Roach, Jeremy J. ; Witten, Michael R....
Journal of Medicinal Chemistry.  65 (2022)  22 - p. 15433-15442 , 2022
Link: https://doi.org/10.1021/..
 
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2

Discovery of Pemigatinib: A Potent and Selective Fibroblast..:

Wu, Liangxing ; Zhang, Colin ; He, Chunhong...
Journal of Medicinal Chemistry.  64 (2021)  15 - p. 10666-10679 , 2021
Link: https://doi.org/10.1021/..
 
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3

INCB054828 (pemigatinib), a potent and selective inhibitor ..:

Liu, Phillip C. C. ; Koblish, Holly ; Wu, Liangxing...
PLOS ONE.  15 (2020)  4 - p. e0231877 , 2020
Link: https://doi.org/10.1371/..
 
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4

A Potent and Selective Dual Inhibitor of AXL and MERTK Poss..:

Rios-Doria, Jonathan ; Favata, Margaret ; Lasky, Kerri...
Frontiers in Oncology.  10 (2020)  - p. , 2020
Link: https://doi.org/10.3389/..
 
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5

Hematopoietic cytokines mediate resistance to targeted ther..:

Sung, Pamela J. ; Sugita, Mayumi ; Koblish, Holly..
Blood Advances.  3 (2019)  7 - p. 1061-1072 , 2019
Link: https://doi.org/10.1182/..
 
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6

Preclinical characterization of INCB053914, a novel pan-PIM..:

Koblish, Holly ; Li, Yun-long ; Shin, Niu...
PLOS ONE.  13 (2018)  6 - p. e0199108 , 2018
Link: https://doi.org/10.1371/..
 
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7

Progress in the Development of Agents to Control the Cell C..:

, In: Topics in Medicinal Chemistry; Cancer,
Moriarty, Kevin J. ; Koblish, Holly ; Johnson, Dana L.. - p. 207-291 , 2007
Link: https://doi.org/10.1007/..
 
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8

Characterization of INCB086550: A Potent and Novel Small-Mo..:

Koblish, Holly K. ; Wu, Liangxing ; Wang, Liang-Chuan S....
Cancer Discovery.  12 (2022)  6 - p. 1482-1499 , 2022
Link: https://doi.org/10.1158/..
 
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9

Characterization of human cancer xenografts in humanized mi..:

Rios-Doria, Jonathan ; Stevens, Christina ; Maddage, Christopher..
Journal for ImmunoTherapy of Cancer.  8 (2020)  1 - p. e000416 , 2020
Link: https://doi.org/10.1136/..
 
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10

INCB050465 (Parsaclisib), a Novel Next-Generation Inhibitor..:

Yue, Eddy W. ; Li, Yun-Long ; Douty, Brent...
ACS Medicinal Chemistry Letters.  10 (2019)  11 - p. 1554-1560 , 2019
Link: https://doi.org/10.1021/..
 
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11

The pan-PIM inhibitor INCB053914 displays potent synergy in..:

Mazzacurati, Lucia ; Collins, Robert J. ; Pandey, Garima...
Blood Advances.  3 (2019)  22 - p. 3503-3514 , 2019
Link: https://doi.org/10.1182/..
 
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12

INCB24360 (Epacadostat), a Highly Potent and Selective Indo..:

Yue, Eddy W. ; Sparks, Richard ; Polam, Padmaja...
ACS Medicinal Chemistry Letters.  8 (2017)  5 - p. 486-491 , 2017
Link: https://doi.org/10.1021/..
 
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13

Discovery of Potent Competitive Inhibitors of Indoleamine 2..:

Yue, Eddy W. ; Douty, Brent ; Wayland, Brian...
Journal of Medicinal Chemistry.  52 (2009)  23 - p. 7364-7367 , 2009
Link: https://doi.org/10.1021/..
 
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14

Enhanced pharmacokinetic properties of 1,4-benzodiazepine-2..:

Parks, Daniel J. ; LaFrance, Louis V. ; Calvo, Raul R....
Bioorganic & Medicinal Chemistry Letters.  16 (2006)  12 - p. 3310-3314 , 2006
Link: https://doi.org/10.1016/..
 
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15

Enantiomerically pure 1,4-benzodiazepine-2,5-diones as Hdm2..:

Marugan, Juan Jose ; Leonard, Kristi ; Raboisson, Pierre...
Bioorganic & Medicinal Chemistry Letters.  16 (2006)  12 - p. 3115-3120 , 2006
Link: https://doi.org/10.1016/..
 
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