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1
Discovery of Novel Oxazepine Derivatives as Akt/ROCK Inhibi..:
Che, Jinxin ; Bing, Shaowei ; Lu, Jialiang...
Journal of Medicinal Chemistry. 66 (2023) 19 - p. 13530-13555 , 2023
Journal of Medicinal Chemistry. 66 (2023) 19 - p. 13530-13555 , 2023
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2
Discovery of N-((3S,4S)-4-(3,4-Difluorophenyl)piperidin-3-y..:
Che, Jinxin ; Dai, Xiaoyang ; Gao, Jian...
Journal of Medicinal Chemistry. 64 (2021) 16 - p. 12163-12180 , 2021
Journal of Medicinal Chemistry. 64 (2021) 16 - p. 12163-12180 , 2021
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3
Discovery of 5,6-Bis(4-methoxy-3-methylphenyl)pyridin-2-ami..:
Che, Jinxin ; Jin, Zegao ; Yan, Fangjie...
Journal of Medicinal Chemistry. 64 (2021) 12 - p. 8621-8643 , 2021
Journal of Medicinal Chemistry. 64 (2021) 12 - p. 8621-8643 , 2021
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4
Development of differentiation modulators and targeted agen..:
Jin, Zegao ; Lu, Yang ; Wu, Yizhe..
European Journal of Medicinal Chemistry. 207 (2020) - p. 112818 , 2020
European Journal of Medicinal Chemistry. 207 (2020) - p. 112818 , 2020
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5
Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as..:
Dong, Xiaowu ; Zhan, Wenhu ; Zhao, Mengting...
Journal of Medicinal Chemistry. 62 (2019) 15 - p. 7264-7288 , 2019
Journal of Medicinal Chemistry. 62 (2019) 15 - p. 7264-7288 , 2019
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6
Combination therapy with p53–MDM2 binding inhibitors for ma..:
Jin, Zegao ; Shen, Jianfeng ; He, Jingyao.
Medicinal Chemistry Research. 24 (2014) 4 - p. 1369-1379 , 2014
Medicinal Chemistry Research. 24 (2014) 4 - p. 1369-1379 , 2014
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7
Discovery of N ‑((3 S ,4 S )‑4-(3,4-Difluorophenyl)piperidi..:
Jinxin Che (791250) ; Xiaoyang Dai (2246731) ; Jian Gao (307118)...
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142492. , 2021
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142492. , 2021
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8
Discovery of N ‑((3 S ,4 S )‑4-(3,4-Difluorophenyl)piperidi..:
Jinxin Che (791250) ; Xiaoyang Dai (2246731) ; Jian Gao (307118)...
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142483. , 2021
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142483. , 2021
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9
Discovery of N ‑((3 S ,4 S )‑4-(3,4-Difluorophenyl)piperidi..:
Jinxin Che (791250) ; Xiaoyang Dai (2246731) ; Jian Gao (307118)...
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142474. , 2021
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142474. , 2021
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10
Discovery of 5,6-Bis(4-methoxy-3-methylphenyl)pyridin-2-ami..:
Jinxin Che (791250) ; Zegao Jin (7037933) ; Fangjie Yan (10904583)...
https://figshare.com/articles/journal_contribution/Discovery_of_5_6-Bis_4-methoxy-3-methylphenyl_pyridin-2-amine_as_a_WSB1_Degrader_to_Inhibit_Cancer_Cell_Metastasis/14710746. , 2021
https://figshare.com/articles/journal_contribution/Discovery_of_5_6-Bis_4-methoxy-3-methylphenyl_pyridin-2-amine_as_a_WSB1_Degrader_to_Inhibit_Cancer_Cell_Metastasis/14710746. , 2021
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11
Discovery of N ‑((3 S ,4 S )‑4-(3,4-Difluorophenyl)piperidi..:
Jinxin Che (791250) ; Xiaoyang Dai (2246731) ; Jian Gao (307118)...
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142486. , 2021
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142486. , 2021
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12
Discovery of N ‑((3 S ,4 S )‑4-(3,4-Difluorophenyl)piperidi..:
Jinxin Che (791250) ; Xiaoyang Dai (2246731) ; Jian Gao (307118)...
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142477. , 2021
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142477. , 2021
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13
Discovery of N ‑((3 S ,4 S )‑4-(3,4-Difluorophenyl)piperidi..:
Jinxin Che (791250) ; Xiaoyang Dai (2246731) ; Jian Gao (307118)...
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142480. , 2021
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142480. , 2021
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14
Discovery of N ‑((3 S ,4 S )‑4-(3,4-Difluorophenyl)piperidi..:
Jinxin Che (791250) ; Xiaoyang Dai (2246731) ; Jian Gao (307118)...
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142489. , 2021
https://figshare.com/articles/dataset/Discovery_of_i_N_i_3_i_S_i_4_i_S_i_4-_3_4-Difluorophenyl_piperidin-3-yl_-2-fluoro-4-_1-methyl_1_i_H_i_pyrazol-5-yl_benzamide_Hu7691_a_Potent_and_Selective_Akt_Inhibitor_That_Enables_Decrease_of_Cutaneous_Toxicity/15142489. , 2021
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15
Discovery of 5,6-Bis(4-methoxy-3-methylphenyl)pyridin-2-ami..:
Jinxin Che (791250) ; Zegao Jin (7037933) ; Fangjie Yan (10904583)...
https://figshare.com/articles/dataset/Discovery_of_5_6-Bis_4-methoxy-3-methylphenyl_pyridin-2-amine_as_a_WSB1_Degrader_to_Inhibit_Cancer_Cell_Metastasis/14710749. , 2021
https://figshare.com/articles/dataset/Discovery_of_5_6-Bis_4-methoxy-3-methylphenyl_pyridin-2-amine_as_a_WSB1_Degrader_to_Inhibit_Cancer_Cell_Metastasis/14710749. , 2021