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Kargman, Stacia
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1

Addition to "Scaffold Hopping and Optimization of Small Mol..:

Sun, Shan ; Fushimi, Makoto ; Rossetti, Thomas...
Journal of Chemical Information and Modeling.  64 (2024)  3 - p. 1106-1106 , 2024
Link: https://doi.org/10.1021/..
 
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2

Lead Optimization of Small Molecule ENL YEATS Inhibitors to..:

Michino, Mayako ; Khan, Tanweer A. ; Miller, Michael W....
ACS Medicinal Chemistry Letters.  15 (2024)  4 - p. 524-532 , 2024
Link: https://doi.org/10.1021/..
 
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3

Scaffold Hopping and Optimization of Small Molecule Soluble..:

Sun, Shan ; Fushimi, Makoto ; Rossetti, Thomas...
Journal of Chemical Information and Modeling.  63 (2023)  9 - p. 2828-2841 , 2023
Link: https://doi.org/10.1021/..
 
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4

Design, Synthesis, and Pharmacological Evaluation of Second..:

Miller, Michael ; Rossetti, Thomas ; Ferreira, Jacob...
Journal of Medicinal Chemistry.  65 (2022)  22 - p. 15208-15226 , 2022
Link: https://doi.org/10.1021/..
 
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5

Small-Molecule Inhibition of the Acyl-Lysine Reader ENL as ..:

Liu, Yiman ; Li, Qinglan ; Alikarami, Fatemeh...
Cancer Discovery.  12 (2022)  11 - p. 2684-2709 , 2022
Link: https://doi.org/10.1158/..
 
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6

A Chemical Strategy toward Novel Brain-Penetrant EZH2 Inhib..:

Liang, Rui ; Tomita, Daisuke ; Sasaki, Yusuke...
ACS Medicinal Chemistry Letters.  13 (2022)  3 - p. 377-387 , 2022
Link: https://doi.org/10.1021/..
 
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7

Discovery of TDI-10229: A Potent and Orally Bioavailable In..:

Fushimi, Makoto ; Buck, Hannes ; Balbach, Melanie...
ACS Medicinal Chemistry Letters.  12 (2021)  8 - p. 1283-1287 , 2021
Link: https://doi.org/10.1021/..
 
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8

Inhibition of 3-phosphoglycerate dehydrogenase (PHGDH) by i..:

Mullarky, Edouard ; Xu, Jiayi ; Robin, Anita D....
Bioorganic & Medicinal Chemistry Letters.  29 (2019)  17 - p. 2503-2510 , 2019
Link: https://doi.org/10.1016/..
 
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9

Antibacterial small molecules targeting the conserved TOPRI..:

Walker, Scott S. ; Labroli, Marc ; Painter, Ronald E....
PLOS ONE.  12 (2017)  7 - p. e0180965 , 2017
Link: https://doi.org/10.1371/..
 
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10

Discovery of MK-8831, A Novel Spiro-Proline Macrocycle as a..:

Neelamkavil, Santhosh F. ; Agrawal, Sony ; Bara, Thomas...
ACS Medicinal Chemistry Letters.  7 (2015)  1 - p. 111-116 , 2015
Link: https://doi.org/10.1021/..
 
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11

Stearoyl-CoA desaturase inhibition blocks formation of hepa..:

Lyn, Rodney K. ; Singaravelu, Ragunath ; Kargman, Stacia...
Scientific Reports.  4 (2014)  1 - p. , 2014
Link: https://doi.org/10.1038/..
 
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12

Discovery of MK‐8742: An HCV NS5A Inhibitor with Broad Geno..:

Coburn, Craig A. ; Meinke, Peter T. ; Chang, Wei...
ChemMedChem.  8 (2013)  12 - p. 1930-1940 , 2013
Link: https://doi.org/10.1002/..
 
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13

Murgocil is a Highly Bioactive Staphylococcal-Specific Inhi..:

Mann, Paul A. ; Müller, Anna ; Xiao, Li...
ACS Chemical Biology.  8 (2013)  11 - p. 2442-2451 , 2013
Link: https://doi.org/10.1021/..
 
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14

The identification of 4,7-disubstituted naphthoic acid deri..:

Gauthier, Jacques Yves ; Belley, Michel ; Deschênes, Denis...
Bioorganic & Medicinal Chemistry Letters.  21 (2011)  10 - p. 2836-2839 , 2011
Link: https://doi.org/10.1016/..
 
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15

Applying the pro-drug approach to afford highly bioavailabl..:

Robichaud, Joël ; Fournier, Jean-François ; Gagné, Sébastien...
Bioorganic & Medicinal Chemistry Letters.  21 (2011)  14 - p. 4366-4368 , 2011
Link: https://doi.org/10.1016/..
 
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