Nagaraja, Raj
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1

Discovery of AG-270, a First-in-Class Oral MAT2A Inhibitor ..:

Konteatis, Zenon ; Travins, Jeremy ; Gross, Stefan...
Journal of Medicinal Chemistry.  64 (2021)  8 - p. 4430-4449 , 2021
 
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2

Vorasidenib (AG-881): A First-in-Class, Brain-Penetrant Dua..:

Konteatis, Zenon ; Artin, Erin ; Nicolay, Brandon...
ACS Medicinal Chemistry Letters.  11 (2020)  2 - p. 101-107 , 2020
 
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3

Effect of Mild and Moderate Hepatic Impairment on the Pharm..:

Fan, Bin ; Dai, David ; Cohen, Marvin...
Clinical Pharmacology in Drug Development.  10 (2020)  1 - p. 99-109 , 2020
 
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7

Exploration of cathepsin S inhibitors characterized by a tr..:

Moss, Neil ; Xiong, Zhaoming ; Burke, Mike...
Bioorganic & Medicinal Chemistry Letters.  22 (2012)  23 - p. 7189-7193 , 2012
 
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8

A new class of 5-HT2B antagonists possesses favorable poten..:

Moss, Neil ; Choi, Younggi ; Cogan, Derek...
Bioorganic & Medicinal Chemistry Letters.  19 (2009)  8 - p. 2206-2210 , 2009
 
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13

Discovery of AG-270, a First-in-Class Oral MAT2A Inhibitor ..:

Zenon Konteatis (2236249) ; Jeremy Travins (4810641) ; Stefan Gross (673951)...
https://figshare.com/articles/journal_contribution/Discovery_of_AG-270_a_First-in-Class_Oral_MAT2A_Inhibitor_for_the_Treatment_of_Tumors_with_Homozygous_i_MTAP_i_Deletion/14387567.  , 2021
 
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14

Discovery of AG-270, a First-in-Class Oral MAT2A Inhibitor ..:

Zenon Konteatis (2236249) ; Jeremy Travins (4810641) ; Stefan Gross (673951)...
https://figshare.com/articles/dataset/Discovery_of_AG-270_a_First-in-Class_Oral_MAT2A_Inhibitor_for_the_Treatment_of_Tumors_with_Homozygous_i_MTAP_i_Deletion/14387570.  , 2021
 
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