I agree that this site is using cookies. You can find further informations here.
X
Nasveschuk, Christopher G
37  results:
Search for persons X
?
1

Mechanistic insights into a heterobifunctional degrader-ind..:

Hao, Qi ; Rathinaswamy, Manoj K. ; Klinge, Kelly L....
Communications Chemistry.  7 (2024)  1 - p. , 2024
Link: https://doi.org/10.1038/..
 
?
2

GNE-064: A Potent, Selective, and Orally Bioavailable Chemi..:

Taylor, Alexander M. ; Bailey, Chris ; Belmont, Lisa D....
Journal of Medicinal Chemistry.  65 (2022)  16 - p. 11177-11186 , 2022
Link: https://doi.org/10.1021/..
 
?
3

A Method for Determining the Kinetics of Small-Molecule-Ind..:

Vieux, Ellen F. ; Agafonov, Roman V. ; Emerson, Lydia...
SLAS Discovery.  26 (2021)  4 - p. 547-559 , 2021
Link: https://doi.org/10.1177/..
 
?
4

Structural Characterization of Degrader-Induced Ternary Com..:

Eron, Scott J. ; Huang, Hongwei ; Agafonov, Roman V....
ACS Chemical Biology.  16 (2021)  11 - p. 2228-2243 , 2021
Link: https://doi.org/10.1021/..
 
?
5

Evaluation of the Small-molecule BRD4 Degrader CFT-2718 in ..:

Sun, Danlin ; Nikonova, Anna S. ; Zhang, Peishan...
Molecular Cancer Therapeutics.  20 (2021)  8 - p. 1367-1377 , 2021
Link: https://doi.org/10.1158/..
 
?
6

GNE-371, a Potent and Selective Chemical Probe for the Seco..:

Wang, Shumei ; Tsui, Vickie ; Crawford, Terry D....
Journal of Medicinal Chemistry.  61 (2018)  20 - p. 9301-9315 , 2018
Link: https://doi.org/10.1021/..
 
?
7

Inhibition of bromodomain-containing protein 9 for the prev..:

Crawford, Terry D. ; Vartanian, Steffan ; Côté, Alexandre...
Bioorganic & Medicinal Chemistry Letters.  27 (2017)  15 - p. 3534-3541 , 2017
Link: https://doi.org/10.1016/..
 
?
8

GNE-886: A Potent and Selective Inhibitor of the Cat Eye Sy..:

Crawford, Terry D. ; Audia, James E. ; Bellon, Steve...
ACS Medicinal Chemistry Letters.  8 (2017)  7 - p. 737-741 , 2017
Link: https://doi.org/10.1021/..
 
?
9

Fragment-Based Discovery of a Selective and Cell-Active Ben..:

Taylor, Alexander M. ; Côté, Alexandre ; Hewitt, Michael C....
ACS Medicinal Chemistry Letters.  7 (2016)  5 - p. 531-536 , 2016
Link: https://doi.org/10.1021/..
 
?
10

Identification of (R)-N-((4-Methoxy-6-methyl-2-oxo-1,2-dihy..:

Vaswani, Rishi G. ; Gehling, Victor S. ; Dakin, Les A....
Journal of Medicinal Chemistry.  59 (2016)  21 - p. 9928-9941 , 2016
Link: https://doi.org/10.1021/..
 
?
11

Diving into the Water: Inducible Binding Conformations for ..:

Crawford, Terry D. ; Tsui, Vickie ; Flynn, E. Megan...
Journal of Medicinal Chemistry.  59 (2016)  11 - p. 5391-5402 , 2016
Link: https://doi.org/10.1021/..
 
?
12

Identification of a Benzoisoxazoloazepine Inhibitor (CPI-06..:

Albrecht, Brian K. ; Gehling, Victor S. ; Hewitt, Michael C....
Journal of Medicinal Chemistry.  59 (2016)  4 - p. 1330-1339 , 2016
Link: https://doi.org/10.1021/..
 
?
13

Corrigendum to "Development of methyl isoxazoleazepines as ..:

Hewitt, Michael C. ; Leblanc, Yves ; Gehling, Victor S....
Bioorganic & Medicinal Chemistry Letters.  25 (2015)  17 - p. 3755 , 2015
Link: https://doi.org/10.1016/..
 
?
14

Discovery, design, and synthesis of indole-based EZH2 inhib..:

Gehling, Victor S. ; Vaswani, Rishi G. ; Nasveschuk, Christopher G....
Bioorganic & Medicinal Chemistry Letters.  25 (2015)  17 - p. 3644-3649 , 2015
Link: https://doi.org/10.1016/..
 
?
15

Development of methyl isoxazoleazepines as inhibitors of BE:

Hewitt, Michael C. ; Leblanc, Yves ; Gehling, Victor S....
Bioorganic & Medicinal Chemistry Letters.  25 (2015)  9 - p. 1842-1848 , 2015
Link: https://doi.org/10.1016/..
 
1-15