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Niosi, Mark
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1

P-GP limits rodent oral absoprtion of protacs:

Steyn, Stefanus ; Niosi, Mark ; Kimoto, Emi.
Drug Metabolism and Pharmacokinetics.  55 (2024)  - p. 100978 , 2024
Link: https://doi.org/10.1016/..
 
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2

Attempting to Unmask the Inhibition of Sulfotransferase 1E1..:

Rodrigues, David ; Niosi, Mark ; Eng, Heather...
The Journal of Clinical Pharmacology.  63 (2023)  8 - p. 875-879 , 2023
Link: https://doi.org/10.1002/..
 
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3

Discovery of Ervogastat (PF-06865571): A Potent and Selecti..:

Futatsugi, Kentaro ; Cabral, Shawn ; Kung, Daniel W....
Journal of Medicinal Chemistry.  65 (2022)  22 - p. 15000-15013 , 2022
Link: https://doi.org/10.1021/..
 
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4

Optimizing the Benefit/Risk of Acetyl-CoA Carboxylase Inhib..:

Huard, Kim ; Smith, Aaron C. ; Cappon, Gregg...
Journal of Medicinal Chemistry.  63 (2020)  19 - p. 10879-10896 , 2020
Link: https://doi.org/10.1021/..
 
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5

P100 - In vitro evaluation of UDP-glucuronosyltransferase (..:

Lapham, Kimberly ; Ferguson, Nicholas ; Novak, Jonathan..
Drug Metabolism and Pharmacokinetics.  35 (2020)  1 - p. S52-S53 , 2020
Link: https://doi.org/10.1016/..
 
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6

In vitro characterization of ertugliflozin glucuronidation:

Lapham, Kimberly ; Callegari, Ernesto ; Lin, Jian...
Drug Metabolism and Pharmacokinetics.  34 (2019)  1 - p. S24 , 2019
Link: https://doi.org/10.1016/..
 
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7

Novel in vitro method to predict in vivo liver-to-plasma un..:

Di, Li ; Riccardi, Keith ; Li, Zhenhong...
Drug Metabolism and Pharmacokinetics.  33 (2018)  1 - p. S91 , 2018
Link: https://doi.org/10.1016/..
 
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8

2-Aminopyridine-Based Mitogen-Activated Protein Kinase Kina..:

Dow, Robert L. ; Ammirati, Mark ; Bagley, Scott W....
Journal of Medicinal Chemistry.  61 (2018)  7 - p. 3114-3125 , 2018
Link: https://doi.org/10.1021/..
 
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9

Delineating the role of cooperativity in the design of pote..:

Zorba, Adelajda ; Nguyen, Chuong ; Xu, Yingrong...
Proceedings of the National Academy of Sciences of the United States of America.  115 (2018)  31 - p. E7285-E7292 , 2018
Link: https://www.jstor.org/st..
 
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10

Delineating the role of cooperativity in the design of pote..:

Zorba, Adelajda ; Nguyen, Chuong ; Xu, Yingrong...
Proceedings of the National Academy of Sciences.  115 (2018)  31 - p. , 2018
Link: https://doi.org/10.1073/..
 
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11

Enantioselective glucuronidation of lorazepam by UGT2B7 and..:

Lin, Jian ; Niosi, Mark ; Lapham, Kimberly..
Drug Metabolism and Pharmacokinetics.  33 (2018)  1 - p. S27 , 2018
Link: https://doi.org/10.1016/..
 
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12

Optimization of a Dicarboxylic Series for in Vivo Inhibitio..:

Huard, Kim ; Gosset, James R. ; Montgomery, Justin I....
Journal of Medicinal Chemistry.  59 (2016)  3 - p. 1165-1175 , 2016
Link: https://doi.org/10.1021/..
 
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13

Discovery and Optimization of Imidazopyridine-Based Inhibit..:

Futatsugi, Kentaro ; Kung, Daniel W. ; Orr, Suvi T. M....
Journal of Medicinal Chemistry.  58 (2015)  18 - p. 7173-7185 , 2015
Link: https://doi.org/10.1021/..
 
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14

Corrigendum to "Novel monobactams utilizing a siderophore u..:

Mitton-Fry, Mark J. ; Arcari, Joel T. ; Brown, Matthew F....
Bioorganic & Medicinal Chemistry Letters.  25 (2015)  18 - p. 4029 , 2015
Link: https://doi.org/10.1016/..
 
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15

Discovery and characterization of novel inhibitors of the s..:

Huard, Kim ; Brown, Janice ; Jones, Jessica C....
Scientific Reports.  5 (2015)  1 - p. , 2015
Link: https://doi.org/10.1038/..
 
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