I agree that this site is using cookies. You can find further informations here.
X
Rombouts, Frederik J. R.
374  results:
Search for persons X
?
1

Discovery of an Oral, Beyond-Rule-of-Five Mcl-1 Protein–Pro..:

Romanov-Michailidis, Fedor ; Hsiao, Chien-Chi ; Urner, Lorenz M....
Journal of Medicinal Chemistry.  66 (2023)  9 - p. 6122-6148 , 2023
Link: https://doi.org/10.1021/..
 
?
2

Macrocyclic Carbon-Linked Pyrazoles As Novel Inhibitors of ..:

Demin, Samuël ; Peschiulli, Aldo ; Velter, Adriana I....
ACS Medicinal Chemistry Letters.  14 (2023)  7 - p. 955-961 , 2023
Link: https://doi.org/10.1021/..
 
?
3

Modulating physicochemical properties of tetrahydropyridine..:

Rombouts, Frederik J.R. ; Hsiao, Chien-Chi ; Bache, Solène...
European Journal of Medicinal Chemistry.  228 (2022)  - p. 114028 , 2022
Link: https://doi.org/10.1016/..
 
?
4

JNJ-67569762, A 2-Aminotetrahydropyridine-Based Selective B..:

Rombouts, Frederik J. R. ; Kusakabe, Ken-ichi ; Alexander, Richard...
Journal of Medicinal Chemistry.  64 (2021)  19 - p. 14175-14191 , 2021
Link: https://doi.org/10.1021/..
 
?
5

Structure-Based Approaches to Improving Selectivity through..:

Fujimoto, Kazuki ; Yoshida, Shuhei ; Tadano, Genta...
Journal of Medicinal Chemistry.  64 (2021)  6 - p. 3075-3085 , 2021
Link: https://doi.org/10.1021/..
 
?
6

A Brain-Penetrant and Bioavailable Pyrazolopiperazine BACE1..:

Peschiulli, Aldo ; Oehlrich, Daniel ; Van Gool, Michiel...
ACS Medicinal Chemistry Letters.  13 (2021)  1 - p. 76-83 , 2021
Link: https://doi.org/10.1021/..
 
?
7

Discovery of Extremely Selective Fused Pyridine-Derived β-S..:

Ueno, Tatsuhiko ; Matsuoka, Eriko ; Asada, Naoya...
Journal of Medicinal Chemistry.  64 (2021)  19 - p. 14165-14174 , 2021
Link: https://doi.org/10.1021/..
 
?
8

Clinical evaluation of [18F] JNJ-64326067, a novel candidat..:

Schmidt, Mark E. ; Janssens, Luc ; Moechars, Diederik...
European Journal of Nuclear Medicine and Molecular Imaging.  47 (2020)  13 - p. 3176-3185 , 2020
Link: https://doi.org/10.1007/..
 
?
9

Correction to Discovery of N-(4-[18F]Fluoro-5-methylpyridin..:

Rombouts, Frederik J. R. ; Declercq, Lieven ; Andrés, José-Ignacio...
Journal of Medicinal Chemistry.  63 (2020)  4 - p. 1775-1775 , 2020
Link: https://doi.org/10.1021/..
 
?
10

Evaluation of a Series of β-Secretase 1 Inhibitors Containi..:

Oehlrich, Daniel ; Peschiulli, Aldo ; Tresadern, Gary...
ACS Medicinal Chemistry Letters.  10 (2019)  8 - p. 1159-1165 , 2019
Link: https://doi.org/10.1021/..
 
?
11

Discovery of N-(4-[18F]Fluoro-5-methylpyridin-2-yl)isoquino..:

Rombouts, Frederik J. R. ; Declercq, Lieven ; Andrés, José-Ignacio...
Journal of Medicinal Chemistry.  62 (2019)  6 - p. 2974-2987 , 2019
Link: https://doi.org/10.1021/..
 
?
12

Optimization of 1,4-Oxazine β-Secretase 1 (BACE1) Inhibitor..:

Gijsen, Harrie J. M. ; Alonso de Diego, Sergio A. ; De Cleyn, Michel...
Journal of Medicinal Chemistry.  61 (2018)  12 - p. 5292-5303 , 2018
Link: https://doi.org/10.1021/..
 
?
13

Correction to Optimization of 1,4-Oxazine β-Secretase 1 (BA..:

Gijsen, Harrie J. M. ; Alonso de Diego, Sergio A. ; De Cleyn, Michel...
Journal of Medicinal Chemistry.  61 (2018)  24 - p. 11415-11415 , 2018
Link: https://doi.org/10.1021/..
 
?
14

Discovery of N-(Pyridin-4-yl)-1,5-naphthyridin-2-amines as ..:

Rombouts, Frederik J. R. ; Andrés, José-Ignacio ; Ariza, Manuela...
Journal of Medicinal Chemistry.  60 (2017)  4 - p. 1272-1291 , 2017
Link: https://doi.org/10.1021/..
 
?
15

Industrial medicinal chemistry insights: neuroscience hit g..:

Tresadern, Gary ; Rombouts, Frederik J.R. ; Oehlrich, Daniel..
Drug Discovery Today.  22 (2017)  10 - p. 1478-1488 , 2017
Link: https://doi.org/10.1016/..
 
1-15