E-LIB Suche - Ergebnisse für: Scheepstra, Marcel

1

Development of Potent Mcl-1 Inhibitors: Structural Investig..:

Hekking, Koen F. W. ; Maroto, Sergio ; van Kekem, Kees...
Journal of Medicinal Chemistry. 67 (2024) 4 - p. 3039-3065 , 2024

Link: https://doi.org/10.1021/..

2

Ligand-Based Design of Allosteric Retinoic Acid Receptor-Re..:

Meijer, Femke A. ; Doveston, Richard G. ; de Vries, Rens M.J.M....
Journal of Medicinal Chemistry. 63 (2019) 1 - p. 241-259 , 2019

Link: https://doi.org/10.1021/..

3

Bivalent Ligands for Protein Degradation in Drug Discovery:

Scheepstra, Marcel ; Hekking, Koen F.W. ; van Hijfte, Luc.
Computational and Structural Biotechnology Journal. 17 (2019) - p. 160-176 , 2019

Link: https://doi.org/10.1016/..

4

Designed Spiroketal Protein Modulation:

Scheepstra, Marcel ; Andrei, Sebastian A. ; Unver, M. Yagiz...
Angewandte Chemie. 129 (2017) 20 - p. 5572-5576 , 2017

Link: https://doi.org/10.1002/..

5

Ligand Dependent Switch from RXR Homo- to RXR-NURR1 Heterod..:

Scheepstra, Marcel ; Andrei, Sebastian A. ; de Vries, Rens M. J. M....
ACS Chemical Neuroscience. 8 (2017) 9 - p. 2065-2077 , 2017

Link: https://doi.org/10.1021/..

6

Designed Spiroketal Protein Modulation:

Scheepstra, Marcel ; Andrei, Sebastian A. ; Unver, M. Yagiz...
Angewandte Chemie International Edition. 56 (2017) 20 - p. 5480-5484 , 2017

Link: https://doi.org/10.1002/..

7

Chiral Dihydrobenzofuran Acids Show Potent Retinoid X Recep..:

Sundén, Henrik ; Schäfer, Anja ; Scheepstra, Marcel...
Journal of Medicinal Chemistry. 59 (2016) 3 - p. 1232-1238 , 2016

Link: https://doi.org/10.1021/..

8

Identification of an allosteric binding site for RORγt inhi..:

Scheepstra, Marcel ; Leysen, Seppe ; van Almen, Geert C....
Nature Communications. 6 (2015) 1 - p. , 2015

Link: https://doi.org/10.1038/..

9

Subtype-Specific Modulation of Estrogen Receptor–Coactivato..:

Tharun, Inga M. ; Nieto, Lidia ; Haase, Christian...
ACS Chemical Biology. 10 (2014) 2 - p. 475-484 , 2014

Link: https://doi.org/10.1021/..

10

A Natural‐Product Switch for a Dynamic Protein Interface:

Scheepstra, Marcel ; Nieto, Lidia ; Hirsch, Anna K. H....
Angewandte Chemie International Edition. 53 (2014) 25 - p. 6443-6448 , 2014

Link: https://doi.org/10.1002/..

11

A Natural‐Product Switch for a Dynamic Protein Interface:

Scheepstra, Marcel ; Nieto, Lidia ; Hirsch, Anna K. H....
Angewandte Chemie. 126 (2014) 25 - p. 6561-6566 , 2014

Link: https://doi.org/10.1002/..

12

Cucurbit[8]uril induced heterodimerization of methylviologe..:

Uhlenheuer, Dana A. ; Young, Jacqui F. ; Nguyen, Hoang D...
Chemical Communications. 47 (2011) 24 - p. 6798 , 2011

Link: https://doi.org/10.1039/..

13

Ligand-Based Design of Allosteric Retinoic Acid Receptor-Re..:

Meijer, Femke A ; Doveston, Richard G ; de Vries, Rens M. J. M...
info:eu-repo/semantics/altIdentifier/issn/0022-2623. , 2020

Link: https://bib-pubdb1.desy...

14

Ligand-based design of allosteric retinoic acid receptor-re..:

Meijer, Femke A ; Doveston, Richard G ; de Vries, Rens M J M...
Meijer , F A , Doveston , R G , de Vries , R M J M , Vos , G M , Vos , A A A , Leysen , S , Scheepstra , M , Ottmann , C , Milroy , L-G & Brunsveld , L 2020 , ' Ligand-based design of allosteric retinoic acid receptor-related orphan receptor γt (RORγt) inverse agonists ' , Journal of Medicinal Chemistry , vol. 63 , no. 1 , pp. 241-259 . https://doi.org/10.1021/acs.jmedchem.9b01372. , 2020

Link: https://research.tue.nl/..

15

Ligand-Based Design of Allosteric Retinoic Acid Receptor-Re..:

Meijer, Femke A ; Doveston, Richard G ; de Vries, Rens M.J.M...
http://www.ncbi.nlm.nih.gov/pmc/articles/PMC6956242/. , 2019

Link: http://www.ncbi.nlm.nih...