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Somers, Don O.
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1

Covalent targeting of non-cysteine residues in PI4KIIIβ:

Cosgrove, Brett ; Grant, Emma K. ; Bertrand, Sophie...
RSC Chemical Biology.  4 (2023)  12 - p. 1111-1122 , 2023
Link: https://doi.org/10.1039/..
 
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2

A knowledge-based, structural-aided discovery of a novel cl..:

Schulte, Christie A. ; Deaton, David N. ; Diaz, Elsie...
Bioorganic & Medicinal Chemistry Letters.  47 (2021)  - p. 128113 , 2021
Link: https://doi.org/10.1016/..
 
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3

Exploring Ligand Stability in Protein Crystal Structures Us..:

Fusani, Lucia ; Palmer, David S. ; Somers, Don O..
Journal of Chemical Information and Modeling.  60 (2020)  3 - p. 1528-1539 , 2020
Link: https://doi.org/10.1021/..
 
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4

Optimisation of a novel series of potent and orally bioavai..:

Garton, Neil S. ; Barker, Michael D. ; Davis, Rob P....
Bioorganic & Medicinal Chemistry Letters.  26 (2016)  19 - p. 4606-4612 , 2016
Link: https://doi.org/10.1016/..
 
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5

Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replac..:

Measom, Nicholas D. ; Down, Kenneth D. ; Hirst, David J....
ACS Medicinal Chemistry Letters.  8 (2016)  1 - p. 43-48 , 2016
Link: https://doi.org/10.1021/..
 
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6

Fragment-Based Approach to the Development of an Orally Bio..:

Woolford, Alison J.-A. ; Day, Philip J. ; Bénéton, Véronique...
Journal of Medicinal Chemistry.  59 (2016)  23 - p. 10738-10749 , 2016
Link: https://doi.org/10.1021/..
 
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7

Pyrazolopyridines as potent PDE4B inhibitors: 5-Heterocycle..:

Mitchell, Charlotte J. ; Ballantine, Stuart P. ; Coe, Diane M....
Bioorganic & Medicinal Chemistry Letters.  20 (2010)  19 - p. 5803-5806 , 2010
Link: https://doi.org/10.1016/..
 
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8

Identification of PDE4B Over 4D subtype-selective inhibitor..:

Kranz, Michael ; Wall, Michael ; Evans, Brian...
Bioorganic & Medicinal Chemistry.  17 (2009)  14 - p. 5336-5341 , 2009
Link: https://doi.org/10.1016/..
 
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9

Quinolines as a novel structural class of potent and select..:

Woodrow, Michael D. ; Ballantine, Stuart P. ; Barker, Michael D....
Bioorganic & Medicinal Chemistry Letters.  19 (2009)  17 - p. 5261-5265 , 2009
Link: https://doi.org/10.1016/..
 
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10

Quinolines as a novel structural class of potent and select..:

Lunniss, Christopher J. ; Cooper, Anthony W.J. ; Eldred, Colin D....
Bioorganic & Medicinal Chemistry Letters.  19 (2009)  5 - p. 1380-1385 , 2009
Link: https://doi.org/10.1016/..
 
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11

Biphenyl amide p38 kinase inhibitors 3: Improvement of cell..:

Angell, Richard ; Aston, Nicola M. ; Bamborough, Paul...
Bioorganic & Medicinal Chemistry Letters.  18 (2008)  15 - p. 4428-4432 , 2008
Link: https://doi.org/10.1016/..
 
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12

Biphenyl amide p38 kinase inhibitors 4: DFG-in and DFG-out ..:

Angell, Richard M. ; Angell, Tony D. ; Bamborough, Paul...
Bioorganic & Medicinal Chemistry Letters.  18 (2008)  15 - p. 4433-4437 , 2008
Link: https://doi.org/10.1016/..
 
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13

Biphenyl amide p38 kinase inhibitors 2: Optimisation and SA:

Angell, Richard M. ; Angell, Tony D. ; Bamborough, Paul...
Bioorganic & Medicinal Chemistry Letters.  18 (2008)  1 - p. 324-328 , 2008
Link: https://doi.org/10.1016/..
 
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14

Pyrazolopyridines as a novel structural class of potent and..:

Hamblin, J. Nicole ; Angell, Tony D.R. ; Ballantine, Stuart P....
Bioorganic & Medicinal Chemistry Letters.  18 (2008)  14 - p. 4237-4241 , 2008
Link: https://doi.org/10.1016/..
 
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15

Kinase array design, back to front: Biaryl amides:

Baldwin, Ian ; Bamborough, Paul ; Haslam, Claudine G....
Bioorganic & Medicinal Chemistry Letters.  18 (2008)  19 - p. 5285-5289 , 2008
Link: https://doi.org/10.1016/..
 
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