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Theodoulou, Natalie H.
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1

Identification and Optimization of a Ligand-Efficient Benzo..:

Humphreys, Philip G. ; Anderson, Niall A. ; Bamborough, Paul...
Journal of Medicinal Chemistry.  65 (2022)  22 - p. 15174-15207 , 2022
Link: https://doi.org/10.1021/..
 
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2

Optimization of Naphthyridones into Selective TATA-Binding ..:

Clegg, Michael A. ; Theodoulou, Natalie H. ; Bamborough, Paul...
ACS Medicinal Chemistry Letters.  12 (2021)  8 - p. 1308-1317 , 2021
Link: https://doi.org/10.1021/..
 
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3

Application of Atypical Acetyl-lysine Methyl Mimetics in th..:

Clegg, Michael A. ; Bamborough, Paul ; Chung, Chun-wa...
Journal of Medicinal Chemistry.  63 (2020)  11 - p. 5816-5840 , 2020
Link: https://doi.org/10.1021/..
 
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4

Clinical progress and pharmacology of small molecule bromod..:

Theodoulou, Natalie H ; Tomkinson, Nicholas CO ; Prinjha, Rab K.
Current Opinion in Chemical Biology.  33 (2016)  - p. 58-66 , 2016
Link: https://doi.org/10.1016/..
 
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5

Isoxazole‐Derived Amino Acids are Bromodomain‐Binding Acety..:

Sekirnik (née Measures), Angelina R. ; Hewings, David S. ; Theodoulou, Natalie H....
Angewandte Chemie International Edition.  55 (2016)  29 - p. 8353-8357 , 2016
Link: https://doi.org/10.1002/..
 
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6

Progress in the Development of non‐BET Bromodomain Chemical..:

Theodoulou, Natalie H. ; Tomkinson, Nicholas C. O. ; Prinjha, Rab K..
ChemMedChem.  11 (2016)  5 - p. 477-487 , 2016
Link: https://doi.org/10.1002/..
 
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7

Isoxazole‐Derived Amino Acids are Bromodomain‐Binding Acety..:

Sekirnik (née Measures), Angelina R. ; Hewings, David S. ; Theodoulou, Natalie H....
Angewandte Chemie.  128 (2016)  29 - p. 8493-8497 , 2016
Link: https://doi.org/10.1002/..
 
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8

Discovery of I-BRD9, a Selective Cell Active Chemical Probe..:

Theodoulou, Natalie H. ; Bamborough, Paul ; Bannister, Andrew J....
Journal of Medicinal Chemistry.  59 (2015)  4 - p. 1425-1439 , 2015
Link: https://doi.org/10.1021/..
 
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9

Alkene anti-Dihydroxylation with Malonoyl Peroxides:

Alamillo-Ferrer, Carla ; Davidson, Stuart C. ; Rawling, Michael J....
Organic Letters.  17 (2015)  20 - p. 5132-5135 , 2015
Link: https://doi.org/10.1021/..
 
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10

Clinical progress and pharmacology of small molecule bromod..:

Theodoulou, Natalie H ; Tomkinson, Nicholas CO ; Prinjha, Rab K.
https://strathprints.strath.ac.uk/57069/1/Theodoulou_etal_COCB2016_Small_molecule_bromodomain_inhibitors.pdf.  , 2016
Link: https://strathprints.str..
 
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11

Discovery of I-BRD9, a selective cell active chemical probe..:

Theodoulou, Natalie H ; Bamborough, Paul ; Bannister, Andrew J...
Theodoulou , N H , Bamborough , P , Bannister , A J , Becher , I , Bit , R A , Che , K H , Chung , C , Dittmann , A , Drewes , G , Drewry , D H , Gordon , L , Grandi , P , Leveridge , M , Lindon , M , Michon , A-M , Molnar , J , Robson , S C , Tomkinson , N C O , Kouzarides , T , Prinjha , R K & Humphreys , P G 2016 , ' Discovery of I-BRD9, a selective cell active chemical probe for bromodomain containing protein 9 inhibition ' Journal of Medicinal Chemistry , vol 59 , no. 4 , pp. 1425-1439 . DOI:10.1021/acs.jmedchem.5b00256.  , 2016
Link: https://doi.org/10.1021/..
 
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12

Isoxazole-Derived Amino Acids are Bromodomain-Binding Acety..:

Sekirnik Née Measures, Angelina R ; Hewings, David S ; Theodoulou, Natalie H...
https://www.repository.cam.ac.uk/handle/1810/316518.  , 2016
Link: https://www.repository.c..
 
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13

The discovery of I-BRD9, a selective cell active chemical p..:

Theodoulou, Natalie H ; Bamborough, Paul ; Bannister, Andrew J...
https://strathprints.strath.ac.uk/56423/1/Open_Access_Reprint.pdf.  , 2016
Link: https://strathprints.str..
 
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14

Optimization of Naphthyridones into Selective TATA-Binding ..:

Michael A. Clegg (8907155) ; Natalie H. Theodoulou (1508650) ; Paul Bamborough (1343466)...
https://figshare.com/articles/journal_contribution/Optimization_of_Naphthyridones_into_Selective_TATA-Binding_Protein_Associated_Factor_1_TAF1_Bromodomain_Inhibitors/15097571.  , 2021
Link: https://doi.org/10.1021/..
 
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15

Design, Synthesis, and Characterization of I‑BET567, a Pan-..:

Philip G. Humphreys (1357530) ; Stephen J. Atkinson (1297362) ; Paul Bamborough (1343466)...
https://figshare.com/articles/dataset/Design_Synthesis_and_Characterization_of_I_BET567_a_Pan-Bromodomain_and_Extra_Terminal_BET_Bromodomain_Oral_Candidate/18064459.  , 1753
Link: https://doi.org/10.1021/..
 
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