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1
A novel pan-selective bromodomain inhibitor for epigenetic ..:
Warstat, Robin ; Pervaiz, Mehrosh ; Regenass, Pierre...
European Journal of Medicinal Chemistry. 249 (2023) - p. 115139 , 2023
European Journal of Medicinal Chemistry. 249 (2023) - p. 115139 , 2023
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2
C–H arylation enables synthesis of imidazole-4-carboxamide ..:
Ueda, Ayaka ; Amaike, Kazuma ; Shirotani, Yoko...
Canadian Journal of Chemistry. 101 (2023) 7 - p. 449-452 , 2023
Canadian Journal of Chemistry. 101 (2023) 7 - p. 449-452 , 2023
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3
4-Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Schäker-Hübner, Linda ; Warstat, Robin ; Ahlert, Heinz...
Journal of Medicinal Chemistry. 64 (2021) 19 - p. 14620-14646 , 2021
Journal of Medicinal Chemistry. 64 (2021) 19 - p. 14620-14646 , 2021
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4
4-Acyl Pyrroles as Dual BET-BRD7/9 Bromodomain Inhibitors A..:
Hügle, Martin ; Regenass, Pierre ; Warstat, Robin...
Journal of Medicinal Chemistry. 63 (2020) 24 - p. 15603-15620 , 2020
Journal of Medicinal Chemistry. 63 (2020) 24 - p. 15603-15620 , 2020
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5
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694476. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694476. , 2021
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6
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694518. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694518. , 2021
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7
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694488. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694488. , 2021
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8
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/journal_contribution/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694467. , 2021
https://figshare.com/articles/journal_contribution/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694467. , 2021
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9
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694530. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694530. , 2021
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10
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694512. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694512. , 2021
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11
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694506. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694506. , 2021
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12
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694491. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694491. , 2021
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13
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694482. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694482. , 2021
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14
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694500. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694500. , 2021
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15
4‑Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for H..:
Linda Schäker-Hübner (8134662) ; Robin Warstat (9732506) ; Heinz Ahlert (4831686)...
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694494. , 2021
https://figshare.com/articles/dataset/4_Acyl_Pyrrole_Capped_HDAC_Inhibitors_A_New_Scaffold_for_Hybrid_Inhibitors_of_BET_Proteins_and_Histone_Deacetylases_as_Antileukemia_Drug_Leads/16694494. , 2021