E-LIB Suche - Ergebnisse für: Waszkowycz, Bohdan

1

Discovery and Optimization of wt-RET/KDR-Selective Inhibito..:

Newton, Rebecca ; Waszkowycz, Bohdan ; Seewooruthun, Chitra...
ACS Medicinal Chemistry Letters. 11 (2020) 4 - p. 497-505 , 2020

Link: https://doi.org/10.1021/..

2

Enhancer Activation by Pharmacologic Displacement of LSD1 f..:

Maiques-Diaz, Alba ; Spencer, Gary J. ; Lynch, James T....
Cell Reports. 22 (2018) 13 - p. 3641-3659 , 2018

Link: https://doi.org/10.1016/..

3

Cell-Active Small Molecule Inhibitors of the DNA-Damage Rep..:

Waszkowycz, Bohdan ; Smith, Kate M. ; McGonagle, Alison E....
Journal of Medicinal Chemistry. 61 (2018) 23 - p. 10767-10792 , 2018

Link: https://doi.org/10.1021/..

4

Discovery and Optimization of Allosteric Inhibitors of Muta..:

Jones, Stuart ; Ahmet, Jonathan ; Ayton, Kelly...
Journal of Medicinal Chemistry. 59 (2016) 24 - p. 11120-11137 , 2016

Link: https://doi.org/10.1021/..

5

Identification of selective inhibitors of RET and compariso..:

Watson, Amanda J. ; Hopkins, Gemma V. ; Hitchin, Samantha...
F1000Research. 5 (2016) - p. 1005 , 2016

Link: https://doi.org/10.12688..

6

Identification of selective inhibitors of RET and compariso..:

Watson, Amanda J. ; Hopkins, Gemma V. ; Hitchin, Samantha...
F1000Research. 5 (2016) - p. 1005 , 2016

Link: https://doi.org/10.12688..

7

First-in-Class Chemical Probes against Poly(ADP-ribose) Gly..:

James, Dominic I. ; Smith, Kate M. ; Jordan, Allan M....
ACS Chemical Biology. 11 (2016) 11 - p. 3179-3190 , 2016

Link: https://doi.org/10.1021/..

8

The discovery of 2-substituted phenol quinazolines as poten..:

Newton, Rebecca ; Bowler, Katherine A. ; Burns, Emily M....
European Journal of Medicinal Chemistry. 112 (2016) - p. 20-32 , 2016

Link: https://doi.org/10.1016/..

9

Anilinoquinazoline inhibitors of the RET kinase domain—Elab..:

Jordan, Allan M. ; Begum, Habiba ; Fairweather, Emma...
Bioorganic & Medicinal Chemistry Letters. 26 (2016) 11 - p. 2724-2729 , 2016

Link: https://doi.org/10.1016/..

10

Application of virtual screening to the discovery of novel ..:

Clark, David E. ; Waszkowycz, Bohdan ; Wong, Melanie...
Bioorganic & Medicinal Chemistry Letters. 26 (2016) 12 - p. 2920-2926 , 2016

Link: https://doi.org/10.1016/..

11

A reversed sulfonamide series of selective RORc inverse ago..:

van Niel, Monique B. ; Fauber, Benjamin P. ; Cartwright, Matthew...
Bioorganic & Medicinal Chemistry Letters. 24 (2014) 24 - p. 5769-5776 , 2014

Link: https://doi.org/10.1016/..

12

Inhibiting NF-κB-inducing kinase (NIK): Discovery, structur..:

Li, Kexue ; McGee, Lawrence R. ; Fisher, Ben...
Bioorganic & Medicinal Chemistry Letters. 23 (2013) 5 - p. 1238-1244 , 2013

Link: https://doi.org/10.1016/..

13

Toxoflavins and Deazaflavins as the First Reported Selectiv..:

Raoof, Ali ; Depledge, Paul ; Hamilton, Niall M....
Journal of Medicinal Chemistry. 56 (2013) 16 - p. 6352-6370 , 2013

Link: https://doi.org/10.1021/..

14

Targeted genetic dependency screen facilitates identificati..:

Fawdar, Shameem ; Trotter, Eleanor W. ; Li, Yaoyong...
Proceedings of the National Academy of Sciences. 110 (2013) 30 - p. 12426-12431 , 2013

Link: https://doi.org/10.1073/..

15

Protein Kinase Cδ Deficiency Causes Mendelian Systemic Lupu..:

Belot, Alexandre ; Kasher, Paul R. ; Trotter, Eleanor W....
Arthritis & Rheumatism. 65 (2013) 8 - p. 2161-2171 , 2013

Link: https://doi.org/10.1002/..