E-LIB Suche - Ergebnisse für: van Veldhoven, Jacobus P. D.

1

Label-free detection of prostaglandin transporter (SLCO2A1)..:

Mocking, Tamara A. M. ; van Oostveen, Wieke M. ; van Veldhoven, Jacobus P. D....
Frontiers in Pharmacology. 15 (2024) - p. , 2024

Link: https://doi.org/10.3389/..

2

Exploring novel dilazep derivatives as hENT1 inhibitors and..:

Dilweg, Majlen A. ; Gorostiola González, Marina ; de Ruiter, Martijn D....
Purinergic Signalling. , 2024

Link: https://doi.org/10.1007/..

3

Development of subtype-selective covalent ligands for the a..:

Beerkens, Bert L. H. ; Wang, Xuesong ; Avgeropoulou, Maria...
RSC Medicinal Chemistry. 13 (2022) 7 - p. 850-856 , 2022

Link: https://doi.org/10.1039/..

4

Crystal Structure and Subsequent Ligand Design of a Nonribo..:

Amelia, Tasia ; van Veldhoven, Jacobus P. D. ; Falsini, Matteo...
Journal of Medicinal Chemistry. 64 (2021) 7 - p. 3827-3842 , 2021

Link: https://doi.org/10.1021/..

5

Targeting the Kv11.1 (hERG) channel with allosteric modulat..:

van Veldhoven, Jacobus P.D. ; Campostrini, Giulia ; van Gessel, Constantijn J.E....
European Journal of Medicinal Chemistry. 212 (2021) - p. 113033 , 2021

Link: https://doi.org/10.1016/..

6

Development of Covalent Ligands for G Protein-Coupled Recep..:

Yang, Xue ; van Veldhoven, Jacobus P. D. ; Offringa, Jelle...
Journal of Medicinal Chemistry. 62 (2019) 7 - p. 3539-3552 , 2019

Link: https://doi.org/10.1021/..

7

Synthesis and Pharmacological Evaluation of Triazolopyrimid..:

Ortiz Zacarías, Natalia V. ; van Veldhoven, Jacobus P. D. ; den Hollander, Lisa S....
Journal of Medicinal Chemistry. 62 (2019) 24 - p. 11035-11053 , 2019

Link: https://doi.org/10.1021/..

8

Pyrrolone Derivatives as Intracellular Allosteric Modulator..:

Ortiz Zacarías, Natalia V. ; van Veldhoven, Jacobus P. D. ; Portner, Laura...
Journal of Medicinal Chemistry. 61 (2018) 20 - p. 9146-9161 , 2018

Link: https://doi.org/10.1021/..

9

Species differences and mechanism of action of A3 adenosine..:

Du, Lili ; Gao, Zhan-Guo ; Paoletta, Silvia...
Purinergic Signalling. 14 (2017) 1 - p. 59-71 , 2017

Link: https://doi.org/10.1007/..

10

Structure–Affinity Relationships and Structure–Kinetics Rel..:

Xia, Lizi ; Burger, Wessel A. C. ; van Veldhoven, Jacobus P. D....
Journal of Medicinal Chemistry. 60 (2017) 17 - p. 7555-7568 , 2017

Link: https://doi.org/10.1021/..

11

The role of the C-terminus of the human hydroxycarboxylic a..:

Liu, Rongfang ; van Veldhoven, Jacobus P.D. ; IJzerman, Adriaan P.
European Journal of Pharmacology. 770 (2016) - p. 70-77 , 2016

Link: https://doi.org/10.1016/..

12

Synthesis and biological evaluation of negative allosteric ..:

Yu, Zhiyi ; van Veldhoven, Jacobus P.D. ; 't Hart, Ingrid M.E....
European Journal of Medicinal Chemistry. 106 (2015) - p. 50-59 , 2015

Link: https://doi.org/10.1016/..

13

Structure–Affinity Relationships (SARs) and Structure–Kinet..:

Yu, Zhiyi ; van Veldhoven, Jacobus P. D. ; Louvel, Julien...
Journal of Medicinal Chemistry. 58 (2015) 15 - p. 5916-5929 , 2015

Link: https://doi.org/10.1021/..

14

Affinity and kinetics study of anthranilic acids as HCA2 re..:

van Veldhoven, Jacobus P.D. ; Liu, Rongfang ; Thee, Stephanie A....
Bioorganic & Medicinal Chemistry. 23 (2015) 14 - p. 4013-4025 , 2015

Link: https://doi.org/10.1016/..

15

Molecular mechanism of allosteric modulation at GPCRs: insi..:

Guo, Dong ; Venhorst, Suzanne N ; Massink, Arnault...
British Journal of Pharmacology. 171 (2014) 23 - p. 5295-5312 , 2014

Link: https://doi.org/10.1111/..