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Discovery of 2,4‑1 H ‑Imidazole Carboxamides as Potent and ..:
Johan J. N. Veerman (3034902)
;
Yorik B. Bruseker (10223438)
;
Eddy Damen (9017717)
...
https://figshare.com/articles/journal_contribution/Discovery_of_2_4_1_i_H_i_Imidazole_Carboxamides_as_Potent_and_Selective_TAK1_Inhibitors/14152940. , 2021
Link:
https://doi.org/10.1021/acsmedchemlett.0c00547.s001
RT Journal T1
Discovery of 2,4‑1 H ‑Imidazole Carboxamides as Potent and Selective TAK1 Inhibitors
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_14152940&Exemplar=1&LAN=DE A1 Johan J. N. Veerman (3034902) A1 Yorik B. Bruseker (10223438) A1 Eddy Damen (9017717) A1 Erik H. Heijne (10223441) A1 Wendy van Bruggen (10223444) A1 Koen F. W. Hekking (8042972) A1 Rob Winkel (8042969) A1 Christopher D. Hupp (2377594) A1 Anthony D. Keefe (3622769) A1 Julie Liu (6557627) A1 Heather A. Thomson (9106382) A1 Ying Zhang (40767) A1 John W. Cuozzo (1665235) A1 Andrew J. McRiner (2512648) A1 Mark J. Mulvihill (1937149) A1 Peter van Rijnsbergen (10223447) A1 Birgit Zech (10223450) A1 Louis M. Renzetti (2299315) A1 Lee Babiss (10223453) A1 Gerhard Müller (1749682) YR 2021 K1 Biochemistry K1 Medicine K1 Cell Biology K1 Pharmacology K1 Plant Biology K1 Space Science K1 Environmental Sciences not elsewhere classified K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 DECL K1 structure-based drug design K1 kinase 1 K1 DNA-encoded chemical library K1 imidazole carboxamides K1 Selective TAK 1 Inhibitors Herein K1 X-ray crystallography K1 pyrrolidine amide K1 growth factor β- K1 binding mode K1 TAK 1 inhibitors K1 potency K1 SBDD K1 dicarboxamide scaffold K1 core hinge-binding imidazole K1 kinome selectivity JF https://figshare.com/articles/journal_contribution/Discovery_of_2_4_1_i_H_i_Imidazole_Carboxamides_as_Potent_and_Selective_TAK1_Inhibitors/14152940 LK http://dx.doi.org/https://doi.org/10.1021/acsmedchemlett.0c00547.s001 DO https://doi.org/10.1021/acsmedchemlett.0c00547.s001 SF ELIB - SuUB Bremen
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