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Scaffold-Hopping Strategy on a Series of Proteasome Inhibit..:
Michael Thomas (279566)
;
Stephen Brand (798331)
;
Manu De Rycker (8377947)
...
https://figshare.com/articles/journal_contribution/Scaffold-Hopping_Strategy_on_a_Series_of_Proteasome_Inhibitors_Led_to_a_Preclinical_Candidate_for_the_Treatment_of_Visceral_Leishmaniasis/14494877. , 2021
Link:
https://doi.org/10.1021/acs.jmedchem.1c00047.s001
RT Journal T1
Scaffold-Hopping Strategy on a Series of Proteasome Inhibitors Led to a Preclinical Candidate for the Treatment of Visceral Leishmaniasis
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_14494877&Exemplar=1&LAN=DE A1 Michael Thomas (279566) A1 Stephen Brand (798331) A1 Manu De Rycker (8377947) A1 Fabio Zuccotto (1533349) A1 Iva Lukac (593803) A1 Peter G. Dodd (2143435) A1 Eun-Jung Ko (5507792) A1 Sujatha Manthri (800548) A1 Kate McGonagle (10708757) A1 Maria Osuna-Cabello (2834318) A1 Jennifer Riley (309910) A1 Caterina Pont (5959331) A1 Frederick Simeons (10708760) A1 Laste Stojanovski (1282575) A1 John Thomas (3125013) A1 Stephen Thompson (1346436) A1 Elisabet Viayna (1828396) A1 Jose M. Fiandor (2272426) A1 Julio Martin (8377944) A1 Paul G. Wyatt (473658) A1 Timothy J. Miles (2029051) A1 Kevin D. Read (165019) A1 Maria Marco (2272447) A1 Ian H. Gilbert (146934) YR 2021 K1 Biochemistry K1 Medicine K1 Pharmacology K1 Biotechnology K1 Infectious Diseases K1 Plant Biology K1 Chemical Sciences not elsewhere classified K1 Visceral Leishmaniasis K1 cryo-EM structure K1 GSK K1 impact K1 proteasome inhibition K1 candidate K1 developable compounds K1 vivo efficacy K1 scaffold-hopping exercise K1 chemistry program K1 phenotypic screen K1 VL K1 Preclinical Candidate K1 Proteasome Inhibitors K1 East Africa K1 Scaffold-Hopping Strategy K1 chemistry design JF https://figshare.com/articles/journal_contribution/Scaffold-Hopping_Strategy_on_a_Series_of_Proteasome_Inhibitors_Led_to_a_Preclinical_Candidate_for_the_Treatment_of_Visceral_Leishmaniasis/14494877 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.1c00047.s001 DO https://doi.org/10.1021/acs.jmedchem.1c00047.s001 SF ELIB - SuUB Bremen
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