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1 Ergebnisse
1
Design and Synthesis of Highly Selective Brain Penetrant p3..:
Niklas M. Tormählen (10783636)
;
Mariella Martorelli (10783639)
;
Annette Kuhn (3494771)
...
https://figshare.com/articles/dataset/Design_and_Synthesis_of_Highly_Selective_Brain_Penetrant_p38_Mitogen-Activated_Protein_Kinase_Inhibitors/14575336. , 2021
Link:
https://doi.org/10.1021/acs.jmedchem.0c01773.s002
RT Journal T1
Design and Synthesis of Highly Selective Brain Penetrant p38α Mitogen-Activated Protein Kinase Inhibitors
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_14575336&Exemplar=1&LAN=DE A1 Niklas M. Tormählen (10783636) A1 Mariella Martorelli (10783639) A1 Annette Kuhn (3494771) A1 Florian Maier (1861138) A1 Jamil Guezguez (1459330) A1 Michael Burnet (1459333) A1 Wolfgang Albrecht (2035297) A1 Stefan A. Laufer (128881) A1 Pierre Koch (560721) YR 2021 K1 Biochemistry K1 Medicine K1 Cell Biology K1 Genetics K1 Molecular Biology K1 Neuroscience K1 Physiology K1 Pharmacology K1 Biotechnology K1 Immunology K1 Infectious Diseases K1 Plant Biology K1 Virology K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 methyl ester prodrugs K1 acid transporters K1 IL -6 K1 novel Skepinone-based p 38α MAP kin K1 p 38α-MAP metabolically K1 Skepinone-N counterpart K1 5.5 nM K1 dibenzo K1 Selective Brain Penetrant p 38α Mit K1 12 nM K1 TNF -α production K1 carboxy analogs K1 difluorophenyl K1 kinase activation modulates cytokin K1 Compound 70 K1 annulene K1 cell-based assays K1 brain-to-plasma ratios K1 -3-carboxamido K1 mouse brain K1 IC K1 brain-to-plasma ratio JF https://figshare.com/articles/dataset/Design_and_Synthesis_of_Highly_Selective_Brain_Penetrant_p38_Mitogen-Activated_Protein_Kinase_Inhibitors/14575336 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.0c01773.s002 DO https://doi.org/10.1021/acs.jmedchem.0c01773.s002 SF ELIB - SuUB Bremen
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