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1 Ergebnisse
1
Discovery of the Oxadiazine FRM-024: A Potent CNS-Penetrant..:
Matthew G. Bursavich (2272390)
;
Bryce A. Harrison (1693699)
;
Raksha Acharya (3829366)
...
https://figshare.com/articles/dataset/Discovery_of_the_Oxadiazine_FRM-024_A_Potent_CNS-Penetrant_Gamma_Secretase_Modulator/16663290. , 2021
Link:
https://doi.org/10.1021/acs.jmedchem.1c00904.s002
RT Journal T1
Discovery of the Oxadiazine FRM-024: A Potent CNS-Penetrant Gamma Secretase Modulator
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_16663290&Exemplar=1&LAN=DE A1 Matthew G. Bursavich (2272390) A1 Bryce A. Harrison (1693699) A1 Raksha Acharya (3829366) A1 Donald E. Costa (3829351) A1 Emily A. Freeman (3829378) A1 Lori A. Hrdlicka (3829354) A1 Hong Jin (65601) A1 Sudarshan Kapadnis (3829360) A1 Jeffrey S. Moffit (3829372) A1 Deirdre Murphy (4595632) A1 Scott J. Nolan (2951415) A1 Holger Patzke (3829375) A1 Cuyue Tang (1443529) A1 Hilliary E. Van Voorhies (11467608) A1 Melody Wen (3829357) A1 Gerhard Koenig (3829345) A1 Jean-François Blain (3829363) A1 Duane A. Burnett (1474750) YR 2021 K1 Biochemistry K1 Medicine K1 Neuroscience K1 Pharmacology K1 Sociology K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 yl ) pyridin K1 yl )- 5 K1 gsm preclinical candidate K1 extensive preclinical profiling K1 safety studies resulted K1 improve amyloid processing K1 chlorophenyl )- 6 K1 3 -( 6 K1 previously reported oxadiazine K1 5 -( 4 K1 familial alzheimer ' K1 42 </ sub K1 alzheimer ' K1 familial form K1 efficacy studies K1 amyloid hypothesis K1 h </ K1 cis </ K1 thereby addressing K1 therapies targeting K1 recent approval K1 quality compounds K1 potent cns K1 potency improvements K1 novel compounds K1 nonhuman primates K1 >- imidazole JF https://figshare.com/articles/dataset/Discovery_of_the_Oxadiazine_FRM-024_A_Potent_CNS-Penetrant_Gamma_Secretase_Modulator/16663290 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.1c00904.s002 DO https://doi.org/10.1021/acs.jmedchem.1c00904.s002 SF ELIB - SuUB Bremen
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