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Discovery of Novel UDP‑ N ‑Acetylglucosamine Acyltransferas..:
M. Dominic Ryan (1677214)
;
Alastair L. Parkes (11485035)
;
David Corbett (324987)
...
https://figshare.com/articles/journal_contribution/Discovery_of_Novel_UDP_i_N_i_Acetylglucosamine_Acyltransferase_LpxA_Inhibitors_with_Activity_against_Pseudomonas_aeruginosa/16685472. , 2021
Link:
https://doi.org/10.1021/acs.jmedchem.1c00888.s001
RT Journal T1
Discovery of Novel UDP‑ N ‑Acetylglucosamine Acyltransferase (LpxA) Inhibitors with Activity against Pseudomonas aeruginosa
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_16685472&Exemplar=1&LAN=DE A1 M. Dominic Ryan (1677214) A1 Alastair L. Parkes (11485035) A1 David Corbett (324987) A1 Anthony P. Dickie (2882588) A1 Michelle Southey (11485038) A1 Ole A. Andersen (2114842) A1 Daniel B. Stein (1600624) A1 Olivier R. Barbeau (2241841) A1 Angelo Sanzone (2001946) A1 Pia Thommes (1833613) A1 John Barker (1677223) A1 Ricky Cain (1300071) A1 Christel Compper (527263) A1 Magali Dejob (11485041) A1 Alain Dorali (11485044) A1 Donnya Etheridge (11485047) A1 Sian Evans (7150334) A1 Adele Faulkner (1359855) A1 Elise Gadouleau (9187663) A1 Timothy Gorman (11485050) A1 Denes Haase (11485053) A1 Maisie Holbrow-Wilshaw (11485056) A1 Thomas Krulle (9187684) A1 Xianfu Li (11485059) A1 Christopher Lumley (7166261) A1 Barbara Mertins (125533) A1 Spencer Napier (2126395) A1 Rajesh Odedra (1951660) A1 Kostas Papadopoulos (9579014) A1 Vasileios Roumpelakis (11485062) A1 Kate Spear (11485065) A1 Emily Trimby (11485068) A1 Jennifer Williams (14164) A1 Michael Zahn (2062351) A1 Anthony D. Keefe (3622769) A1 Ying Zhang (40767) A1 Holly T. Soutter (11485071) A1 Paolo A. Centrella (1463083) A1 Matthew A. Clark (1370337) A1 John W. Cuozzo (1665235) A1 Christoph E. Dumelin (1272561) A1 Boer Deng (9964680) A1 Avery Hunt (11485074) A1 Eric A. Sigel (3622766) A1 Dawn M. Troast (2197303) A1 Boudewijn L. M. DeJonge (11485077) YR 2021 K1 Biochemistry K1 Medicine K1 Microbiology K1 Pharmacology K1 Cancer K1 Science Policy K1 Infectious Diseases K1 Virology K1 Environmental Sciences not elsewhere classified K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 mouse infection models K1 maximal inhibitory concentration K1 encoded compound library K1 >‑ acetylglucosamine acyltransferase K1 >- acetylglucosamine acyltransferase K1 novel udp ‑< K1 50 </ sub K1 escherichia coli lpxa K1 pseudomonas aeruginosa lpxa K1 udp -< K1 pseudomonas aeruginosa K1 n </ K1 aeruginosa lpxa K1 study describes K1 selective inhibitor K1 resistant isolates K1 ray crystallography K1 original hit K1 novel series K1 ml ) K1 mediated selection K1 genetic analyses K1 efficacy studies K1 biochemical potency K1 best half K1 5 nm K1 4 μg K1 20 μm K1 128 μg JF https://figshare.com/articles/journal_contribution/Discovery_of_Novel_UDP_i_N_i_Acetylglucosamine_Acyltransferase_LpxA_Inhibitors_with_Activity_against_Pseudomonas_aeruginosa/16685472 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.1c00888.s001 DO https://doi.org/10.1021/acs.jmedchem.1c00888.s001 SF ELIB - SuUB Bremen
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